Search Results - "COSTI ROBERTA" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Synthesis, biological evaluation and structure–activity correlation study of a series of imidazol-based compounds as Candida albicans inhibitors

Synthesis, biological evaluation and structure–activity correlation study of a series of imidazol-based compounds as Candida albicans inhibitors

by Moraca, Francesca, De Vita, Daniela, Pandolfi, Fabiana, Di Santo, Roberto, Costi, Roberta, Cirilli, Roberto, D’Auria, Felicia Diodata, Panella, Simona, Palamara, Anna Teresa, Simonetti, Giovanna, Botta, Maurizio, Scipione, Luigi
Published in European journal of medicinal chemistry (18.08.2014)

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New N,N-dimethylcarbamate inhibitors of acetylcholinesterase: design synthesis and biological evaluation

New N,N-dimethylcarbamate inhibitors of acetylcholinesterase: design synthesis and biological evaluation

by De Vita, Daniela, Pandolfi, Fabiana, Ornano, Luigi, Feroci, Marta, Chiarotto, Isabella, Sileno, Ilaria, Pepi, Federico, Costi, Roberta, Di Santo, Roberto, Scipione, Luigi
Published in Journal of enzyme inhibition and medicinal chemistry (04.11.2016)

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Oxidative stress and visual system

Oxidative stress and visual system

by Samanta Taurone, Massimo Ralli, Marco Artico, Valentina Noemi Madia, Susanna Scarpa, Stefania Annarita Nottola, Antonio Maconi, Marta Betti, Pietro Familiari, Marcella Nebbioso, Roberta Costi, Alessandra Micera
Published in EXCLI journal (01.03.2022)

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Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells

Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells

by Valente, Sergio, Lepore, Ilaria, Dell'Aversana, Carmela, Tardugno, Maria, Castellano, Sabrina, Sbardella, Gianluca, Tomassi, Stefano, Di Maro, Salvatore, Novellino, Ettore, Di Santo, Roberto, Costi, Roberta, Altucci, Lucia, Mai, Antonello
Published in Biochimie (01.11.2012)

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Design, Synthesis, and Structure–Activity Relationship of N‑Arylnaphthylamine Derivatives as Amyloid Aggregation Inhibitors

Design, Synthesis, and Structure–Activity Relationship of N‑Arylnaphthylamine Derivatives as Amyloid Aggregation Inhibitors

by Di Santo, Roberto, Costi, Roberta, Cuzzucoli Crucitti, Giuliana, Pescatori, Luca, Rosi, Federica, Scipione, Luigi, Celona, Diana, Vertechy, Mario, Ghirardi, Orlando, Piovesan, Paola, Marzi, Mauro, Caccia, Silvio, Guiso, Giovanna, Giorgi, Fabrizio, Minetti, Patrizia
Published in Journal of medicinal chemistry (11.10.2012)

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New Nucleotide-Competitive Non-Nucleoside Inhibitors of Terminal Deoxynucleotidyl Transferase: Discovery, Characterization, and Crystal Structure in Complex with the Target

New Nucleotide-Competitive Non-Nucleoside Inhibitors of Terminal Deoxynucleotidyl Transferase: Discovery, Characterization, and Crystal Structure in Complex with the Target

by Costi, Roberta, Cuzzucoli Crucitti, Giuliana, Pescatori, Luca, Messore, Antonella, Scipione, Luigi, Tortorella, Silvano, Amoroso, Alessandra, Crespan, Emmanuele, Campiglia, Pietro, Maresca, Bruno, Porta, Amalia, Granata, Ilaria, Novellino, Ettore, Gouge, Jérôme, Delarue, Marc, Maga, Giovanni, Di Santo, Roberto
Published in Journal of medicinal chemistry (26.09.2013)

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6-[1-(4-Fluorophenyl)methyl-1 H-pyrrol-2-yl)]-2,4-dioxo-5-hexenoic acid ethyl ester a novel diketo acid derivative which selectively inhibits the HIV-1 viral replication in cell culture and the ribonuclease H activity in vitro

6-[1-(4-Fluorophenyl)methyl-1 H-pyrrol-2-yl)]-2,4-dioxo-5-hexenoic acid ethyl ester a novel diketo acid derivative which selectively inhibits the HIV-1 viral replication in cell culture and the ribonuclease H activity in vitro

by Tramontano, Enzo, Esposito, Francesca, Badas, Roberta, Di Santo, Roberto, Costi, Roberta, La Colla, Paolo
Published in Antiviral research (01.02.2005)

