Selective Cyclooxygenase-2 Inhibitors: Heteroaryl Modified 1,2-Diarylimidazoles Are Potent, Orally Active Antiinflammatory Agents
Khanna, Ish K, Yu, Yi, Huff, Renee M, Weier, Richard M, Xu, Xiangdong, Koszyk, Francis J, Collins, Paul W, Cogburn, J. Nita, Isakson, Peter C, Koboldt, Carol M, Masferrer, Jaime L, Perkins, William E, Seibert, Karen, Veenhuizen, Amy W, Yuan, Jinhua, Yang, Dai-Chang, Zhang, Yan Y
Published in Journal of medicinal chemistry (10.08.2000)
Published in Journal of medicinal chemistry (10.08.2000)
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Pharmacokinetics, Tissue Distribution, Metabolism, and Excretion of Celecoxib in Rats
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Published in Drug metabolism and disposition (01.05.2000)
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Published in Drug metabolism and disposition (01.05.2000)
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Synthesis and Biological Evaluation of the 1,5-Diarylpyrazole Class of Cyclooxygenase-2 Inhibitors: Identification of 4-[5-(4-Methylphenyl)-3- (trifluoromethyl)-1H-pyrazol-1-yl]benzenesulfonamide (SC-58635, Celecoxib)
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Published in Journal of medicinal chemistry (25.04.1997)
Published in Journal of medicinal chemistry (25.04.1997)
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Diarylspiro[2.4]heptenes as Orally Active, Highly Selective Cyclooxygenase-2 Inhibitors: Synthesis and Structure−Activity Relationships
Huang, Horng-Chih, Li, James J, Garland, Danny J, Chamberlain, Timothy S, Reinhard, Emily J, Manning, Robert E, Seibert, Karen, Koboldt, Carol M, Gregory, Susan A, Anderson, Gary D, Veenhuizen, Amy W, Zhang, Yan, Perkins, William E, Burton, Earl G, Cogburn, J. Nita, Isakson, Peter C, Reitz, David B
Published in Journal of medicinal chemistry (05.01.1996)
Published in Journal of medicinal chemistry (05.01.1996)
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Simultaneous sulfation of endogenous chondroitin sulfate and chondroitin-derived oligosaccharides. Studies with separate 4-sulfating and 6-sulfating microsomal systems
Sugumaran, G, Cogburn, J N, Silbert, J E
Published in The Journal of biological chemistry (25.09.1986)
Published in The Journal of biological chemistry (25.09.1986)
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Synthesis and biological evaluation of the 1,5-diarylpyrazole class of cyclooxygenase-2 inhibitors: identification of 4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl]benze nesulfonamide (SC-58635, celecoxib)
Penning, T D, Talley, J J, Bertenshaw, S R, Carter, J S, Collins, P W, Docter, S, Graneto, M J, Lee, L F, Malecha, J W, Miyashiro, J M, Rogers, R S, Rogier, D J, Yu, S S, AndersonGD, Burton, E G, Cogburn, J N, Gregory, S A, Koboldt, C M, Perkins, W E, Seibert, K, Veenhuizen, A W, Zhang, Y Y, Isakson, P C
Published in Journal of medicinal chemistry (25.04.1997)
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Published in Journal of medicinal chemistry (25.04.1997)
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1,2-Diarylcyclopentenes as Selective Cyclooxygenase-2 Inhibitors and Orally Active Anti-inflammatory Agents
Li, James J, Anderson, Gary D, Burton, Earl G, Cogburn, J. Nita, Collins, Joe T, Garland, Danny J, Gregory, Susan A, Huang, Horng-Chih, Isakson, Peter C
Published in Journal of medicinal chemistry (01.10.1995)
Published in Journal of medicinal chemistry (01.10.1995)
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1,2-DIARYLCYCLOPENTENES AS SELECTIVE CYCLOOXYGENASE-2 INHIBITORS AND ORALLY-ACTIVE ANTIINFLAMMATORY AGENTS
LI, JJ, ANDERSON, GD, BURTON, EG, COGBURN, JN, COLLINS, JT, GARLAND, DJ, GREGORY, SA, HUANG, HC, ISAKSON, PC, KOBOLDT, CM, LOGUSCH, EW, NORTON, MB, PERKINS, WE, REINHARD, EJ, SEIBERT, K, VEENHUIZEN, AW, ZHANG, Y, REITZ, DB
Published in Journal of medicinal chemistry (27.10.1995)
Published in Journal of medicinal chemistry (27.10.1995)
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Increased proteoglycan synthesis following the differentiation of F9 embryonal carcinoma cells: Formation of a differentiation-specific proteoheparan sulfate
Baldwin, Clinton T., Silbert, Jeremiah E., Humphries, Donald E., Nita Cogburn, J., Smith, Barbara D.
Published in Matrix (Stuttgart) (01.11.1989)
Published in Matrix (Stuttgart) (01.11.1989)
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1,2-Diarylcyclopentenes as selective cyclooxygenase-2 inhibitors and orally active anti-inflammatory agents
Li, J J, Anderson, G D, Burton, E G, Cogburn, J N, Collins, J T, Garland, D J, Gregory, S A, Huang, H C, Isakson, P C, Koboldt, C M
Published in Journal of medicinal chemistry (27.10.1995)
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Published in Journal of medicinal chemistry (27.10.1995)
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Delivery device for a powder aerosol
WOODCOCK DEREK A, STANIFORTH JOHN N, DOCKHORN DOUGLAS R, PRATHER SUSAN J, MITCHELL EDGAR W, PRICE ROBERT, DOCKHORN ROBERT J, BYRNES JAMES A, COGBURN J. N, YOUNG PAUL M
Year of Publication 15.03.2007
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Year of Publication 15.03.2007
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Delivery device for a powder aerosol
WOODCOCK DEREK A, STANIFORTH JOHN N, DOCKHORN DOUGLAS R, PRATHER SUSAN J, MITCHELL EDGAR W, PRICE ROBERT, DOCKHORN ROBERT J, BYRNES JAMES A, COGBURN J. N, YOUNG PAUL M
Year of Publication 28.09.2006
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Year of Publication 28.09.2006
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