In Vitro Drug Metabolism Using Liver Microsomes
Knights, Kathleen M, Stresser, David M, Miners, John O, Crespi, Charles L
Published in Current protocols in pharmacology (01.09.2016)
Published in Current protocols in pharmacology (01.09.2016)
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Substrate-Dependent Modulation of CYP3A4 Catalytic Activity: Analysis of 27 Test Compounds with Four Fluorometric Substrates
STRESSER, David M, BLANCHARD, Andrew P, TURNER, Stephanie D, ERVE, John C. L, DANDENEAU, Andre A, MILLER, Vaughn P, CRESPI, Charles L
Published in Drug metabolism and disposition (01.12.2000)
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Published in Drug metabolism and disposition (01.12.2000)
Journal Article
HIGHLY SELECTIVE INHIBITION OF HUMAN CYP3A IN VITRO BY AZAMULIN AND EVIDENCE THAT INHIBITION IS IRREVERSIBLE
STRESSER, David M, BROUDY, Marc I, PATTEN, Christopher J, DEHAL, Shangara S, CRESPI, Charles L, THUY HO, CARGILL, Catherine E, BLANCHARD, Andrew P, SHARMA, Raman, DANDENEAU, Andre A, GOODWIN, Joseph J, TURNER, Stephanie D, ERVE, John C. L
Published in Drug metabolism and disposition (01.01.2004)
Published in Drug metabolism and disposition (01.01.2004)
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Comparison between Cytochrome P450 (CYP) Content and Relative Activity Approaches to Scaling from cDNA-Expressed CYPs to Human Liver Microsomes: Ratios of Accessory Proteins as Sources of Discrepancies between the Approaches
VENKATAKRISHNAN, Karthik, VON MOLTKE, Lisa L, COURT, Michael H, HARMATZ, Jerold S, CRESPI, Charles L, GREENBLATT, David J
Published in Drug metabolism and disposition (01.12.2000)
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Published in Drug metabolism and disposition (01.12.2000)
Journal Article
Cytochrome P450 Fluorometric Substrates: Identification of Isoform-Selective Probes for Rat CYP2D2 and Human CYP3A4
STRESSER, David M, TURNER, Stephanie D, BLANCHARD, Andrew P, MILLER, Vaughn P, CRESPI, Charles L
Published in Drug metabolism and disposition (01.07.2002)
Published in Drug metabolism and disposition (01.07.2002)
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Journal Article
A Novel Design of Artificial Membrane for Improving the PAMPA Model
Chen, Xiaoxi, Murawski, Anthony, Patel, Karishma, Crespi, Charles L., Balimane, Praveen V.
Published in Pharmaceutical research (01.07.2008)
Published in Pharmaceutical research (01.07.2008)
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Differential Time- and NADPH-Dependent Inhibition of CYP2C19 by Enantiomers of Fluoxetine
STRESSER, David M, MASON, Andrew K, PERLOFF, Elke S, HO, Thuy, CRESPI, Charles L, DANDENEAU, Andre A, MORGAN, Ling, DEHAL, Shangara S
Published in Drug metabolism and disposition (01.04.2009)
Published in Drug metabolism and disposition (01.04.2009)
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Journal Article
Human-Cell Mutagens in Respirable Airborne Particles in the Northeastern United States. 1. Mutagenicity of Fractionated Samples
Pedersen, Daniel U., Durant, John L., Penman, Bruce W., Crespi, Charles L., Hemond, Harold F., Lafleur, Arthur L., Cass, Glen R.