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Structure–Activity Relationships on Cinnamoyl Derivatives as Inhibitors of p300 Histone Acetyltransferase

Structure–Activity Relationships on Cinnamoyl Derivatives as Inhibitors of p300 Histone Acetyltransferase

by Madia, Valentina Noemi, Benedetti, Rosaria, Barreca, Maria Letizia, Ngo, Liza, Pescatori, Luca, Messore, Antonella, Pupo, Giovanni, Saccoliti, Francesco, Valente, Sergio, Mai, Antonello, Scipione, Luigi, Zheng, Yujun George, Tintori, Cristina, Botta, Maurizio, Cecchetti, Violetta, Altucci, Lucia, Di Santo, Roberto, Costi, Roberta
Published in ChemMedChem (22.08.2017)

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Pharmacophore Assessment Through 3-D QSAR: Evaluation of the Predictive Ability on New Derivatives by the Application on a Series of Antitubercular Agents

Pharmacophore Assessment Through 3-D QSAR: Evaluation of the Predictive Ability on New Derivatives by the Application on a Series of Antitubercular Agents

by Friggeri, Laura, Ballante, Flavio, Ragno, Rino, Musmuca, Ira, De Vita, Daniela, Manetti, Fabrizio, Biava, Mariangela, Scipione, Luigi, Di Santo, Roberto, Costi, Roberta, Feroci, Marta, Tortorella, Silvano
Published in Journal of chemical information and modeling (24.06.2013)

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Structure-guided approach identifies a novel class of HIV-1 ribonuclease H inhibitors: binding mode insights through magnesium complexation and site-directed mutagenesis studiesElectronic supplementary information (ESI) available. See DOI: 10.1039/c7md00600d

Structure-guided approach identifies a novel class of HIV-1 ribonuclease H inhibitors: binding mode insights through magnesium complexation and site-directed mutagenesis studiesElectronic supplementary information (ESI) available. See DOI: 10.1039/c7md00600d

by Poongavanam, Vasanthanathan, Corona, Angela, Steinmann, Casper, Scipione, Luigi, Grandi, Nicole, Pandolfi, Fabiana, Di Santo, Roberto, Costi, Roberta, Esposito, Francesca, Tramontano, Enzo, Kongsted, Jacob
Year of Publication 20.03.2018

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Structure-guided approach identifies a novel class of HIV-1 ribonuclease H inhibitors: binding mode insights through magnesium complexation and site-directed mutagenesis studies† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c7md00600d

Structure-guided approach identifies a novel class of HIV-1 ribonuclease H inhibitors: binding mode insights through magnesium complexation and site-directed mutagenesis studies† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c7md00600d

by Poongavanam, Vasanthanathan, Corona, Angela, Steinmann, Casper, Scipione, Luigi, Grandi, Nicole, Pandolfi, Fabiana, Di Santo, Roberto, Costi, Roberta, Esposito, Francesca, Tramontano, Enzo, Kongsted, Jacob
Published in MedChemComm (01.02.2018)

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Antifungal Agents. 11. N-Substituted Derivatives of 1-[(Aryl)(4-aryl-1H-pyrrol-3-yl)methyl]-1H-imidazole: Synthesis, Anti-Candida Activity, and QSAR Studies

Antifungal Agents. 11. N-Substituted Derivatives of 1-[(Aryl)(4-aryl-1H-pyrrol-3-yl)methyl]-1H-imidazole: Synthesis, Anti-Candida Activity, and QSAR Studies

by Di Santo, Roberto, Tafi, Andrea, Costi, Roberta, Botta, Maurizo, Artico, Marino, Corelli, Federico, Forte, Michela, Caporuscio, Fabiana, Angiolella, Letizia, Palamara, Anna Teresa
Published in Journal of medicinal chemistry (11.08.2005)

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Cinnamoyl Compounds as Simple Molecules that Inhibit p300 Histone Acetyltransferase

Cinnamoyl Compounds as Simple Molecules that Inhibit p300 Histone Acetyltransferase

by Costi, Roberta, Di Santo, Roberto, Artico, Marino, Miele, Gaetano, Valentini, Paola, Novellino, Ettore, Cereseto, Anna
Published in Journal of medicinal chemistry (19.04.2007)

