Search Results - "COOYMANS, LUDWIG P" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

The discovery and preclinical characterization of 6-chloro-N-(2-(4,4-difluoropiperidin-1-yl)-2-(2-(trifluoromethyl)pyrimidin-5-yl)ethyl)quinoline-5-carboxamide based P2X7 antagonists

The discovery and preclinical characterization of 6-chloro-N-(2-(4,4-difluoropiperidin-1-yl)-2-(2-(trifluoromethyl)pyrimidin-5-yl)ethyl)quinoline-5-carboxamide based P2X7 antagonists

by Rech, Jason C., Bhattacharya, Anindya, Branstetter, Bryan J., Love, Christopher J., Leenaerts, Joseph E., Cooymans, Ludwig P., Eckert, William A., Ao, Hong, Wang, Qi, Chaplan, Sandra R., Wickenden, Alan D., Lebsack, Alec D., Breitenbucher, J. Guy
Published in Bioorganic & medicinal chemistry letters (01.10.2016)

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Journal Article

NOVEL ALPHA-DIARYL-4-ARYL-4-HYDROXY-1-PIPERIDINEBUTANAAMIDE-N-OXIDES

NOVEL ALPHA-DIARYL-4-ARYL-4-HYDROXY-1-PIPERIDINEBUTANAAMIDE-N-OXIDES

by WALS, LOWRENS, COOYMANS, LUDWIG P
Year of Publication 05.03.1994

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Patent

The discovery and preclinical characterization of 6-chloro-N-(2-(4,4-difluoropiperidin-1-yl)-2-(2-(trifluoromethyl)p y rimidin-5-yl)ethyl)quinoline-5-carboxamide based P2X7 antagonists

The discovery and preclinical characterization of 6-chloro-N-(2-(4,4-difluoropiperidin-1-yl)-2-(2-(trifluoromethyl)p y rimidin-5-yl)ethyl)quinoline-5-carboxamide based P2X7 antagonists

by Rech, Jason C, Bhattacharya, Anindya, Branstetter, Bryan J, Love, Christopher J, Leenaerts, Joseph E, Cooymans, Ludwig P, Eckert, William A, Ao, Hong, Wang, Qi, Chaplan, Sandra R, Wickenden, Alan D, Lebsack, Alec D, Breitenbucher, JGuy
Published in Bioorganic & medicinal chemistry letters (01.10.2016)

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Journal Article

DIARYL-4-ARYL-4-HYDROXY-1-PIPERIDINEBUTANAMIDE, N-OXIDES

DIARYL-4-ARYL-4-HYDROXY-1-PIPERIDINEBUTANAMIDE, N-OXIDES

by WALS, LOURENS, COOYMANS, LUDWIG P
Year of Publication 04.10.1994

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Patent

2,4-DISUBSTITUTED THIAZOLYL DERIVATIVES

2,4-DISUBSTITUTED THIAZOLYL DERIVATIVES

by LUDO EDMOND JOSEPHINE KENNIS, JEAN PIERRE FRANS VAN WAUWE, NELE, VANDERMAESEN, CHRISTOPHER JOHN LOVE, LUDWIG P. COOYMANS, MARC J. DE BRABANDER
Year of Publication 31.05.2010

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Patent

N-OXIDES OF ALPHA, ALPHA-DIARYL-4-ARYL-4-HYDROXY-1-PIEPRIDINEBUTANEAMIDES, PROCESS OF THEIR PREPARATION AND PHARMACEUTICALS BASED THEREON

N-OXIDES OF ALPHA, ALPHA-DIARYL-4-ARYL-4-HYDROXY-1-PIEPRIDINEBUTANEAMIDES, PROCESS OF THEIR PREPARATION AND PHARMACEUTICALS BASED THEREON

by WALS LOURENS, COOYMANS LUDWIG P
Year of Publication 15.04.1992

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Patent

N-OXIDES OF ALPHA, ALPHA-DIARYL-4-ARYL-4-HYDROXY-1-PIEPRIDINEBUTANEAMIDES, PROCESS OF THEIR PREPARATION AND PHARMACEUTICALS BASED THEREON

N-OXIDES OF ALPHA, ALPHA-DIARYL-4-ARYL-4-HYDROXY-1-PIEPRIDINEBUTANEAMIDES, PROCESS OF THEIR PREPARATION AND PHARMACEUTICALS BASED THEREON

by WALS LOURENS, COOYMANS LUDWIG P
Year of Publication 15.04.1992

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Patent

Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors

Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors

by BUIJINSTERS PETER JACOBUS J.A, LOVE CHRISTOPHER J, VANDERMAESEN NELE, COOYMANS LUDWIG P, EDGARD FREYNE EDDY J
Year of Publication 14.09.2006

