Comparison of amine additives most effective in the new methyltrioxorhenium-catalyzed epoxidation process
Adolfsson, Hans, Converso, Antonella, Sharpless, K.Barry
Published in Tetrahedron letters (21.05.1999)
Published in Tetrahedron letters (21.05.1999)
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Journal Article
Studies toward the Synthesis of Azadirachtin, Part 2: Construction of Fully Functionalized ABCD Ring Frameworks and Unusual Intramolecular Reactions Induced by Close-Proximity Effects
Nicolaou, K. C., Sasmal, Pradip K., Koftis, Theocharis V., Converso, Antonella, Loizidou, Eriketi, Kaiser, Florian, Roecker, A. J., Dellios, Constantinos C., Sun, Xiao-Wen, Petrovic, Goran
Published in Angewandte Chemie (International ed.) (30.05.2005)
Published in Angewandte Chemie (International ed.) (30.05.2005)
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Journal Article
Simple and efficient routes for the preparation of isoxazolidinyl nucleosides containing cytosine and 5-methyl-cytosine as new potential anti-HIV drugs
Colacino, Evelina, Converso, Antonella, Liguori, Angelo, Napoli, Anna, Siciliano, Carlo, Sindona, Giovanni
Published in Tetrahedron (01.10.2001)
Published in Tetrahedron (01.10.2001)
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Journal Article
Dose Number as a Tool to Guide Lead Optimization for Orally Bioavailable Compounds in Drug Discovery
Wuelfing, W. Peter, El Marrouni, Abdellatif, Lipert, Maya P, Daublain, Pierre, Kesisoglou, Filippos, Converso, Antonella, Templeton, Allen C
Published in Journal of medicinal chemistry (10.02.2022)
Published in Journal of medicinal chemistry (10.02.2022)
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Journal Article
Development of a sp2–sp3 Stille Cross-Coupling for Rapid Synthesis of HIV NNRTI Doravirine Analogues
ElMarrouni, Abdellatif, Campbell, Mark, Perkins, James J, Converso, Antonella
Published in Organic letters (16.06.2017)
Published in Organic letters (16.06.2017)
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Journal Article
Discovery of arylsulfonamides as a novel class of allosteric integrase inhibitors with antiviral activity
Wang, Cheng, Adam, Gregory C., Burlein, Christine, Carroll, Steven, Dankulich, William, Diamond, Tracy, Grobler, Jay, Heath, Jeffrey, Johnson, Adam, Klein, Daniel, Krosky, Daniel, Narayan, Kartik, Ou, Yangsi, Sanders, John, Sharma, Sujata, Xu, Min, Converso, Antonella
Published in Bioorganic & medicinal chemistry letters (01.06.2023)
Published in Bioorganic & medicinal chemistry letters (01.06.2023)
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Journal Article
Augmenting Hit Identification by Virtual Screening Techniques in Small Molecule Drug Discovery
Yan, Xin Cindy, Sanders, John M, Gao, Ying-Duo, Tudor, Matthew, Haidle, Andrew M, Klein, Daniel J, Converso, Antonella, Lesburg, Charles A, Zang, Yi, Wood, Harold B
Published in Journal of chemical information and modeling (28.09.2020)
Published in Journal of chemical information and modeling (28.09.2020)
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Journal Article
Potent targeted activator of cell kill molecules eliminate cells expressing HIV-1
Balibar, Carl J, Klein, Daniel J, Zamlynny, Beata, Diamond, Tracy L, Fang, Zhiyu, Cheney, Carol A, Kristoff, Jan, Lu, Meiqing, Bukhtiyarova, Marina, Ou, Yangsi, Xu, Min, Ba, Lei, Carroll, Steven S, El Marrouni, Abdellatif, Fay, John F, Forster, Ashley, Goh, Shih Lin, Gu, Meigang, Krosky, Daniel, Rosenbloom, Daniel I S, Sheth, Payal, Wang, Deping, Wu, Guoxin, Zebisch, Matthias, Zhao, Tian, Zuck, Paul, Grobler, Jay, Hazuda, Daria J, Howell, Bonnie J, Converso, Antonella
Published in Science translational medicine (22.02.2023)
Published in Science translational medicine (22.02.2023)
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Journal Article
A Phenotypic Screen Identifies Potent DPP9 Inhibitors Capable of Killing HIV‑1 Infected Cells
Moore, Keith P., Schwaid, Adam G., Tudor, Matthew, Park, Sangho, Beshore, Douglas C., Converso, Antonella, Shipe, William D., Anand, Rajan, Lan, Ping, Moningka, Remond, Rothman, Deborah M., Sun, Wanying, Chi, An, Cornella-Taracido, Ivan, Adam, Gregory C., Bahnck-Teets, Carolyn, Carroll, Steven S., Fay, John F., Goh, Shih Lin, Lusen, Jeffrey, Quan, Shuo, Rodriguez, Silveria, Xu, Min, Andrews, Christine L., Song, Cheng, Filzen, Tracey, Li, Jing, Hollenstein, Kaspar, Klein, Daniel J., Lammens, Alfred, Lim, U-Ming, Fang, Zhiyu, McHale, Carolyn, Li, Yuan, Lu, Meiqing, Diamond, Tracy L., Howell, Bonnie J., Zuck, Paul, Balibar, Carl J.
