Discovery of PiragliatinFirst Glucokinase Activator Studied in Type 2 Diabetic Patients
Sarabu, Ramakanth, Bizzarro, Fred T, Corbett, Wendy L, Dvorozniak, Mark T, Geng, Wanping, Grippo, Joseph F, Haynes, Nancy-Ellen, Hutchings, Stanley, Garofalo, Lisa, Guertin, Kevin R, Hilliard, Darryl W, Kabat, Marek, Kester, Robert F, Ka, Wang, Liang, Zhenmin, Mahaney, Paige E, Marcus, Linda, Matschinsky, Franz M, Moore, David, Racha, Jagdish, Radinov, Roumen, Ren, Yi, Qi, Lida, Pignatello, Michael, Spence, Cheryl L, Steele, Thomas, Tengi, John, Grimsby, Joseph
Published in Journal of medicinal chemistry (23.08.2012)
Published in Journal of medicinal chemistry (23.08.2012)
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Journal Article
Allosteric Activators of Glucokinase: Potential Role in Diabetes Therapy
Grimsby, Joseph, Sarabu, Ramakanth, Corbett, Wendy L., Haynes, Nancy-Ellen, Bizzarro, Fred T., Coffey, John W., Guertin, Kevin R., Hilliard, Darryl W., Kester, Robert F., Mahaney, Paige E., Marcus, Linda, Qi, Lida, Spence, Cheryl L., Tengi, John, Magnuson, Mark A., Chu, Chang An, Dvorozniak, Mark T., Matschinsky, Franz M., Grippo, Joseph F.
Published in Science (American Association for the Advancement of Science) (18.07.2003)
Published in Science (American Association for the Advancement of Science) (18.07.2003)
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Discovery, Structure−Activity Relationships, Pharmacokinetics, and Efficacy of Glucokinase Activator (2R)-3-Cyclopentyl-2-(4-methanesulfonylphenyl)-N-thiazol-2-yl-propionamide (RO0281675)
Haynes, Nancy-Ellen, Corbett, Wendy L, Bizzarro, Fred T, Guertin, Kevin R, Hilliard, Darryl W, Holland, George W, Kester, Robert F, Mahaney, Paige E, Qi, Lida, Spence, Cheryl L, Tengi, John, Dvorozniak, Mark T, Railkar, Aruna, Matschinsky, Franz M, Grippo, Joseph F, Grimsby, Joseph, Sarabu, Ramakanth
Published in Journal of medicinal chemistry (13.05.2010)
Published in Journal of medicinal chemistry (13.05.2010)
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Journal Article
2,3-Disubstituted acrylamides as potent glucokinase activators
Sidduri, Achyutharao, Grimsby, Joseph S., Corbett, Wendy L., Sarabu, Ramakanth, Grippo, Joseph F., Lou, Jianping, Kester, Robert F., Dvorozniak, Mark, Marcus, Linda, Spence, Cheryl, Racha, Jagdish K., Moore, David J.
