Discovery of a Potent and Selective Tyrosine Kinase 2 Inhibitor: TAK-279
Leit, Silvana, Greenwood, Jeremy, Carriero, Samantha, Mondal, Sayan, Abel, Robert, Ashwell, Mark, Blanchette, Heather, Boyles, Nicholas A., Cartwright, Mark, Collis, Alan, Feng, Shulu, Ghanakota, Phani, Harriman, Geraldine C., Hosagrahara, Vinayak, Kaila, Neelu, Kapeller, Rosanna, Rafi, Salma B., Romero, Donna L., Tarantino, Paul M., Timaniya, Jignesh, Toms, Angela V., Wester, Ronald T., Westlin, William, Srivastava, Bhaskar, Miao, Wenyan, Tummino, Peter, McElwee, Joshua J., Edmondson, Scott D., Masse, Craig E.
Published in Journal of medicinal chemistry (10.08.2023)
Published in Journal of medicinal chemistry (10.08.2023)
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Journal Article
Syntheses and Biological Evaluation of (+)-Lactacystin and Analogs
Masse, Craig E., Morgan, Adam J., Adams, Julian, Panek, James S.
Published in European journal of organic chemistry (01.07.2000)
Published in European journal of organic chemistry (01.07.2000)
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Journal Article
A General Method for the Enantioselective Synthesis of Pantolactone Derivatives
Evans, David A, Wu, Jimmy, Masse, Craig E, MacMillan, David W. C
Published in Organic letters (03.10.2002)
Published in Organic letters (03.10.2002)
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Journal Article
Potent and selective TYK2-JH1 inhibitors highly efficacious in rodent model of psoriasis
Leit, Silvana, Greenwood, Jeremy R., Mondal, Sayan, Carriero, Samantha, Dahlgren, Markus, Harriman, Geraldine C., Kennedy-Smith, Joshua J., Kapeller, Rosana, Lawson, Jon P., Romero, Donna L., Toms, Angela V., Shelley, Mee, Wester, Ronald T., Westlin, William, McElwee, Joshua J., Miao, Wenyan, Edmondson, Scott D., Masse, Craig E.
Published in Bioorganic & medicinal chemistry letters (01.10.2022)
Published in Bioorganic & medicinal chemistry letters (01.10.2022)
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Journal Article
Anti‐leukaemic activity of the TYK2 selective inhibitor NDI‐031301 in T‐cell acute lymphoblastic leukaemia
Akahane, Koshi, Li, Zhaodong, Etchin, Julia, Berezovskaya, Alla, Gjini, Evisa, Masse, Craig E., Miao, Wenyan, Rocnik, Jennifer, Kapeller, Rosana, Greenwood, Jeremy R., Tiv, Hong, Sanda, Takaomi, Weinstock, David M., Look, A. Thomas
Published in British journal of haematology (01.04.2017)
Published in British journal of haematology (01.04.2017)
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Journal Article
X‑ray Crystal Structures of Escherichia coli RNA Polymerase with Switch Region Binding Inhibitors Enable Rational Design of Squaramides with an Improved Fraction Unbound to Human Plasma Protein
Molodtsov, Vadim, Fleming, Paul R, Eyermann, Charles J, Ferguson, Andrew D, Foulk, Melinda A, McKinney, David C, Masse, Craig E, Buurman, Ed T, Murakami, Katsuhiko S
Published in Journal of medicinal chemistry (09.04.2015)
Published in Journal of medicinal chemistry (09.04.2015)
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Journal Article
The Exceptional Chelating Ability of Dimethylaluminum Chloride and Methylaluminum Dichloride. The Merged Stereochemical Impact of α- and β-Stereocenters in Chelate-Controlled Carbonyl Addition Reactions with Enolsilane and Hydride Nucleophiles
Evans, David A, Allison, Brett D, Yang, Michael G, Masse, Craig E
Published in Journal of the American Chemical Society (07.11.2001)
Published in Journal of the American Chemical Society (07.11.2001)
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Journal Article
Lewis Acid-Mediated Carbocyclization Reactions of Chiral (E)-Crotylsilanes
Masse, Craig E, Dakin, Les A, Knight, Bradford S, Panek, James S
Published in Journal of organic chemistry (26.12.1997)
Published in Journal of organic chemistry (26.12.1997)
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Journal Article
Design and synthesis of deuterated boceprevir analogs with enhanced pharmacokinetic properties
Morgan, Adam J., Nguyen, Sophia, Uttamsingh, Vinita, Bridson, Gary, Harbeson, Scott, Tung, Roger, Masse, Craig E.
Published in Journal of labelled compounds & radiopharmaceuticals (01.07.2011)
Published in Journal of labelled compounds & radiopharmaceuticals (01.07.2011)
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Journal Article
TYK2 INHIBITOR AND USE OF THE SAME
SILVANA MARCEL LEIT DE MORADEI, THOMAS H MCLEAN, JEREMY ROBERT GREENWOOD, CRAIG E MASSE, SAYAN MONDAL, GERALDINE C HARRIMAN
Year of Publication 01.08.2023
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Year of Publication 01.08.2023
Patent
TYK2 INHIBITOR AND USE THEREOF
JOSHUA JAHMIL KENNEDY-SMITH, MARKUS DAHLGREN, JEREMY ROBERT GREENWOOD, MEE SHELLEY, DONNA L ROMERO, RONALD T WESTER, CRAIG E MASSE, SAYAN MONDAL, GERALDINE C HARRIMAN
Year of Publication 09.09.2021
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Year of Publication 09.09.2021
Patent
ACC INHIBITORS AND USES THEREOF
JEREMY ROBERT GREENWOOD, CRAIG E MASSE, GERALDINE C HARRIMAN, JAMES HARWOOD, SATHESH BHAT
Year of Publication 05.09.2019
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Year of Publication 05.09.2019
Patent
ACC INHIBITORS AND USES THEREOF
JEREMY ROBERT GREENWOOD, CRAIG E MASSE, GERALDINE C HARRIMAN, JAMES HARWOOD, SATHESH BHAT
Year of Publication 05.04.2018
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Year of Publication 05.04.2018
Patent
TYK2 INHIBITOR AND USE THEREOF
JOSHUA JAHMIL KENNEDY-SMITH, MARKUS DAHLGREN, JEREMY ROBERT GREENWOOD, MEE SHELLEY, DONNA L ROMERO, RONALD T WESTER, CRAIG E MASSE, SAYAN MONDAL, GERALDINE C HARRIMAN
Year of Publication 10.10.2019
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Year of Publication 10.10.2019
Patent