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Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-Associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity

Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-Associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity

by Cheng, Donghang, Valente, Sergio, Castellano, Sabrina, Sbardella, Gianluca, Di Santo, Roberto, Costi, Roberta, Bedford, Mark T, Mai, Antonello
Published in Journal of medicinal chemistry (14.07.2011)

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Convenient Route to 2 H -Pyrrolo[3,4- b ]quinolin-9(4 H )-one Skeleton via TosMIC Reaction

Convenient Route to 2 H -Pyrrolo[3,4- b ]quinolin-9(4 H )-one Skeleton via TosMIC Reaction

by Rosi, Federica, Crucitti, Giuliana Cuzzucoli, Iacovo, Alberto, Miele, Gaetano, Pescatori, Luca, Santo, Roberto Di, Costi, Roberta
Published in Synthetic communications (01.03.2013)

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Design, synthesis and QSAR studies on N-aryl heteroarylisopropanolamines, a new class of non-peptidic HIV-1 protease inhibitors

Design, synthesis and QSAR studies on N-aryl heteroarylisopropanolamines, a new class of non-peptidic HIV-1 protease inhibitors

by DI SANTO, Roberto, COSTI, Roberta, ARTICO, Marino, MASSA, Silvio, RAGNO, Rino, MARSHALL, Garland R, LA COLLA, Paolo
Published in Bioorganic & medicinal chemistry (01.08.2002)

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Novel Quinolinonyl Diketo Acid Derivatives as HIV-1 Integrase Inhibitors: Design, Synthesis, and Biological Activities

Novel Quinolinonyl Diketo Acid Derivatives as HIV-1 Integrase Inhibitors: Design, Synthesis, and Biological Activities

by Di Santo, Roberto, Costi, Roberta, Roux, Alessandra, Miele, Gaetano, Crucitti, Giuliana Cuzzucoli, Iacovo, Alberto, Rosi, Federica, Lavecchia, Antonio, Marinelli, Luciana, Di Giovanni, Carmen, Novellino, Ettore, Palmisano, Lucia, Andreotti, Mauro, Amici, Roberta, Galluzzo, Clementina Maria, Nencioni, Lucia, Palamara, Anna Teresa, Pommier, Yves, Marchand, Christophe
Published in Journal of medicinal chemistry (14.08.2008)

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Novel Bifunctional Quinolonyl Diketo Acid Derivatives as HIV-1 Integrase Inhibitors: Design, Synthesis, Biological Activities, and Mechanism of Action

Novel Bifunctional Quinolonyl Diketo Acid Derivatives as HIV-1 Integrase Inhibitors: Design, Synthesis, Biological Activities, and Mechanism of Action

by Di Santo, Roberto, Costi, Roberta, Roux, Alessandra, Artico, Marino, Lavecchia, Antonio, Marinelli, Luciana, Novellino, Ettore, Palmisano, Lucia, Andreotti, Mauro, Amici, Roberta, Galluzzo, Clementina Maria, Nencioni, Lucia, Palamara, Anna Teresa, Pommier, Yves, Marchand, Christophe
Published in Journal of medicinal chemistry (23.03.2006)

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New Promising Compounds with in Vitro Nanomolar Activity against Trypanosoma cruzi

New Promising Compounds with in Vitro Nanomolar Activity against Trypanosoma cruzi

by Friggeri, Laura, Scipione, Luigi, Costi, Roberta, Kaiser, Marcel, Moraca, Francesca, Zamperini, Claudio, Botta, Bruno, Di Santo, Roberto, De Vita, Daniela, Brun, Reto, Tortorella, Silvano
Published in ACS medicinal chemistry letters (13.06.2013)

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Efeitos da intervenção multidisciplinar sobre a ingestão alimentar em adolescentes obesos

Efeitos da intervenção multidisciplinar sobre a ingestão alimentar em adolescentes obesos

by Andrade, Maria Laura Siqueira de Souza, Silva, Humberto José Gomes da, Lofrano-Prado, Mara Cristina, Ferreira, Moacir De Novaes Lima, Lins, Tatiana Acioli, Costi, Roberta Burkhardt, Prado, Wagner Luiz
Published in Conscientiae saúde (11.07.2012)

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