Syntheses of the opioid substructures 1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocine and 2,3,4,5-tetrahydro-1,5-methano-1H-2-benzazepine
Coe, Jotham W., Brooks, Paige R., Vetelino, Michael G., Bashore, Crystal G., Bianco, Krista, Flick, Andrew C.
Published in Tetrahedron letters (02.03.2011)
Published in Tetrahedron letters (02.03.2011)
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Convenient preparation of N-substituted indoles by modified Leimgruber-Batcho indole synthesis
Coe, Jotham W, Vetelino, Michael G, Bradlee, Michael J
Published in Tetrahedron letters (19.08.1996)
Published in Tetrahedron letters (19.08.1996)
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In pursuit of α4β2 nicotinic receptor partial agonists for smoking cessation: Carbon analogs of (−)-cytisine
Coe, Jotham W., Vetelino, Michael G., Bashore, Crystal G., Wirtz, Michael C., Brooks, Paige R., Arnold, Eric P., Lebel, Lorraine A., Fox, Carol B., Sands, Steven B., Davis, Thomas I., Schulz, David W., Rollema, Hans, Tingley, F. David, O’Neill, Brian T.
Published in Bioorganic & medicinal chemistry letters (15.06.2005)
Published in Bioorganic & medicinal chemistry letters (15.06.2005)
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Cyclopentadiene: The Impact of Storage Conditions on Thermal Stability
am Ende, David J, Whritenour, David C, Coe, Jotham W
Published in Organic process research & development (01.11.2007)
Published in Organic process research & development (01.11.2007)
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3,5-Bicyclic aryl piperidines: A novel class of α4β2 neuronal nicotinic receptor partial agonists for smoking cessation
Coe, Jotham W., Brooks, Paige R., Wirtz, Michael C., Bashore, Crystal G., Bianco, Krista E., Vetelino, Michael G., Arnold, Eric P., Lebel, Lorraine A., Fox, Carol B., Tingley, F. David, Schulz, David W., Davis, Thomas I., Sands, Steven B., Mansbach, Robert S., Rollema, Hans, O’Neill, Brian T.
Published in Bioorganic & medicinal chemistry letters (15.11.2005)
Published in Bioorganic & medicinal chemistry letters (15.11.2005)
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CD38의 헤테로아릴 아미드 억제제
FELSTEAD STEVE, VERDIN ERIC, NELSON FREDERICK R, VOLKMANN ROBERT A, PERRONE ROSALBA, SILVA ELENA, JACKSON MARGARET, COE JOTHAM W
Year of Publication 13.07.2023
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Year of Publication 13.07.2023
Patent
A novel series of [3.2.1] azabicyclic biaryl ethers as α3β4 and α6/4β4 nicotinic receptor agonists
Lowe, John A., DeNinno, Shari L., Coe, Jotham W., Zhang, Lei, Mente, Scot, Hurst, Raymond S., Mather, Robert J., Ward, Karen M., Shrikhande, Alka, Rollema, Hans, Johnson, David E., Horner, Weldon, Gorczyca, Roxanne, Tingley, F. David, Kozak, Rouba, Majchrzak, Mark J., Tritto, Theresa, Sadlier, Jen, Shaffer, Chris L., Ellerbrock, Brenda, Osgood, Sarah M., MacDougall, Mary C., McDowell, Laura L.
