Annexin A2 is a natural extrahepatic inhibitor of the PCSK9-induced LDL receptor degradation
Seidah, Nabil G, Poirier, Steve, Denis, Maxime, Parker, Rex, Miao, Bowman, Mapelli, Claudio, Prat, Annik, Wassef, Hanny, Davignon, Jean, Hajjar, Katherine A, Mayer, Gaétan
Published in PloS one (27.07.2012)
Published in PloS one (27.07.2012)
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Journal Article
An optimized agonist peptide of protease-activated receptor 4 and its use in a validated platelet-aggregation assay
Yang, Jing, Mapelli, Claudio, Wang, Zhaoqing, Sum, Chi Shing, Hua, Ji, Lawrence, R. Michael, Ni, Yan, Seiffert, Dietmar A.
Published in Platelets (Edinburgh) (03.10.2022)
Published in Platelets (Edinburgh) (03.10.2022)
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Journal Article
Mcl-1 antagonism is a potential therapeutic strategy in a subset of solid cancers
Modugno, Michele, Banfi, Patrizia, Gasparri, Fabio, Borzilleri, Robert, Carter, Percy, Cornelius, Lyndon, Gottardis, Marco, Lee, Ving, Mapelli, Claudio, Naglich, Joseph G., Tebben, Andrew, Vite, Gregory, Pastori, Wilma, Albanese, Clara, Corti, Emiliana, Ballinari, Dario, Galvani, Arturo
Published in Experimental cell research (15.03.2015)
Published in Experimental cell research (15.03.2015)
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Journal Article
Formation of α-chiral centers by asymmetric β-C(sp3)-H arylation, alkenylation, and alkynylation
Wu, Qing-Feng, Shen, Peng-Xiang, He, Jian, Wang, Xiao-Bing, Zhang, Forrest, Shao, Qian, Zhu, Ru-Yi, Mapelli, Claudio, Qiao, Jennifer X, Poss, Michael A, Yu, Jin-Quan
Published in Science (American Association for the Advancement of Science) (03.02.2017)
Published in Science (American Association for the Advancement of Science) (03.02.2017)
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Journal Article
Omomyc Reveals New Mechanisms To Inhibit the MYC Oncogene
Demma, Mark J., Mapelli, Claudio, Sun, Angie, Bodea, Smaranda, Ruprecht, Benjamin, Javaid, Sarah, Wiswell, Derek, Muise, Eric, Chen, Shiying, Zelina, John, Orvieto, Federica, Santoprete, Alessia, Altezza, Simona, Tucci, Federica, Escandon, Enrique, Hall, Brian, Ray, Kallol, Walji, Abbas, O'Neil, Jennifer
Published in Molecular and cellular biology (01.11.2019)
Published in Molecular and cellular biology (01.11.2019)
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Journal Article
Inhibition of Myc transcriptional activity by a mini‐protein based upon Mxd1
Demma, Mark J., Hohn, Michael J., Sun, Angie, Mapelli, Claudio, Hall, Brian, Walji, Abbas, O'Neil, Jennifer
Published in FEBS letters (01.05.2020)
Published in FEBS letters (01.05.2020)
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Journal Article
Ligand-Enabled β‑C–H Arylation of α‑Amino Acids Using a Simple and Practical Auxiliary
Chen, Gang, Shigenari, Toshihiko, Jain, Pankaj, Zhang, Zhipeng, Jin, Zhong, He, Jian, Li, Suhua, Mapelli, Claudio, Miller, Michael M, Poss, Michael A, Scola, Paul M, Yeung, Kap-Sun, Yu, Jin-Quan
Published in Journal of the American Chemical Society (11.03.2015)
Published in Journal of the American Chemical Society (11.03.2015)
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Journal Article
Process Development of a Macrocyclic Peptide Inhibitor of PD-L1
Mukherjee, Subha, Rogers, Amanda, Creech, Gardner, Hang, Chao, Ramirez, Antonio, Dummeldinger, Michael, Brueggemeier, Shawn, Mapelli, Claudio, Zaretsky, Serge, Huang, Masano, Black, Regina, Peddicord, Michael B., Cuniere, Nicolas, Kempson, James, Pawluczyk, Joseph, Allen, Martin, Parsons, Rodney, Sfouggatakis, Chris
Published in Journal of organic chemistry (17.05.2024)
Published in Journal of organic chemistry (17.05.2024)
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Journal Article
Ultra-high-throughput SPE-MALDI workflow: Blueprint for efficient purification and screening of peptide libraries
Bennett, Raffeal, Pirrone, Gregory F., Nowak, Timothy, Mukherjee, Debopreeti, Shchurik, Vladimir, Mapelli, Claudio, Hickey, Jennifer L., Regalado, Erik L., Mangion, Ian, Makarov, Alexey A.