Published in ACS chemical biology (16.09.2022)
Published in ACS chemical biology (16.09.2022)
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Journal Article
Discovery of 4-arylquinoline-2-carboxamides, highly potent and selective class of mGluR2 negative allosteric modulators: From HTS to activity in animal models
Shu, Youheng, Diamond, Tracy L., Hershey, James C., Huang, Shaei, Magliaro, Brian C., O'Brien, Julie A., Schlegel, Kelly-Ann S., Puri, Vanita, Uebele, Victor N., Uslaner, Jason M., Wang, Cheng, Converso, Antonella
Published in Bioorganic & medicinal chemistry letters (01.05.2020)
Published in Bioorganic & medicinal chemistry letters (01.05.2020)
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Journal Article
선택적 세포독성제로서의 테트라히드로퀴나졸린 유도체
FORSTER ASHLEY, WANG CHENG, SHAW ANTHONY W, ZHANG YUNLONG, CONVERSO ANTONELLA, EL MARROUNI ABDELLATIF, HUNTER DAVID N
Year of Publication 28.04.2023
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Year of Publication 28.04.2023
Patent
Discovery of a Distinct Chemical and Mechanistic Class of Allosteric HIV‑1 Integrase Inhibitors with Antiretroviral Activity
Burlein, Christine, Wang, Cheng, Xu, Min, Bhatt, Triveni, Stahlhut, Mark, Ou, Yangsi, Adam, Gregory C, Heath, Jeffrey, Klein, Daniel J, Sanders, John, Narayan, Kartik, Abeywickrema, Pravien, Heo, Mee Ra, Carroll, Steven S, Grobler, Jay A, Sharma, Sujata, Diamond, Tracy L, Converso, Antonella, Krosky, Daniel J
Published in ACS chemical biology (17.11.2017)
Published in ACS chemical biology (17.11.2017)
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Journal Article
Discovery of MK-8768, a Potent and Selective mGluR2 Negative Allosteric Modulator
Rudd, Michael T., Manley, Peter J., Hanney, Barbara, Meng, Zhaoyang, Shu, Youheng, de Leon, Pablo, Frie, Jessica L., Han, Yongxin, Wai, Jenny Miu-Chun, Yang, Zhi-Qiang, Perkins, James J., Hurzy, Danielle M., Manikowski, Jesse J., Zhu, Hong, Bungard, Christopher J., Converso, Antonella, Meissner, Robert S., Cosden, Mali L., Hayashi, Ikuo, Ma, Lei, O’Brien, Julie, Uebele, Victor N., Schachter, Joel B., Bhandari, Neetesh, Ward, Gwendolyn J., Fillgrove, Kerry L., Lu, Bing, Liang, Yuexia, Dubost, David C., Puri, Vanita, Eddins, Donnie M., Vardigan, Joshua D., Drolet, Robert E., Kern, Jonathan T., Uslaner, Jason M.
Published in ACS medicinal chemistry letters (10.08.2023)
Published in ACS medicinal chemistry letters (10.08.2023)
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Journal Article
HIV 감염된 세포에 대한 선택적 세포독성제로서의 피리디논 유도체
FORSTER ASHLEY, WANG CHENG, WANG DEPING, FRIE JESSICA L, CONVERSO ANTONELLA, EL MARROUNI ABDELLATIF, HUNTER DAVID N
Year of Publication 28.01.2022
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Year of Publication 28.01.2022
Patent
Studies toward the Synthesis of Azadirachtin, Part 2: Construction of Fully Functionalized ABCD Ring Frameworks and Unusual Intramolecular Reactions Induced by Close-Proximity Effects
Nicolaou, K. C., Sasmal, Pradip K., Koftis, Theocharis V., Converso, Antonella, Loizidou, Eriketi, Kaiser, Florian, Roecker, A. J., Dellios, Constantinos C., Sun, Xiao-Wen, Petrovic, Goran
Published in Angewandte Chemie (30.05.2005)
Published in Angewandte Chemie (30.05.2005)
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Journal Article
Kinetic Analysis of Membrane Potential Dye Response to NaV1.7 Channel Activation Identifies Antagonists with Pharmacological Selectivity against NaV1.5
Finley, Michael, Cassaday, Jason, Kreamer, Tony, Li, Xinnian, Solly, Kelli, O'Donnell, Greg, Clements, Michelle, Converso, Antonella, Cook, Sean, Daley, Chris, Kraus, Richard, Lai, Ming-Tain, Layton, Mark, Lemaire, Wei, Staas, Donnette, Wang, Jixin
Published in Journal of biomolecular screening (01.06.2016)
Published in Journal of biomolecular screening (01.06.2016)
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