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Published in Angewandte Chemie International Edition (04.06.2018)
Published in Angewandte Chemie International Edition (04.06.2018)
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Enantiospecific and regioselective opening of 2-alkyl nosylaziridines by indoles mediated by boron trifluoride. Application to a practical synthesis of a GnRH antagonist
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Published in Tetrahedron: asymmetry (14.11.2003)
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페녹시 디아미노피리미딘 화합물의 신규 합성 방법
DI MASO MICHAEL JAMES, LEE ALFRED Y, CHUNG JOHN Y.L, BASU KALLOL, MALONEY KEVIN M, DESMOND RICHARD, LEHNHERR DAN, REN HONG, WEISEL MARK, LARPENT PATRICK, PENG FENG, ZHANG SIWEI, HUMPHREY GUY R
Year of Publication 14.01.2021
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Year of Publication 14.01.2021
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Practical chemoenzymatic synthesis of a 3-pyridylethanolamino β3 adrenergic receptor agonist
Chung, John Y.L, Ho, Guo-Jie, Chartrain, Michel, Roberge, Chris, Zhao, Dalian, Leazer, John, Farr, Roger, Robbins, Michael, Emerson, Kateeta, Mathre, David J, McNamara, James M, Hughes, David L, Grabowski, Edward J.J, Reider, Paul J
Published in Tetrahedron letters (10.09.1999)
Published in Tetrahedron letters (10.09.1999)
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Diastereoselective FeCl3·6H2O/NaBH4 Reduction of Oxime Ether for the Synthesis of β‑Lactamase Inhibitor Relebactam
Chung, John Y. L, Meng, Dongfang, Shevlin, Michael, Gudipati, Venugopal, Chen, Qinghao, Liu, Yizhou, Lam, Yu-hong, Dumas, Aaron, Scott, Jeremy, Tu, Qiang, Xu, Feng
Published in Journal of organic chemistry (17.01.2020)
Published in Journal of organic chemistry (17.01.2020)
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Kilogram-Scale Synthesis of 2′‑C‑Methyl-arabino-Uridine from Uridine via Dynamic Selective Dipivaloylation
Chung, John Y. L, Kassim, Amude M, Simmons, Bryon, Davis, Tyler A, Song, Zhiguo J, Limanto, John, Dalby, Stephen M, He, Cyndi Q, Calabria, Ralph, Wright, Timothy J, Campeau, Louis-Charles
Published in Organic process research & development (18.03.2022)
Published in Organic process research & development (18.03.2022)
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Efficient synthesis of antiviral agent uprifosbuvir enabled by new synthetic methods
Klapars, Artis, Chung, John Y. L, Limanto, John, Calabria, Ralph, Campeau, Louis-Charles, Campos, Kevin R, Chen, Wenyong, Dalby, Stephen M, Davis, Tyler A, DiRocco, Daniel A, Hyde, Alan M, Kassim, Amude M, Larsen, Mona Utne, Liu, Guiquan, Maligres, Peter E, Moment, Aaron, Peng, Feng, Ruck, Rebecca T, Shevlin, Michael, Simmons, Bryon L, Song, Zhiguo Jake, Tan, Lushi, Wright, Timothy J, Zultanski, Susan L
Published in Chemical science (Cambridge) (07.07.2021)
Published in Chemical science (Cambridge) (07.07.2021)
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Evolution of a Manufacturing Route to Omarigliptin, A Long-Acting DPP‑4 Inhibitor for the Treatment of Type 2 Diabetes
Chung, John Y. L, Scott, Jeremy P, Anderson, Camille, Bishop, Brian, Bremeyer, Nadine, Cao, Yang, Chen, Qinghao, Dunn, Robert, Kassim, Amude, Lieberman, David, Moment, Aaron J, Sheen, Faye, Zacuto, Michael
Published in Organic process research & development (20.11.2015)
Published in Organic process research & development (20.11.2015)
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Development of a Commercial Manufacturing Route to 2‑Fluoroadenine, The Key Unnatural Nucleobase of Islatravir
Hong, Cynthia M, Xu, Yingju, Chung, John Y. L, Schultz, Danielle M, Weisel, Mark, Varsolona, Richard J, Zhong, Yong-Li, Purohit, Akasha K, He, Cyndi Q, Gauthier, Donald R, Humphrey, Guy R, Maloney, Kevin M, Lévesque, François, Wang, Zhixun, Whittaker, Aaron M, Sirota, Eric, McMullen, Jonathan P
Published in Organic process research & development (19.03.2021)