Published in Bioorganic & medicinal chemistry letters (15.08.2010)
Published in Bioorganic & medicinal chemistry letters (15.08.2010)
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Enantioselective Synthesis of Nicotinic Receptor Probe 7,8-Difluoro-1,2,3,4,5,6- hexahydro-1,5-methano-3-benzazocine
Bashore, Crystal G, Vetelino, Michael G, Wirtz, Michael C, Brooks, Paige R, Frost, Heather N, McDermott, Ruth E, Whritenour, David C, Ragan, John A, Rutherford, Jennifer L, Makowski, Teresa W, Brenek, Steven J, Coe, Jotham W
Published in Organic letters (21.12.2006)
Published in Organic letters (21.12.2006)
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Boron Trichloride/Tetra-n-Butylammonium Iodide: A Mild, Selective Combination Reagent for the Cleavage of Primary Alkyl Aryl Ethers
Brooks, Paige R, Wirtz, Michael C, Vetelino, Michael G, Rescek, Diane M, Woodworth, Graeme F, Morgan, Bradley P, Coe, Jotham W
Published in Journal of organic chemistry (24.12.1999)
Published in Journal of organic chemistry (24.12.1999)
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Journal Article
Varenicline: An α4β2 Nicotinic Receptor Partial Agonist for Smoking Cessation
Coe, Jotham W, Brooks, Paige R, Vetelino, Michael G, Wirtz, Michael C, Arnold, Eric P, Huang, Jianhua, Sands, Steven B, Davis, Thomas I, Lebel, Lorraine A, Fox, Carol B, Shrikhande, Alka, Heym, James H, Schaeffer, Eric, Rollema, Hans, Lu, Yi, Mansbach, Robert S, Chambers, Leslie K, Rovetti, Charles C, Schulz, David W, Tingley, F. David, O'Neill, Brian T
Published in Journal of medicinal chemistry (19.05.2005)
Published in Journal of medicinal chemistry (19.05.2005)
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Journal Article
Design considerations for chiral frustrated Lewis pairs: B/N FLPs derived from 3,5-bicyclic aryl piperidinesElectronic supplementary information (ESI) available: Spectral and crystallographic data. CCDC 1868691-1868693 for compounds: 12, 5 and 10, respectively. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c8dt04070b
Lam, Jolie, Sampaolesi, Susanna, LaFortune, James H. W, Coe, Jotham W, Stephan, Douglas W
Year of Publication 18.12.2018
Year of Publication 18.12.2018
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Journal Article
Correction to “Catalytic Enantioselective Synthesis of a cis-β-Boronyl Cyclobutylcarboxyester Scaffold and Its Highly Diastereoselective Nickel/Photoredox Dual-Catalyzed Csp3–Csp2 Cross-Coupling to Access Elusive trans-β-Aryl/Heteroaryl Cyclobutylcarboxyesters”
Nguyen, Kevin, Clement, Helen A, Bernier, Louise, Coe, Jotham W, Farrell, William, Helal, Christopher J, Reese, Matthew R, Sach, Neal W, Lee, Jack C, Hall, Dennis G
Published in ACS catalysis (16.04.2021)
Published in ACS catalysis (16.04.2021)
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Journal Article
Correction to “Catalytic Enantioselective Synthesis of a cis -β-Boronyl Cyclobutylcarboxyester Scaffold and Its Highly Diastereoselective Nickel/Photoredox Dual-Catalyzed Csp 3 –Csp 2 Cross-Coupling to Access Elusive trans -β-Aryl/Heteroaryl Cyclobutylcarboxyesters”
Nguyen, Kevin, Clement, Helen A., Bernier, Louise, Coe, Jotham W., Farrell, William, Helal, Christopher J., Reese, Matthew R., Sach, Neal W., Lee, Jack C., Hall, Dennis G.
Published in ACS catalysis (16.04.2021)
Published in ACS catalysis (16.04.2021)
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Journal Article
Catalytic Enantioselective Synthesis of a cis-β-Boronyl Cyclobutylcarboxyester Scaffold and Its Highly Diastereoselective Nickel/Photoredox Dual-Catalyzed Csp3–Csp2 Cross-Coupling to Access Elusive trans-β-Aryl/Heteroaryl Cyclobutylcarboxyesters
Nguyen, Kevin, Clement, Helen A, Bernier, Louise, Coe, Jotham W, Farrell, William, Helal, Christopher J, Reese, Matthew R, Sach, Neal W, Lee, Jack C, Hall, Dennis G
Published in ACS catalysis (01.01.2021)
Published in ACS catalysis (01.01.2021)
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Journal Article
Catalytic Enantioselective Synthesis of a cis -β-Boronyl Cyclobutylcarboxyester Scaffold and Its Highly Diastereoselective Nickel/Photoredox Dual-Catalyzed Csp 3 –Csp 2 Cross-Coupling to Access Elusive trans -β-Aryl/Heteroaryl Cyclobutylcarboxyesters
Nguyen, Kevin, Clement, Helen A., Bernier, Louise, Coe, Jotham W., Farrell, William, Helal, Christopher J., Reese, Matthew R., Sach, Neal W., Lee, Jack C., Hall, Dennis G.
Published in ACS catalysis (01.01.2021)
Published in ACS catalysis (01.01.2021)
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