Practical Synthesis of a S1P Receptor 1 Agonist via a Guareschi–Thorpe Reaction
Schmidt, Gunther, Bolli, Martin H, Lescop, Cyrille, Abele, Stefan
Published in Organic process research & development (16.09.2016)
Published in Organic process research & development (16.09.2016)
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Journal Article
Synthetic sphingosine 1-phosphate receptor modulators--opportunities and potential pitfalls
Bolli, Martin H, Lescop, Cyrille, Nayler, Oliver
Published in Current topics in medicinal chemistry (01.03.2011)
Published in Current topics in medicinal chemistry (01.03.2011)
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Journal Article
A New Synthesis of 2-Azabicyclo[2.1.1]hexanes
Lescop, Cyrille, Mévellec, Laurence, Huet, François
Published in Journal of organic chemistry (15.06.2001)
Published in Journal of organic chemistry (15.06.2001)
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Journal Article
Discovery of a Novel Orally Active, Selective LPA Receptor Type 1 Antagonist, 4‑(4-(2-Isopropylphenyl)-4-((2-methoxy-4-methylphenyl)carbamoyl)piperidin-1-yl)-4-oxobutanoic Acid, with a Distinct Molecular Scaffold
Lescop, Cyrille, Brotschi, Christine, Williams, Jodi T., Sager, Christoph P., Birker, Magdalena, Morrison, Keith, Froidevaux, Sylvie, Delahaye, Stéphane, Nayler, Oliver, Bolli, Martin H.
Published in Journal of medicinal chemistry (22.02.2024)
Published in Journal of medicinal chemistry (22.02.2024)
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Journal Article
Discovery of the Novel, Orally Active, and Selective LPA1 Receptor Antagonist ACT-1016-0707 as a Preclinical Candidate for the Treatment of Fibrotic Diseases
Lescop, Cyrille, Birker, Magdalena, Brotschi, Christine, Bürki, Cédric, Morrison, Keith, Froidevaux, Sylvie, Delahaye, Stéphane, Nayler, Oliver, Bolli, Martin H.
Published in Journal of medicinal chemistry (22.02.2024)
Published in Journal of medicinal chemistry (22.02.2024)
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Journal Article
S1P1 Modulator-Induced G αi Signaling and β-Arrestin Recruitment Are Both Necessary to Induce Rapid and Efficient Reduction of Blood Lymphocyte Count In Vivo
Birker-Robaczewska, Magdalena, Bolli, Martin, Rey, Markus, de Kanter, Ruben, Kohl, Christopher, Lescop, Cyrille, Boucher, Maxime, Poirey, Sylvie, Steiner, Beat, Nayler, Oliver
Published in Molecular pharmacology (01.02.2018)
Published in Molecular pharmacology (01.02.2018)
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Journal Article
Novel S1P(1) receptor agonists - Part 5: From amino-to alkoxy-pyridines
Bolli, Martin H., Lescop, Cyrille, Birker, Magdalena, de Kanter, Ruben, Hess, Patrick, Kohl, Christopher, Nayler, Oliver, Rey, Markus, Sieber, Patrick, Velker, Jorg, Weller, Thomas, Steiner, Beat
Published in European journal of medicinal chemistry (10.06.2016)
Published in European journal of medicinal chemistry (10.06.2016)
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Journal Article
S1P 1 Modulator-Induced G α i Signaling and β -Arrestin Recruitment Are Both Necessary to Induce Rapid and Efficient Reduction of Blood Lymphocyte Count In Vivo
Birker-Robaczewska, Magdalena, Bolli, Martin, Rey, Markus, de Kanter, Ruben, Kohl, Christopher, Lescop, Cyrille, Boucher, Maxime, Poirey, Sylvie, Steiner, Beat, Nayler, Oliver
Published in Molecular pharmacology (01.02.2018)
Published in Molecular pharmacology (01.02.2018)
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Journal Article
Novel S1P(1) receptor agonists - Part 4: Alkylaminomethyl substituted aryl head groups
Lescop, Cyrille, Muller, Claus, Mathys, Boris, Birker, Magdalena, de Kanter, Ruben, Kohl, Christopher, Hess, Patrick, Nayler, Oliver, Rey, Markus, Sieber, Patrick, Steiner, Beat, Weller, Thomas, Bolli, Martin H.