Published in Organic process research & development (19.03.2021)
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Development of a Green and Sustainable Manufacturing Process for Gefapixant Citrate (MK-7264) Part 3: Development of a One-Pot Formylation–Cyclization Sequence to the Diaminopyrimidine Core
Basu, Kallol, Lehnherr, Dan, Martin, Gary E, Desmond, Richard A, Lam, Yu-hong, Peng, Feng, Chung, John Y. L, Arvary, Rebecca A, Zompa, Michael A, Zhang, Si-Wei, Liu, Jinchu, Dance, Zachary E. X, Larpent, Patrick, Cohen, Ryan D, Guzman, Francisco J, Rogus, Nicholas J, Di Maso, Michael J, Ren, Hong, Maloney, Kevin M
Published in Organic process research & development (20.11.2020)
Published in Organic process research & development (20.11.2020)
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Asymmetric Formal Synthesis of the Long-Acting DPP-4 Inhibitor Omarigliptin
Peng, Feng, Chen, Yonggang, Chen, Cheng-yi, Dormer, Peter G, Kassim, Amude, McLaughlin, Mark, Reamer, Robert A, Sherer, Edward C, Song, Zhiguo J, Tan, Lushi, Tudge, Matthew T, Wan, Baoqiang, Chung, John Y. L
Published in Journal of organic chemistry (01.09.2017)
Published in Journal of organic chemistry (01.09.2017)
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Asymmetric Synthesis of cis-2,5-Disubstituted Pyrrolidine, the Core Scaffold of β3‑AR Agonists
Xu, Feng, Chung, John Y. L, Moore, Jeffery C, Liu, Zhuqing, Yoshikawa, Naoki, Hoerrner, R. Scott, Lee, Jaemoon, Royzen, Maksim, Cleator, Ed, Gibson, Andrew G, Dunn, Robert, Maloney, Kevin M, Alam, Mahbub, Goodyear, Adrian, Lynch, Joseph, Yasuda, Nobuyashi, Devine, Paul N
Published in Organic letters (15.03.2013)
Published in Organic letters (15.03.2013)
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Asymmetric Synthesis of Cyclic Indole Aminals via 1,3-Stereoinduction
Li, Hongmei, Chen, Cheng-yi, Nguyen, Hoa, Cohen, Ryan, Maligres, Peter E, Yasuda, Nobuyoshi, Mangion, Ian, Zavialov, Ilia, Reibarkh, Mikhail, Chung, John Y. L
Published in Journal of organic chemistry (19.09.2014)
Published in Journal of organic chemistry (19.09.2014)
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Synthesis of ((3R,6R)‑6-Methylpiperidin-3-yl)methanol via Biocatalytic Transamination and Crystallization-Induced Dynamic Resolution
Chung, John Y. L, Marcune, Benjamin, Strotman, Hallena R, Petrova, Rositza I, Moore, Jeffrey C, Dormer, Peter G
Published in Organic process research & development (16.10.2015)
Published in Organic process research & development (16.10.2015)
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Unusual Pyrimidine Participation: Efficient Stereoselective Synthesis of Potent Dual Orexin Receptor Antagonist MK-6096
Chung, John Y. L, Zhong, Yong-Li, Maloney, Kevin M, Reamer, Robert A, Moore, Jeffrey C, Strotman, Hallena, Kalinin, Alexei, Feng, Ronnie, Strotman, Neil A, Xiang, Bangping, Yasuda, Nobuyoshi
Published in Organic letters (21.11.2014)
Published in Organic letters (21.11.2014)
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Diastereoselective Friedel−Crafts Alkylation of Indoles with Chiral α-Phenyl Benzylic Cations. Asymmetric Synthesis of Anti-1,1,2-Triarylalkanes
Chung, John Y. L, Mancheno, Danny, Dormer, Peter G, Variankaval, Narayan, Ball, Richard G, Tsou, Nancy N
Published in Organic letters (17.07.2008)
Published in Organic letters (17.07.2008)
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Asymmetric Synthesis of a Glucagon Receptor Antagonist via Friedel–Crafts Alkylation of Indole with Chiral α‑Phenyl Benzyl Cation
Chung, John Y. L, Steinhuebel, Dietrich, Krska, Shane W, Hartner, Fred W, Cai, Chaoxian, Rosen, Jonathan, Mancheno, Danny E, Pei, Tao, DiMichele, Lisa, Ball, Richard G, Chen, Cheng-yi, Tan, Lushi, Alorati, Antony D, Brewer, Sarah E, Scott, Jeremy P
Published in Organic process research & development (16.11.2012)
Published in Organic process research & development (16.11.2012)
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