Published in Analytica chimica acta (15.01.2021)
Published in Analytica chimica acta (15.01.2021)
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Journal Article
Orientation of Peptide Fragments from Sos Proteins Bound to the N-Terminal SH3 Domain of Grb2 Determined by NMR Spectroscopy
Wittekind, Michael, Mapelli, Claudio, Farmer, Bennett T, Suen, Ki-Ling, Goldfarb, Valentina, Tsao, Jonglin, Lavoie, Thomas, Barbacid, Mariano, Meyers, Chester A, Mueller, Luciano
Published in Biochemistry (Easton) (01.11.1994)
Published in Biochemistry (Easton) (01.11.1994)
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Journal Article
Multiple Synthetic Routes to the Mini-Protein Omomyc and Coiled-Coil Domain Truncations
Brown, Zachary Z, Mapelli, Claudio, Farasat, Iman, Shoultz, Alycia V, Johnson, Scott A, Orvieto, Federica, Santoprete, Alessia, Bianchi, Elisabetta, McCracken, Amy Bittner, Chen, Kuanchang, Zhu, Xiaohong, Demma, Mark J, Lacey, Brian M, Canada, Keith A, Garbaccio, Robert M, O’Neil, Jennifer, Walji, Abbas
Published in Journal of organic chemistry (07.02.2020)
Published in Journal of organic chemistry (07.02.2020)
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Journal Article
Formation of [alpha]-chiral centers by asymmetric [beta]-C(sp3)-H arylation, alkenylation, and alkynylation
Qing-Feng, Wu, Peng-Xiang, Shen, He, Jian, Xiao-Bing, Wang, Zhang, rest, Shao, Qian, Ru-Yi Zhu, Mapelli, Claudio, Qiao, Jennifer X, Poss, Michael A, Jin-Quan, Yu
Published in Science (American Association for the Advancement of Science) (03.02.2017)
Published in Science (American Association for the Advancement of Science) (03.02.2017)
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Journal Article
Formation of a-chiral centers by asymmetric β-C(sp³)–H arylation, alkenylation, and alkynylation
Wu, Qing-Feng, Shen, Peng-Xiang, He, Jian, Wang, Xiao-Bing, Zhang, Forrest, Shao, Qian, Zhu, Ru-Yi, Mapelli, Claudio, Qiao, Jennifer X., Poss, Michael A., Yu, Jin-Quan
Published in Science (American Association for the Advancement of Science) (03.02.2017)
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Published in Science (American Association for the Advancement of Science) (03.02.2017)
Journal Article
Eleven Amino Acid Glucagon-like Peptide-1 Receptor Agonists with Antidiabetic Activity
Mapelli, Claudio, Natarajan, Sesha I, Meyer, Jean-Philippe, Bastos, Margarita M, Bernatowicz, Michael S, Lee, Ving G, Pluscec, Jelka, Riexinger, Douglas J, Sieber-McMaster, Ellen S, Constantine, Keith L, Smith-Monroy, Constance A, Golla, Rajasree, Ma, Zhengping, Longhi, Daniel A, Shi, Dan, Xin, Li, Taylor, Joseph R, Koplowitz, Barry, Chi, Cecilia L, Khanna, Ashish, Robinson, Gordon W, Seethala, Ramakrishna, Antal-Zimanyi, Ildiko A, Stoffel, Robert H, Han, Songping, Whaley, Jean M, Huang, Christine S, Krupinski, John, Ewing, William R
Published in Journal of medicinal chemistry (10.12.2009)
Published in Journal of medicinal chemistry (10.12.2009)
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Journal Article
Synthesis of racemic (E)- and (Z)-2,3-methanotyrosine: new cyclopropane analogs of tyrosine
Mapelli, Claudio, Turocy, Gregory, Switzer, Frank L, Stammer, Charles H
Published in Journal of organic chemistry (01.01.1989)
Published in Journal of organic chemistry (01.01.1989)
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Journal Article
P2‐008: Modified Aβ42 peptides as immunoassay calibrators improve the measurement of native Aβ42 peptides in clinical samples
Berisha, Flora, Wong, Oitak (Allen), Mapelli, Claudio, Witmer, Mark, Neely, Robert, Zhang, Yan, Simon, Adam, Desilva, Binodh, Rhyne, Paul
Published in Alzheimer's & dementia (01.07.2012)
Published in Alzheimer's & dementia (01.07.2012)
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Journal Article
Modified Aβ42 peptides as immunoassay calibrators improve the measurement of native Aβ42 peptides in clinical samples
Berisha, Flora, Wong, Oitak (Allen), Mapelli, Claudio, Witmer, Mark, Neely, Robert, Zhang, Yan, Simon, Adam, Desilva, Binodh, Rhyne, Paul
Published in Alzheimer's & dementia (01.07.2012)
Published in Alzheimer's & dementia (01.07.2012)
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Journal Article
Synthesis of a stable isotopically labeled universal surrogate peptide for use as an internal standard in LC-MS/MS bioanalysis of human IgG and Fc-fusion protein drug candidates
Voronin, Kimberly, Allentoff, Alban J., Bonacorsi Jr, Samuel J., Mapelli, Claudio, Gong, Sharon X., Lee, Ving, Riexinger, Douglas, Sanghvi, Nishith, Jiang, Hao, Zeng, Jianing
Published in Journal of labelled compounds & radiopharmaceuticals (01.07.2014)
Published in Journal of labelled compounds & radiopharmaceuticals (01.07.2014)
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Journal Article
Identification of potent 11mer Glucagon-Like Peptide-1 Receptor agonist peptides with novel C-terminal amino acids: Homohomophenylalanine analogs
Haque, Tasir S., Lee, Ving G., Riexinger, Douglas, Lei, Ming, Malmstrom, Sarah, Xin, Li, Han, Songping, Mapelli, Claudio, Cooper, Christopher B., Zhang, Ge, Ewing, William R., Krupinski, John
Published in Peptides (New York, N.Y. : 1980) (01.05.2010)
Published in Peptides (New York, N.Y. : 1980) (01.05.2010)
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Journal Article
In vitro Proteolytic Activity and Active‐Site Identification of the Human Cytomegalovirus Protease
Stevens, John T., Mapelli, Claudio, Tsao, Jonglin, Hail, Mark, O'Boyle, Donald, Weinheimer, Steven P., Diianni, Carolyn L.
Published in European journal of biochemistry (01.12.1994)
Published in European journal of biochemistry (01.12.1994)
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