New Inhibitors of Glycogen Phosphorylase as Potential Antidiabetic Agents
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Structural Studies on Phospho-CDK2/Cyclin A Bound to Nitrate, a Transition State Analogue: Implications for the Protein Kinase Mechanism
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Published in Proteins, structure, function, and bioinformatics (01.12.2005)
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Crystallographic Studies on α- and β-D-glucopyranosyl Formamide Analogues, Inhibitors of Glycogen Phosphorylase
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Kinetic and crystallographic studies on 2‐(β‐D‐glucopyranosyl)‐5‐methyl‐1, 3, 4‐oxadiazole, ‐benzothiazole, and ‐benzimidazole, inhibitors of muscle glycogen phosphorylase b. Evidence for a new binding site
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Published in Protein science (01.04.2005)
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Kinetic and crystallographic studies of glucopyranose spirohydantoin and glucopyranosylamine analogs inhibitors of glycogen phosphorylase
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Published in Proteins, structure, function, and bioinformatics (01.12.2005)
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High‐resolution crystal structures of ribonuclease A complexed with adenylic and uridylic nucleotide inhibitors. Implications for structure‐based design of ribonucleolytic inhibitors
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Published in Protein science (01.11.2003)
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Crystallographic studies on acyl ureas, a new class of glycogen phosphorylase inhibitors, as potential antidiabetic drugs
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Published in Protein science (01.07.2005)
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Indirubin and indigo analogues inhibit glycogen phosphorylase b by binding at the inhibitor or/and allosteric site
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Published in Acta crystallographica. Section A, Foundations of crystallography (26.08.2004)
Published in Acta crystallographica. Section A, Foundations of crystallography (26.08.2004)
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Crystallographic studies on acyl ureas, a new class of inhibitors of glycogen phosphorylase
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Published in Acta crystallographica. Section A, Foundations of crystallography (23.08.2005)
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Published in Bioorganic & medicinal chemistry (2006)
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Binding of β- d-glucopyranosyl bismethoxyphosphoramidate to glycogen phosphorylase b: kinetic and crystallographic studies
Chrysina, Evangelia D., Kosmopoulou, Magda N., Kardakaris, Rozina, Bischler, Nicolas, Leonidas, Demetres D., Kannan, Thanukrishnan, Loganathan, Duraikkannu, Oikonomakos, Nikos G.
Published in Bioorganic & medicinal chemistry (01.02.2005)
Published in Bioorganic & medicinal chemistry (01.02.2005)
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The structure of glycogen phosphorylase b with an alkyldihydropyridine-dicarboxylic acid compound, a novel and potent inhibitor
Zographos, Spyros E, Oikonomakos, Nikos G, Tsitsanou, Katerina E, Leonidas, Demetrios D, Chrysina, Evangelia D, Skamnaki, Vicky T, Bischoff, Hilmar, Goldmann, Siegfried, Watson, Kimberly A, Johnson, Louise N
Published in Structure (London) (15.11.1997)
Published in Structure (London) (15.11.1997)
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Binding of the potential antitumour agent indirubin-5-sulphonate at the inhibitor site of rabbit muscle glycogen phosphorylase b. Comparison with ligand binding to pCDK2-cyclin A complex
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Published in European journal of biochemistry (01.06.2004)
Published in European journal of biochemistry (01.06.2004)
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