Published in Bioorganic & medicinal chemistry letters (01.10.2010)
Published in Bioorganic & medicinal chemistry letters (01.10.2010)
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Journal Article
Identification of RO4597014, a Glucokinase Activator Studied in the Clinic for the Treatment of Type 2 Diabetes
Qian, Yimin, Corbett, Wendy L, Berthel, Steven J, Choi, Duk Soon, Dvorozniak, Mark T, Geng, Wanping, Gillespie, Paul, Guertin, Kevin R, Haynes, Nancy-Ellen, Kester, Robert F, Mennona, Francis A, Moore, David, Racha, Jagdish, Radinov, Roumen, Sarabu, Ramakanth, Scott, Nathan R, Grimsby, Joseph, Mallalieu, Navita L
Published in ACS medicinal chemistry letters (11.04.2013)
Published in ACS medicinal chemistry letters (11.04.2013)
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Journal Article
Room-temperature, endo-specific 1-aza-1,3-butadiene Diels-Alder reactions: acceleration of the LUMOdiene-controlled [4 + 2] cycloaddition reactions through noncomplementary aza diene substitution
Boger, Dale L, Corbett, Wendy L, Wiggins, J. Mark
Published in Journal of organic chemistry (01.05.1990)
Published in Journal of organic chemistry (01.05.1990)
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Journal Article
Inverse electron-demand Diels-Alder reactions of N-sulfonyl .alpha.,.beta.-unsaturated imines: a general approach to implementation of the 4.pi. participation of 1-aza-1,3-butadienes in Diels-Alder reactions
Boger, Dale L, Corbett, Wendy L, Curran, Timothy T, Kasper, A. M
Published in Journal of the American Chemical Society (01.02.1991)
Published in Journal of the American Chemical Society (01.02.1991)
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Journal Article
Inverse electron demand diels-alder reactions of N-sulfonyl α,β-unsaturated imines : a general approach to implementation of the 4π participation of 1-aza-1,3-butadienes in diels-alder reactions
BOGER, D. L, CORBETT, W. L, CURRAN, T. T, KASPER, A. M
Published in Journal of the American Chemical Society (27.02.1991)
Published in Journal of the American Chemical Society (27.02.1991)
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Journal Article
Crystals of Glucokinase and methods of growing them
CORBETT WENDY L, LUKACS CHRISTINE M, CROWTHER ROBERT L, KAMMLOTT R. URSULA, DUNTEN PETE W
Year of Publication 29.06.2006
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Year of Publication 29.06.2006
Patent
Heteroaromatic glucokinase activators
BIZZARRO FRED T, KESTER ROBERT F, HOLLAND GEORGE W, CORBETT WENDY L, GRIPPO JOSEPH F, MAHANEY PAIGE E, SARABU RAMAKANTH, HAYNES NANCY-ELLEN
Year of Publication 30.08.2007
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Year of Publication 30.08.2007
Patent
Substituted-cycloalkyl and oxygenated-cycloalkyl glucokinase activators
GRIMSBY JOSEPH S, KESTER ROBERT F, RACHA JAGDISH K, CORBETT WENDY L, MAHANEY PAIGE E, SARABU RAMAKANTH, HAYNES NANCY-ELLEN, WANG KA
Year of Publication 10.08.2006
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Year of Publication 10.08.2006
Patent
Heteroaromatic glucokinase activators
KESTER ROBERT F, HOLLAND GEORGE W, CORBETT WENDY L, GRIPPO JOSEPH F, MAHANEY PAIGE E, BIZZARO FRED T, SARABU RAMAKANTH, HAYNES NANCY-ELLEN
Year of Publication 24.11.2005
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Year of Publication 24.11.2005
Patent
FUSED HETEROAROMATIC GLUCOKINASE ACTIVATORS
GRIMSBY JOSEPH S, KESTER ROBERT F, CORBETT WENDY L, MAHANEY PAIGE E, SARABU RAMAKANTH, HAYNES NANCY-ELLEN
Year of Publication 15.08.2002
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Year of Publication 15.08.2002
Patent
FUSED HETEROAROMATIC GLUCOKINASE ACTIVATORS
GRIMSBY JOSEHP S, KESTER ROBERT F, CORBETT WENDY L, MAHANEY PAIGE E, SARABU RAMAKANTH, HAYNES NANCY-ELLEN
Year of Publication 01.08.2002
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Year of Publication 01.08.2002
Patent
ACTIVADORES CICLOALQUIL SUSTITUIDOS Y CICLOALQUIL OXIGENADOS DE GLUCOQUINASA
JOSEPH S. GRIMSBY, RAMAKANTH SARABU, JAGDISH K. RACHA, ROBERT F.KESTER, NANCY-ELLEN HAYNES, KA WANG, PAIGE E. MAHENEY, WENDY L. CORBETT
Year of Publication 31.10.2003
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Year of Publication 31.10.2003
Patent