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The design and synthesis of novel α-ketoamide-based p38 MAP kinase inhibitors
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Published in Bioorganic & medicinal chemistry letters (15.03.2008)
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Published in Bioorganic & medicinal chemistry letters (15.10.2008)
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SUBSTITUTED BICYCLIC ALKOXY PYRAZOLE ANALOGS AS ALLOSTERIC MODULATORS OF MGLUR5 RECEPTORS
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Published in ACS chemical neuroscience (15.05.2019)
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Year of Publication 18.09.2012
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Year of Publication 18.09.2012
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Discovery of VU0409551/JNJ-46778212: An mGlu5 Positive Allosteric Modulator Clinical Candidate Targeting Schizophrenia
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Published in ACS medicinal chemistry letters (11.06.2015)
Published in ACS medicinal chemistry letters (11.06.2015)
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Published in Journal of medicinal chemistry (22.01.2015)
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Published in Bioorganic & medicinal chemistry letters (15.01.2016)
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Published in Bioorganic & medicinal chemistry letters (01.09.2015)
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Further optimization of the mGlu5 PAM clinical candidate VU0409551/JNJ-46778212: Progress and challenges towards a back-up compound
Zhou, Ya, Malosh, Chrysa, Conde-Ceide, Susana, Martínez-Viturro, Carlos Manuel, Alcázar, Jesus, Lavreysen, Hilde, Mackie, Claire, Bridges, Thomas M., Daniels, J. Scott, Niswender, Colleen M., Jones, Carrie K., Macdonald, Gregor J., Steckler, Thomas, Conn, P. Jeffrey, Stauffer, Shaun R., Bartolomé-Nebreda, José Manuel, Lindsley, Craig W.
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Published in Bioorganic & medicinal chemistry letters (01.09.2015)
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