Future challenges facing the development of specific active-site-directed synthetic inhibitors of MMPs
Cuniasse, P., Devel, L., Makaritis, A., Beau, F., Georgiadis, D., Matziari, M., Yiotakis, A., Dive, V.
Published in Biochimie (01.03.2005)
Published in Biochimie (01.03.2005)
Get full text
Journal Article
Phosphinic peptides as zinc metalloproteinase inhibitors
Dive, V, Georgiadis, D, Matziari, M, Makaritis, A, Beau, F, Cuniasse, P, Yiotakis, A
Published in Cellular and molecular life sciences : CMLS (01.08.2004)
Published in Cellular and molecular life sciences : CMLS (01.08.2004)
Get full text
Journal Article
Signatures of Lévy flights with annealed disorder
Baudouin, Q, Pierrat, R, Eloy, A, Nunes-Pereira, E J, Cuniasse, P-A, Mercadier, N, Kaiser, R
Published in Physical review. E, Statistical, nonlinear, and soft matter physics (01.11.2014)
Published in Physical review. E, Statistical, nonlinear, and soft matter physics (01.11.2014)
Get more information
Journal Article
Structure-Based Secondary Structure-Independent Approach To Design Protein Ligands: Application to the Design of Kv1.2 Potassium Channel Blockers
Magis, C, Gasparini, D, Lecoq, A, Le Du, M. H, Stura, E, Charbonnier, J. B, Mourier, G, Boulain, J.-C, Pardo, L, Caruana, A, Joly, A, Lefranc, M, Masella, M, Menez, A, Cuniasse, P
Published in Journal of the American Chemical Society (20.12.2006)
Published in Journal of the American Chemical Society (20.12.2006)
Get full text
Journal Article
Development of Selective Inhibitors and Substrate of Matrix Metalloproteinase-12
Devel, Laurent, Rogakos, Vassilis, David, Arnaud, Makaritis, Anastasios, Beau, Fabrice, Cuniasse, Philippe, Yiotakis, Athanasios, Dive, Vincent
Published in The Journal of biological chemistry (21.04.2006)
Published in The Journal of biological chemistry (21.04.2006)
Get full text
Journal Article
Evaluation of P-1'-diversified phosphinic peptides leads to the development of highly selective inhibitors of MMP-11
Matziari, M, Beau, F, Cuniasse, P, Dive, Yiotakis, A
Published in Journal of medicinal chemistry (15.01.2004)
Published in Journal of medicinal chemistry (15.01.2004)
Get full text
Journal Article
Abasic frameshift in DNA. Solution conformation determined by proton NMR and molecular mechanics calculations
Cuniasse, P, Sowers, L. C, Eritja, R, Kaplan, B, Goodman, M. F, Cognet, J. A. H, Le Bret, M, Guschlbauer, W, Fazakerley, G. V
Published in Biochemistry (Easton) (07.03.1989)
Published in Biochemistry (Easton) (07.03.1989)
Get full text
Journal Article
Residues Determining the Binding Specificity of Uncompetitive Inhibitors to Tissue‐Nonspecific Alkaline Phosphatase
Kozlenkov, Alexey, Le Du, Marie Helene, Cuniasse, Philippe, Ny, Tor, Hoylaerts, Marc F, Millán, José Luis
Published in Journal of bone and mineral research (01.11.2004)
Published in Journal of bone and mineral research (01.11.2004)
Get full text
Journal Article
RXP 407, a Phosphinic Peptide, Is a Potent Inhibitor of Angiotensin I Converting Enzyme Able to Differentiate between Its Two Active Sites
Dive, Vincent, Cotton, Joël, Yiotakis, Athanasios, Michaud, Annie, Vassiliou, Stamatia, Jiracek, Jiri, Vazeux, Gilles, Chauvet, Marie-Thérèse, Cuniasse, Philippe, Corvol, Pierre
Published in Proceedings of the National Academy of Sciences - PNAS (13.04.1999)
Published in Proceedings of the National Academy of Sciences - PNAS (13.04.1999)
Get full text
Journal Article
Selective Inhibition of the C-Domain of Angiotensin I Converting Enzyme by Bradykinin Potentiating Peptides
Cotton, Joël, Hayashi, Mirian A. F, Cuniasse, Philippe, Vazeux, Gilles, Ianzer, Danielle, De Camargo, Antonio C. M, Dive, Vincent
Published in Biochemistry (Easton) (14.05.2002)
Published in Biochemistry (Easton) (14.05.2002)
Get full text
Journal Article
Crystal structure of the stromelysin-3 (MMP-11) catalytic domain complexed with a phosphinic inhibitor mimicking the transition-state
Gall, Anne-Laure, Ruff, Marc, Kannan, Rama, Cuniasse, Philippe, Yiotakis, Athanasios, Dive, Vincent, Rio, Marie-Christine, Basset, Paul, Moras, Dino
Published in Journal of molecular biology (23.03.2001)
Published in Journal of molecular biology (23.03.2001)
Get full text
Journal Article
Combined use of selective inhibitors and fluorogenic substrates to study the specificity of somatic wild‐type angiotensin‐converting enzyme
Jullien, Nicolas D., Cuniasse, Philippe, Georgiadis, Dimitris, Yiotakis, Athanasios, Dive, Vincent
Published in The FEBS journal (01.04.2006)
Published in The FEBS journal (01.04.2006)
Get full text
Journal Article
Phosphinic Pseudo-Tripeptides as Potent Inhibitors of Matrix Metalloproteinases: A Structure−Activity Study
Vassiliou, Stamatia, Mucha, Artur, Cuniasse, Philippe, Georgiadis, Dimitris, Lucet-Levannier, Karine, Beau, Fabrice, Kannan, Rama, Murphy, Gillian, Knäuper, Vera, Rio, Marie-Christine, Basset, Paul, Yiotakis, Athanasios, Dive, Vincent
Published in Journal of medicinal chemistry (15.07.1999)
Published in Journal of medicinal chemistry (15.07.1999)
Get full text
Journal Article
Membrane type-1 matrix metalloprotease and stromelysin-3 cleave more efficiently synthetic substrates containing unusual amino acids in their P1' positions
Mucha, A, Cuniasse, P, Kannan, R, Beau, F, Yiotakis, A, Basset, P, Dive, V
Published in The Journal of biological chemistry (30.01.1998)
Published in The Journal of biological chemistry (30.01.1998)
Get full text
Journal Article
Potency and selectivity of RXP407 on human, rat, and mouse angiotensin-converting enzyme
Vazeux, Gille, Cotton, Joël, Cuniasse, Philippe, Dive, Vincent
Published in Biochemical pharmacology (01.04.2001)
Published in Biochemical pharmacology (01.04.2001)
Get full text
Journal Article
Accounting for Conformational Variability in NMR Structure of Cyclopeptides: Ensemble Averaging of Interproton Distance and Coupling Constant Restraints
Cuniasse, Philippe, Raynal, Isabelle, Yiotakis, Athanosios, Dive, Vincent
Published in Journal of the American Chemical Society (04.06.1997)
Published in Journal of the American Chemical Society (04.06.1997)
Get full text
Journal Article
Role of the S1‘ Subsite Glutamine 215 in Activity and Specificity of Stromelysin-3 by Site-Directed Mutagenesis
Holtz, Béatrice, Cuniasse, Philippe, Boulay, Anne, Kannan, Rama, Mucha, Artur, Beau, Fabrice, Basset, Paul, Dive, Vincent
Published in Biochemistry (Easton) (14.09.1999)
Published in Biochemistry (Easton) (14.09.1999)
Get full text
Journal Article