Differential protein acetylation induced by novel histone deacetylase inhibitors
Glaser, K.B., Li, J., Pease, L.J., Staver, M.J., Marcotte, P.A., Guo, J., Frey, R.R., Garland, R.B., Heyman, H.R., Wada, C.K., Vasudevan, A., Michaelides, M.R., Davidsen, S.K., Curtin, M.L.
Published in Biochemical and biophysical research communications (17.12.2004)
Published in Biochemical and biophysical research communications (17.12.2004)
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Journal Article
Thienopyrimidine Ureas as Novel and Potent Multitargeted Receptor Tyrosine Kinase Inhibitors
Dai, Yujia, Guo, Yan, Frey, Robin R, Ji, Zhiqin, Curtin, Michael L, Ahmed, Asma A, Albert, Daniel H, Arnold, Lee, Arries, Shannon S, Barlozzari, Teresa, Bauch, Joy L, Bouska, Jennifer J, Bousquet, Peter F, Cunha, George A, Glaser, Keith B, Guo, Jun, Li, Junling, Marcotte, Patrick A, Marsh, Kennan C, Moskey, Maria D, Pease, Lori J, Stewart, Kent D, Stoll, Vincent S, Tapang, Paul, Wishart, Neil, Davidsen, Steven K, Michaelides, Michael R
Published in Journal of medicinal chemistry (22.09.2005)
Published in Journal of medicinal chemistry (22.09.2005)
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Journal Article
The design, synthesis, and structure-activity relationships of a series of macrocyclic MMP inhibitors
Steinman, Douglas H., Curtin, Michael L., Garland, Robert B., Davidsen, Steven K., Heyman, H.Robin, Holms, James H., Albert, Daniel H., Magoc, Terry J., Nagy, Ildiko B., Marcotte, Patrick A., Li, Junling, Morgan, Douglas W., Hutchins, Charles, Summers, James B.
Published in Bioorganic & medicinal chemistry letters (18.08.1998)
Published in Bioorganic & medicinal chemistry letters (18.08.1998)
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Journal Article
Phenoxyphenyl Sulfone N-Formylhydroxylamines (Retrohydroxamates) as Potent, Selective, Orally Bioavailable Matrix Metalloproteinase Inhibitors
Wada, Carol K, Holms, James H, Curtin, Michael L, Dai, Yujia, Florjancic, Alan S, Garland, Robert B, Guo, Yan, Heyman, H. Robin, Stacey, Jamie R, Steinman, Douglas H, Albert, Daniel H, Bouska, Jennifer J, Elmore, Ildiko N, Goodfellow, Carole L, Marcotte, Patrick A, Tapang, Paul, Morgan, Douglas W, Michaelides, Michael R, Davidsen, Steven K
Published in Journal of medicinal chemistry (03.01.2002)
Published in Journal of medicinal chemistry (03.01.2002)
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Journal Article
ABT-491, a highly potent and selective PAF antagonist, inhibits nasal vascular permeability associated with experimental allergic rhinitis in brown Norway rats
Albert, D H, Tapang, P, Morgan, D W, Curtin, M L, Sheppard, G S, Davidsen, S K, Summers, J B, Carter, G W
Published in Inflammation research (01.08.1997)
Published in Inflammation research (01.08.1997)
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Journal Article
Biaryl Ether Retrohydroxamates as Potent, Long-lived, Orally Bioavailable MMP Inhibitors
Michaelides, Michael R., Dellaria, Joseph F., Gong, Jane, Holms, James H., Bouska, Jennifer J., Stacey, Jamie, Wada, Carol K., Heyman, H.Robin, Curtin, Michael L., Guo, Yan, Goodfellow, Carole L., Elmore, Ildiko B., Albert, Daniel H., Magoc, Terrance J., Marcotte, Patrick A., Morgan, Douglas W., Davidsen, Steven K.
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
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Journal Article
Discovery and characterization of the potent, selective and orally bioavailable MMP inhibitor ABT-770
Curtin, Michael L., Florjancic, Alan S., Heyman, H.Robin, Michaelides, Michael R., Garland, Robert B., Holms, James H., Steinman, Douglas H., Dellaria, Joseph F., Gong, Jane, Wada, Carol K., Guo, Yan, Elmore, Ildiko B., Tapang, Paul, Albert, Daniel H., Magoc, Terrance J., Marcotte, Patrick A., Bouska, Jennifer J., Goodfellow, Carole L., Bauch, Joy L., Marsh, Kennan C., Morgan, Douglas W., Davidsen, Steven K.
