One-Pot Synthesis of Symmetrical and Unsymmetrical Bisarylethynes by a Modification of the Sonogashira Coupling Reaction
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Discovery of Clinical Candidate 4-[2-(5-Amino-1H-pyrazol-4-yl)-4-chlorophenoxy]-5-chloro-2-fluoro-N-1,3-thiazol-4-ylbenzenesulfonamide (PF-05089771): Design and Optimization of Diaryl Ether Aryl Sulfonamides as Selective Inhibitors of Na V 1.7
Swain, Nigel A, Batchelor, Dave, Beaudoin, Serge, Bechle, Bruce M, Bradley, Paul A, Brown, Alan D, Brown, Bruce, Butcher, Ken J, Butt, Richard P, Chapman, Mark L, Denton, Stephen, Ellis, David, Galan, Sebastien R G, Gaulier, Steven M, Greener, Ben S, de Groot, Marcel J, Glossop, Mel S, Gurrell, Ian K, Hannam, Jo, Johnson, Matthew S, Lin, Zhixin, Markworth, Christopher J, Marron, Brian E, Millan, David S, Nakagawa, Shoko, Pike, Andy, Printzenhoff, David, Rawson, David J, Ransley, Sarah J, Reister, Steven M, Sasaki, Kosuke, Storer, R Ian, Stupple, Paul A, West, Christopher W
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Swain, Nigel. A., Batchelor, Dave, Beaudoin, Serge, Bechle, Bruce M., Bradley, Paul A., Brown, Alan D., Brown, Bruce, Butcher, Kent J., Butt, Richard P., Chapman, Mark L., Denton, Stephen, Ellis, David, Galan, Sebastien R. G., Gaulier, Steven M., Greener, Ben S., de Groot, Marcel J., Glossop, Mel S., Gurrell, Ian K., Hannan, Jo, Johnson, Matthew S., Lin, Zhixin, Markworth, Christopher J., Marron, Brian E., Milan, David S., Nakaawa, Shoko, Pike, Andy, Printzephoff, David, Rawson, David J., Ransley, Sarah J., Reister, Steven M., Sasaki, Kosuke, Storer, R. Ian, Stupple, Paul A., West, Christopher W.
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Year of Publication 25.12.2008
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Year of Publication 25.12.2008
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One-Pot Synthesis of Symmetrical and Unsymmetrical Bisarylethynes by a Modification of the Sonogashira Coupling Reaction
Mio, Matthew J., Kopel, Lucas C., Braun, Julia B., Gadzikwa, Tendai L., Hull, Kami L., Brisbois, Ronald G., Markworth, Christopher J., Grieco, Paul A.
Published in ChemInform (21.01.2003)
Published in ChemInform (21.01.2003)
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Year of Publication 01.08.2007
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INDOLE, BENZIMIDAZOLE, AND BENZOLACTAM BORONIC ACID COMPOUNDS, ANALOGS THEREOF AND METHODS OF USE THEREOF
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Year of Publication 12.02.2009
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