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Patent

alpha , alpha -Diaryl-4-aryl-4-hydroxyl-1-piperidinebutanamide, N-oxides and pharmaceutical use

alpha , alpha -Diaryl-4-aryl-4-hydroxyl-1-piperidinebutanamide, N-oxides and pharmaceutical use

by COOYMANS; LUDWIG P, WALS; LOURENS
Year of Publication 06.02.1990

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Patent

alpha , alpha -diaryl-4-aryl-4-hydroxy-1-piperidinebutanamide, N-oxides and method of treating diarrhea

alpha , alpha -diaryl-4-aryl-4-hydroxy-1-piperidinebutanamide, N-oxides and method of treating diarrhea

by COOYMANS; LUDWIG P, WALS; LOURENS
Year of Publication 25.04.1989

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Patent

Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors

Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors

by LOVE CHRISTOPHER J, WILLEMS MARC, EMBRECHTS WERNER C.J, FREYNE EDDY J.E, VANDERMAESEN NELE, BUIJNSTERS PETER JACOBUS J.A, COOYMANS LUDWIG P
Year of Publication 17.08.2006

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Patent

IMIDAZO[1,2-A](PYRROLO, THIENO OR FURANO)[3,2-D]AZEPINE DERIVATIVES, COMPOSITIONS AND METHODS OF USE

IMIDAZO[1,2-A](PYRROLO, THIENO OR FURANO)[3,2-D]AZEPINE DERIVATIVES, COMPOSITIONS AND METHODS OF USE

by DIELS, GASTON S. M, JANSSENS, FRANS E, COOYMANS, LUDWIG P, LEENAERTS, JOSEPH E
Year of Publication 26.11.2002

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Patent

2-Amino-4,5-Trisubstituted Thiazolyl Derivatives

2-Amino-4,5-Trisubstituted Thiazolyl Derivatives

by COESEMANS ERWIN, DOYON JULIEN GEORGES P, LOVE CHRISTOPHER J, ANTONIUS BUIJNSTERS PETER JACOBUS J, BOECKX GUSTAAF M, VAN LOMMEN GUY R.E, HENDRICKX ROBERT J.M, BONGARTZ JEAN-PIERRE A.M, VANDERMAESEN NELE, VAN DER AA MARCEL J.M, COOYMANS LUDWIG P
Year of Publication 30.08.2007

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Patent

NEW OXAZOLYL DERIVATIVES

NEW OXAZOLYL DERIVATIVES

by SOMMEN, FRANCOIS M, JANSSENS, FRANS E, DIERCKX, ANN C, COOYMANS, LUDWIG P
Year of Publication 30.06.1997

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Patent

METHOD OF OBTAINING NOVEL DERIVATIVES OF IMIDAZO[1,2-A](PYROLLE, THIENE OR FURAANE)-[3,2-D] AZEPINS

METHOD OF OBTAINING NOVEL DERIVATIVES OF IMIDAZO[1,2-A](PYROLLE, THIENE OR FURAANE)-[3,2-D] AZEPINS

by DIELS GASTON S. M, LEENAERTS JOSEPH E, COOYMANS LUDWIG P, JANSSENS FRANS E
Year of Publication 31.12.1996

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Patent

METHOD OF OBTAINING NOVEL OXAZOLYL DERIVATIVES

METHOD OF OBTAINING NOVEL OXAZOLYL DERIVATIVES

by DIERCKX ANN CH. J, SOMMEN FRANCOIS M, COOYMANS LUDWIG P, JANSSENS FRANS E
Year of Publication 31.07.1996

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Patent

OXAZOLE DERIVATIVES METHOD OF THEIR PRODUCTION AND ANTIALERGIC PREPARATIONS ON THEIR BASE

OXAZOLE DERIVATIVES METHOD OF THEIR PRODUCTION AND ANTIALERGIC PREPARATIONS ON THEIR BASE

by DIERCKX ANN CHRISTINA J, SOMMEN FRANCOIS M, COOYMANS LUDWIG P, JANSSENS FRANS E
Year of Publication 07.02.1996

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Patent

Imidazo[1,2-a](pyrrolo, thieno or furano) [3,2a-d]azepine derivatives, compositions and methods of use

Imidazo[1,2-a](pyrrolo, thieno or furano) [3,2a-d]azepine derivatives, compositions and methods of use

by LEENAERTS; JOSEPH E, JANSSENS; FRANS E, COOYMANS; LUDWIG P, DIELS; GASTON S. M
Year of Publication 24.10.1995

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Patent

Oxazolyl imidazol[4,5-b]pyridin and pyrimidine compounds

Oxazolyl imidazol[4,5-b]pyridin and pyrimidine compounds

by JANSSENS; FRANS E, DIERCKX; ANN C. J, COOYMANS; LUDWIG P, SOMMEN; FRANCOIS M
Year of Publication 11.01.1994

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Patent

Oxazolyl and piperidinyl substituted benimidazolyl compounds

Oxazolyl and piperidinyl substituted benimidazolyl compounds

by JANSSENS; FRANS E, DIERCKX; ANN C. J, COOYMANS; LUDWIG P, SOMMEN; FRANCOIS M
Year of Publication 08.06.1993

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Patent