Published in European journal of medicinal chemistry (30.06.2016)
Published in European journal of medicinal chemistry (30.06.2016)
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Journal Article
Substituted Cyclobutenes, Their Preparation, and Their Versatility in Synthesis
Gauvry, Noëlle, Lescop, Cyrille, Huet, François
Published in European Journal of Organic Chemistry (01.12.2006)
Published in European Journal of Organic Chemistry (01.12.2006)
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Journal Article
Novel S1P1 receptor agonists – Part 5: From amino-to alkoxy-pyridines
Bolli, Martin H., Lescop, Cyrille, Birker, Magdalena, de Kanter, Ruben, Hess, Patrick, Kohl, Christopher, Nayler, Oliver, Rey, Markus, Sieber, Patrick, Velker, Jörg, Weller, Thomas, Steiner, Beat
Published in European journal of medicinal chemistry (10.06.2016)
Published in European journal of medicinal chemistry (10.06.2016)
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Journal Article
Novel S1P 1 receptor agonists – Part 4: Alkylaminomethyl substituted aryl head groups
Lescop, Cyrille, Müller, Claus, Mathys, Boris, Birker, Magdalena, de Kanter, Ruben, Kohl, Christopher, Hess, Patrick, Nayler, Oliver, Rey, Markus, Sieber, Patrick, Steiner, Beat, Weller, Thomas, Bolli, Martin H.
Published in European journal of medicinal chemistry (01.06.2016)
Published in European journal of medicinal chemistry (01.06.2016)
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Journal Article
Novel S1P(1) Receptor Agonists - Part 3: From Thiophenes to Pyridines
Bolli, Martin H., Abele, Stefan, Birker, Magdalena, Bravo, Roberto, Bur, Daniel, de Kanter, Ruben, Kohl, Christopher, Grimont, Julien, Hess, Patrick, Lescop, Cyrille, Mathys, Boris, Mueller, Claus, Nayler, Oliver, Rey, Markus, Scherz, Michael, Schmidt, Gunther, Seifert, Juergen, Steiner, Beat, Velker, Joerg, Weller, Thomas
Published in Journal of medicinal chemistry (09.01.2014)
Published in Journal of medicinal chemistry (09.01.2014)
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Journal Article
Novel S1P1 receptor agonists – Part 4: Alkylaminomethyl substituted aryl head groups
Lescop, Cyrille, Müller, Claus, Mathys, Boris, Birker, Magdalena, de Kanter, Ruben, Kohl, Christopher, Hess, Patrick, Nayler, Oliver, Rey, Markus, Sieber, Patrick, Steiner, Beat, Weller, Thomas, Bolli, Martin H.
Published in European journal of medicinal chemistry (30.06.2016)
Published in European journal of medicinal chemistry (30.06.2016)
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Journal Article
Cenerimod, a novel selective S1P1 receptor modulator with unique signaling properties
Piali, Luca, Birker‐Robaczewska, Magdalena, Lescop, Cyrille, Froidevaux, Sylvie, Schmitz, Nicole, Morrison, Keith, Kohl, Christopher, Rey, Markus, Studer, Rolf, Vezzali, Enrico, Hess, Patrick, Clozel, Martine, Steiner, Beat, Bolli, Martin H., Nayler, Oliver
Published in Pharmacology research & perspectives (01.12.2017)
Published in Pharmacology research & perspectives (01.12.2017)
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Journal Article
Novel S1P1 Receptor Agonists − Part 3: From Thiophenes to Pyridines
Bolli, Martin H, Abele, Stefan, Birker, Magdalena, Bravo, Roberto, Bur, Daniel, de Kanter, Ruben, Kohl, Christopher, Grimont, Julien, Hess, Patrick, Lescop, Cyrille, Mathys, Boris, Müller, Claus, Nayler, Oliver, Rey, Markus, Scherz, Michael, Schmidt, Gunther, Seifert, Jürgen, Steiner, Beat, Velker, Jörg, Weller, Thomas
Published in Journal of medicinal chemistry (09.01.2014)
Published in Journal of medicinal chemistry (09.01.2014)
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Journal Article