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
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Journal Article
Broad spectrum matrix metalloproteinase inhibitors : An examination of succinamide hydroxamate inhibitors with p1 Cα gem-disubstitution
CURTIN, M. L, GARLAND, R. B, DAVIDSEN, S. K, MARCOTTE, P. A, ALBERT, D. H, MAGOC, T. J, HUTCHINS, C
Published in Bioorganic & medicinal chemistry letters (16.06.1998)
Published in Bioorganic & medicinal chemistry letters (16.06.1998)
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Journal Article
The Role of Platelet-Activating Factor (PAF) and the Efficacy of ABT-491, a Highly Potent and Selective PAF Antagonist, in Experimental Allergic Rhinitis
Albert, D H, Malo, P E, Tapang, P, Shaughnessy, T K, Morgan, D W, Wegner, C D, Curtin, M L, Sheppard, G S, Xu, L, Davidsen, S K, Summers, J B, Carter, G W
Published in The Journal of pharmacology and experimental therapeutics (01.01.1998)
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Published in The Journal of pharmacology and experimental therapeutics (01.01.1998)
Journal Article
Evaluation of the Inhibition of other Metalloproteinases by Matrix Metalloproteinase Inhibitors
Marcotte, Patrick A., Elmore, Ildiko N., Guan, Zhiwen, Magoc, Terrance J., Albert, Daniel H., Morgan, Douglas W., Curtin, Michael L., Garland, Robert B., Guo, Yan, Heyman, H. Robin, Holms, James H., Sheppard, George S., Steinman, Douglas H., Wada, Carol K., Davidsen, Steven K.
Published in Journal of enzyme inhibition (01.01.1999)
Published in Journal of enzyme inhibition (01.01.1999)
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Journal Article
Novel reactions of 1-triptycylcarbinols with thionyl chloride-dimethylformamide
Crumrine, David S, Curtin, Michael L, Iwamura, Hiizu
Published in Journal of organic chemistry (01.02.1990)
Published in Journal of organic chemistry (01.02.1990)
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Journal Article
Studies on the synthesis of nargenicin A(1): Highly stereoselective synthesis of the complete carbon framework via the transannular Diels-Alder reaction of an 18-membered macrolide
Roush, WR, Koyama, K, Curtin, ML, Moriarty, KJ
Published in Journal of the American Chemical Society (14.08.1996)
Published in Journal of the American Chemical Society (14.08.1996)
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Journal Article
Trifluoromethyl ketones as inhibitors of histone deacetylase
Frey, Robin R., Wada, Carol K., Garland, Robert B., Curtin, Michael L., Michaelides, Michael R., Li, Junling, Pease, Lori J., Glaser, Keith B., Marcotte, Patrick A., Bouska, Jennifer J., Murphy, Shannon S., Davidsen, Steven K.
Published in Bioorganic & medicinal chemistry letters (02.12.2002)
Published in Bioorganic & medicinal chemistry letters (02.12.2002)
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Journal Article
Succinimide hydroxamic acids as potent inhibitors of histone deacetylase (HDAC)
CURTIN, Michael L, GARLAND, Robert B, HEYMAN, H. Robin, FREY, Robin R, MICHAELIDES, Michael R, JUNLING LI, PEASE, Lori J, GLASER, Keith B, MARCOTTE, Patrick A, DAVIDSEN, Steven K
Published in Bioorganic & medicinal chemistry letters (21.10.2002)
Published in Bioorganic & medicinal chemistry letters (21.10.2002)
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Journal Article
α-Keto amides as inhibitors of histone deacetylase
Wada, Carol K., Frey, Robin R., Ji, Zhiqin, Curtin, Michael L., Garland, Robert B., Holms, James H., Li, Junling, Pease, Lori J., Guo, Jun, Glaser, Keith B., Marcotte, Patrick A., Richardson, Paul L., Murphy, Shannon S., Bouska, Jennifer J., Tapang, Paul, Magoc, Terrance J., Albert, Daniel H., Davidsen, Steven K., Michaelides, Michael R.
Published in Bioorganic & medicinal chemistry letters (06.10.2003)
Published in Bioorganic & medicinal chemistry letters (06.10.2003)
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Journal Article
Expression and functional characterization of recombinant human HDAC1 and HDAC3
Li, Junling, Staver, Michael J, Curtin, Michael L, Holms, James H, Frey, Robin R, Edalji, Rohinton, Smith, Richard, Michaelides, Mike R, Davidsen, Steven K, Glaser, Keith B
Published in Life sciences (1973) (16.04.2004)
Published in Life sciences (1973) (16.04.2004)
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Journal Article
Heterocyclic ketones as inhibitors of histone deacetylase
Vasudevan, Anil, Ji, Zhiqin, Frey, Robin R., Wada, Carol K., Steinman, Douglas, Heyman, H.Robin, Guo, Yan, Curtin, Michael L., Guo, Jun, Li, Junling, Pease, Lori, Glaser, Keith B., Marcotte, Patrick A., Bouska, Jennifer J., Davidsen, Steven K., Michaelides, Michael R.
Published in Bioorganic & medicinal chemistry letters (17.11.2003)
Published in Bioorganic & medicinal chemistry letters (17.11.2003)
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Journal Article
Isoindolinone ureas: a novel class of KDR kinase inhibitors
Curtin, Michael L, Frey, Robin R, Heyman, H.Robin, Sarris, Kathy A, Steinman, Douglas H, Holmes, James H, Bousquet, Peter F, Cunha, George A, Moskey, Maria D, Ahmed, Asma A, Pease, Lori J, Glaser, Keith B, Stewart, Kent D, Davidsen, Steven K, Michaelides, Michael R
Published in Bioorganic & medicinal chemistry letters (06.09.2004)
Published in Bioorganic & medicinal chemistry letters (06.09.2004)
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Journal Article