Recent Developments in PROTAC‐Mediated Protein Degradation: From Bench to Clinic
Hu, Zhenyi, Crews, Craig M.
Published in Chembiochem : a European journal of chemical biology (19.01.2022)
Published in Chembiochem : a European journal of chemical biology (19.01.2022)
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Journal Article
Waste disposal—An attractive strategy for cancer therapy
Salami, Jemilat, Crews, Craig M.
Published in Science (American Association for the Advancement of Science) (17.03.2017)
Published in Science (American Association for the Advancement of Science) (17.03.2017)
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Journal Article
MDM2-Recruiting PROTAC Offers Superior, Synergistic Antiproliferative Activity via Simultaneous Degradation of BRD4 and Stabilization of p53
Hines, John, Lartigue, Schan, Dong, Hanqing, Qian, Yimin, Crews, Craig M
Published in Cancer research (Chicago, Ill.) (01.01.2019)
Published in Cancer research (Chicago, Ill.) (01.01.2019)
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Journal Article
Targeted Protein Degradation by Small Molecules
Bondeson, Daniel P, Crews, Craig M
Published in Annual review of pharmacology and toxicology (06.01.2017)
Published in Annual review of pharmacology and toxicology (06.01.2017)
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Journal Article
Differential PROTAC substrate specificity dictated by orientation of recruited E3 ligase
Smith, Blake E, Wang, Stephen L, Jaime-Figueroa, Saul, Harbin, Alicia, Wang, Jing, Hamman, Brian D, Crews, Craig M
Published in Nature communications (10.01.2019)
Published in Nature communications (10.01.2019)
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Journal Article
Modular PROTAC Design for the Degradation of Oncogenic BCR-ABL
Lai, Ashton C., Toure, Momar, Hellerschmied, Doris, Salami, Jemilat, Jaime-Figueroa, Saul, Ko, Eunhwa, Hines, John, Crews, Craig M.
Published in Angewandte Chemie (International ed.) (11.01.2016)
Published in Angewandte Chemie (International ed.) (11.01.2016)
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Journal Article
Targeting the C481S Ibrutinib-Resistance Mutation in Bruton’s Tyrosine Kinase Using PROTAC-Mediated Degradation
Buhimschi, Alexandru D, Armstrong, Haley A, Toure, Momar, Jaime-Figueroa, Saul, Chen, Timothy L, Lehman, Amy M, Woyach, Jennifer A, Johnson, Amy J, Byrd, John C, Crews, Craig M
Published in Biochemistry (Easton) (03.07.2018)
Published in Biochemistry (Easton) (03.07.2018)
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Journal Article
Targeted degradation of transcription factors by TRAFTACs: TRAnscription Factor TArgeting Chimeras
Samarasinghe, Kusal T.G., Jaime-Figueroa, Saul, Burgess, Michael, Nalawansha, Dhanusha A., Dai, Katherine, Hu, Zhenyi, Bebenek, Adrian, Holley, Scott A., Crews, Craig M.
Published in Cell chemical biology (20.05.2021)
Published in Cell chemical biology (20.05.2021)
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Journal Article
PROTAC-induced BET protein degradation as a therapy for castration-resistant prostate cancer
Raina, Kanak, Lu, Jing, Qian, Yimin, Altieri, Martha, Gordon, Deborah, Rossi, Ann Marie K., Wang, Jing, Chen, Xin, Dong, Hanqing, Siu, Kam, Winkler, James D., Crew, Andrew P., Crews, Craig M., Coleman, Kevin G.
Published in Proceedings of the National Academy of Sciences - PNAS (28.06.2016)
Published in Proceedings of the National Academy of Sciences - PNAS (28.06.2016)
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Journal Article