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Published in Journal of medicinal chemistry (21.11.1997)
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Structure of recombinant human rheumatoid arthritic synovial fluid phospholipase A2 at 2.2 A resolution
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Published in Journal of medicinal chemistry (24.10.1997)
Published in Journal of medicinal chemistry (24.10.1997)
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The crystal structures of human α-thrombin complexed with active site-directed diamino benzo[b]thiophene derivatives: A binding mode for a structurally novel class of inhibitors
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Published in Protein science (01.01.2000)
Published in Protein science (01.01.2000)
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The crystal structure of human α‐thrombin complexed with LY178550, a nonpeptidyl, active site‐directed inhibitor
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Published in Protein science (01.07.1997)
Published in Protein science (01.07.1997)
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Dibasic benzo[ b]thiophene derivatives as a novel class of active site directed thrombin inhibitors. 2. Exploring interactions at the proximal (S 2) binding site
Sall, Daniel J., Briggs, Stephen L., Chirgadze, Nickolay Y., Clawson, David K., Gifford-Moore, Donetta S., Klimkowski, Valentine J., McCowan, Jefferson R., Smith, Gerald F., Wikel, James H.
Published in Bioorganic & medicinal chemistry letters (22.09.1998)
Published in Bioorganic & medicinal chemistry letters (22.09.1998)
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Dibasic benzo[ b]thiophene derivatives as a novel class of active site directed thrombin inhibitors: 2: sidechain optimization and demonstration of in vivo efficacy
Zhang, Minsheng, Bailey, Dianna L., Bastian, Jolie A., Briggs, Stephen L., Chirgadze, Nickolay Y., Clawson, David K., Denney, Michael L., Gifford-Moore, Donetta S., Harper, Richard W., Johnson, Lea M., Klimkowski, Valentine J., Kohn, Todd J., Lin, Ho-Shen, McCowan, Jefferson R., Richett, Michael E., Sall, Daniel J., Smith, Amy J., Smith, Gerald F., Snyder, David W., Takeuchi, Kumiko, Utterback, Barbara G., Yan, Sau-Chi B.
Published in Bioorganic & medicinal chemistry letters (08.03.1999)
Published in Bioorganic & medicinal chemistry letters (08.03.1999)
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Dihydropyrrolopyrazole Transforming Growth Factor-β Type I Receptor Kinase Domain Inhibitors: A Novel Benzimidazole Series with Selectivity versus Transforming Growth Factor-β Type II Receptor Kinase and Mixed Lineage Kinase-7
Li, Hong-yu, Wang, Yan, Heap, Charles R, King, Chi-Hsin R, Mundla, Sreenivasa R, Voss, Matthew, Clawson, David K, Yan, Lei, Campbell, Robert M, Anderson, Bryan D, Wagner, Jill R, Britt, Karen, Lu, Ku X, McMillen, William T, Yingling, Jonathan M
Published in Journal of medicinal chemistry (23.03.2006)
Published in Journal of medicinal chemistry (23.03.2006)
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Indole Inhibitors of Human Nonpancreatic Secretory Phospholipase A2. 1. Indole-3-acetamides
Dillard, Robert D., Bach, Nicholas J., Draheim, Susan E., Berry, Dennis R., Carlson, Donald G., Chirgadze, Nickolay Y., Clawson, David K., Hartley, Lawrence W., Johnson, Lea M., Jones, Noel D., McKinney, Emma R., Mihelich, Edward D., Olkowski, Jennifer L., Schevitz, Richard W., Smith, Amy C., Snyder, David W., Sommers, Cynthia D., Wery, Jean-Pierre
Published in Journal of medicinal chemistry (20.12.1996)
Published in Journal of medicinal chemistry (20.12.1996)
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The deep posterior compartmental syndrome of the leg
Matsen, 3rd, F A, Clawson, D K
Published in Journal of bone and joint surgery. American volume (01.01.1975)
Published in Journal of bone and joint surgery. American volume (01.01.1975)
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Indole Inhibitors of Human Nonpancreatic Secretory Phospholipase A2. 3. Indole-3-glyoxamides
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Published in Journal of medicinal chemistry (20.12.1996)
Published in Journal of medicinal chemistry (20.12.1996)
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A convenient synthesis of 9,9-dialkyl-9,10-dihydroanthracenes and 10,10-dialkylanthrones: silicon-mediated regioselective dialkylation of 9,10-dihydroanthracene
Dhar, Raj K, Clawson, D. K, Fronczek, Frank R, Rabideau, Peter W
Published in Journal of organic chemistry (01.05.1992)
Published in Journal of organic chemistry (01.05.1992)
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