Published in Environmental science & technology (01.02.2004)
Published in Environmental science & technology (01.02.2004)
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Comparison of Species Differences of P-Glycoproteins in Beagle Dog, Rhesus Monkey, and Human Using ATPase Activity Assays
Xia, Cindy Q, Xiao, Guangqing, Liu, Ning, Pimprale, Satish, Fox, Lisa, Patten, Chris J, Crespi, Charles L, Miwa, Gerald, Gan, Liang-Shang
Published in Molecular pharmaceutics (01.01.2006)
Published in Molecular pharmaceutics (01.01.2006)
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HUMAN CYTOCHROME P450 INDUCTION AND INHIBITION POTENTIAL OF CLEVIDIPINE AND ITS PRIMARY METABOLITE H152/81
ZHANG, J. George, DEHAL, Shangara S, HO, Thuy, JOHNSON, Jennifer, CHANDLER, Catherine, BLANCHARD, Andrew P, CLARK, Robert J, CRESPI, Charles L, STRESSER, David M, WONG, James
Published in Drug metabolism and disposition (01.05.2006)
Published in Drug metabolism and disposition (01.05.2006)
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Journal Article
Bioassay-Directed Chemical Analysis of Los Angeles Airborne Particulate Matter Using a Human Cell Mutagenicity Assay
Hannigan, Michael P, Cass, Glen R, Penman, Bruce W, Crespi, Charles L, Lafleur, Arthur L, Busby, William F, Thilly, William G, Simoneit, Bernd R. T
Published in Environmental science & technology (15.11.1998)
Published in Environmental science & technology (15.11.1998)
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Mutagenicity of C24H14 PAH in human cells expressing CYP1A1
DURANT, J. L, LAFLEUR, A. L, BUSBY, W. F, DONHOFFNER, L. L, PENMAN, B. W, CRESPI, C. L
Published in Mutation research. Genetic toxicology and environmental mutagenesis (01.10.1999)
Published in Mutation research. Genetic toxicology and environmental mutagenesis (01.10.1999)
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Quantitative RT-PCR Measurement of Cytochromes p450 1A1, 1B1, and 2B7, Microsomal Epoxide Hydrolase, and NADPH Oxidoreductase Expression in Lung Cells of Smokers and Nonsmokers
Willey, James C, Coy, Erin L, Frampton, Mark W, Torres, Alfonso, Apostolakos, Michael J, Hoehn, Gerard, Schuermann, Wolfgang H, Thilly, William G, Olson, Dan E, Hammersley, Jeffrey R, Crespi, Charles L, Utell, Mark J
Published in American journal of respiratory cell and molecular biology (01.07.1997)
Published in American journal of respiratory cell and molecular biology (01.07.1997)
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The role of 12 cDNA-expressed human, rodent, and rabbit cytochromes P450 in the metabolism of benzo[a]pyrene and benzo[a]pyrene trans-7,8-dihydrodiol
Shou, M, Korzekwa, K R, Crespi, C L, Gonzalez, F J, Gelboin, H V
Published in Molecular carcinogenesis (01.07.1994)
Published in Molecular carcinogenesis (01.07.1994)
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CYP2C8 polymorphisms in Caucasians and their relationship with paclitaxel 6α-hydroxylase activity in human liver microsomes
Bahadur, Namrata, Leathart, Julian B.S, Mutch, Elaine, Steimel-Crespi, Dorothy, Dunn, Stuart A, Gilissen, Ron, Houdt, Jos Van, Hendrickx, Jan, Mannens, Geert, Bohets, Hilde, Williams, Faith M, Armstrong, Martin, Crespi, Charles L, Daly, Ann K
Published in Biochemical pharmacology (01.12.2002)
Published in Biochemical pharmacology (01.12.2002)
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A new cell-based model to study the important matters of OATP1B on drug disposition: Genetic variants and species differences
Li, Na, Wang, Jie, Cooper, Kirsten, Bourgea, Joanne, Singh, Ritu, Creegan, Tim, Crespi, Charles L., Patten, Christopher J.
Published in Drug metabolism and pharmacokinetics (01.01.2017)
Published in Drug metabolism and pharmacokinetics (01.01.2017)
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Journal Article
Characterizations of corning® hepatocells as a novel in vitro tool for drug metabolism and hepatotoxicity studies
Crespi, Charles L., Zuo, Rongjun, Li, Feng, Parikh, Sweta, Cooper, Kirsten, Liu, Jin, Faris, Ronald A., Patten, Christopher J.
Published in Drug metabolism and pharmacokinetics (01.01.2017)
Published in Drug metabolism and pharmacokinetics (01.01.2017)
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Journal Article
Microtiter Plate Assays for Inhibition of Human, Drug-Metabolizing Cytochromes P450
Crespi, Charles L., Miller, Vaughn P., Penman, Bruce W.
Published in Analytical biochemistry (15.05.1997)
Published in Analytical biochemistry (15.05.1997)
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Journal Article
Human cell mutagenicity of chlorinated and unchlorinated water and the disinfection byproduct 3-chloro-4-(dichloromethyl)-5-hydroxy-2(5 H)-furanone (MX)
Woodruff, Nathaniel W, Durant, John L, Donhoffner, Lawrence L, Crespi, Charles L, Penman, Bruce W
Published in Mutation research (22.08.2001)
Published in Mutation research (22.08.2001)
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