Peripheral selectivity of the novel cannabinoid receptor antagonist TM38837 in healthy subjects
Klumpers, Linda E., Fridberg, Marianne, Kam, Marieke L., Little, Paul B., Jensen, Niels Ole, Kleinloog, Hendrik D., Elling, Christian E., Gerven, Joop M. A.
Published in British journal of clinical pharmacology (01.12.2013)
Published in British journal of clinical pharmacology (01.12.2013)
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Metal Ion Site Engineering Indicates a Global Toggle Switch Model for Seven-transmembrane Receptor Activation
Elling, Christian E., Frimurer, Thomas M., Gerlach, Lars-Ole, Jorgensen, Rasmus, Holst, Birgitte, Schwartz, Thue W.
Published in The Journal of biological chemistry (23.06.2006)
Published in The Journal of biological chemistry (23.06.2006)
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Metal Ion-mediated Agonism and Agonist Enhancement in Melanocortin MC1 and MC4 Receptors
Holst, Birgitte, Elling, Christian E., Schwartz, Thue W.
Published in The Journal of biological chemistry (06.12.2002)
Published in The Journal of biological chemistry (06.12.2002)
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Characterization of G-Protein Coupled Receptor Kinase Interaction with the Neurokinin-1 Receptor Using Bioluminescence Resonance Energy Transfer
Jorgensen, Rasmus, Holliday, Nicholas D, Hansen, Jakob L, Vrecl, Milka, Heding, Anders, Schwartz, Thue W, Elling, Christian E
Published in Molecular pharmacology (01.02.2008)
Published in Molecular pharmacology (01.02.2008)
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Efficacy in diet-induced obese mice of the hepatotropic, peripheral cannabinoid 1 receptor inverse agonist TM38837
Cooper, Martin E, Nørregaard, Pia K, Högberg, Thomas, Andersson, Gunnar, Receveur, Jean-Marie, Linget, Jean-Michel, Elling, Christian E
Published in British journal of pharmacology (01.10.2024)
Published in British journal of pharmacology (01.10.2024)
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Journal Article
Conversion of antagonist-binding site to metal-ion site in the tachykinin NK-1 receptor
Elling, Christian E, Nielsen, Søren Møller, Schwartz, Thue W
Published in Nature (London) (02.03.1995)
Published in Nature (London) (02.03.1995)
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Journal Article
Long-Acting Lipidated Analogue of Human Pancreatic Polypeptide Is Slowly Released into Circulation
Bellmann-Sickert, Kathrin, Elling, Christian E, Madsen, Andreas N, Little, Paul B, Lundgren, Karsten, Gerlach, Lars-Ole, Bergmann, Ralf, Holst, Birgitte, Schwartz, Thue W, Beck-Sickinger, Annette G
Published in Journal of medicinal chemistry (28.04.2011)
Published in Journal of medicinal chemistry (28.04.2011)
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Low brain CB1 receptor occupancy by a second generation CB1 receptor antagonist TM38837 in comparison with rimonabant in nonhuman primates: A PET study
Takano, Akihiro, Gulyás, Balázs, Varnäs, Katarina, Little, Paul Brian, Noerregaard, Pia K., Jensen, Niels Ole, Elling, Christian e., Halldin, Christer
Published in Synapse (New York, N.Y.) (01.03.2014)
Published in Synapse (New York, N.Y.) (01.03.2014)
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Beta-Arrestin2 as a Competitor for GRK2 Interaction with the GLP-1 Receptor upon Receptor Activation
Jorgensen, Rasmus, Norklit Roed, Sarah, Heding, Anders, Elling, Christian E.
Published in Pharmacology (01.01.2011)
Published in Pharmacology (01.01.2011)
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Steric Hindrance Mutagenesis versus Alanine Scan in Mapping of Ligand Binding Sites in the Tachykinin NK1 Receptor
Holst, B, Zoffmann, S, Elling, C E, Hjorth, S A, Schwartz, T W
Published in Molecular pharmacology (01.01.1998)
Published in Molecular pharmacology (01.01.1998)
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Journal Article
Disulfide Bridge Engineering in the Tachykinin NK1 Receptor
Elling, Christian E, Raffetseder, Ute, Nielsen, Søren Møller, Schwartz, Thue W
Published in Biochemistry (Easton) (01.02.2000)
Published in Biochemistry (Easton) (01.02.2000)
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Oxyntomodulin Differentially Affects Glucagon-Like Peptide-1 Receptor β-Arrestin Recruitment and Signaling through Gα
Jorgensen, Rasmus, Kubale, Valentina, Vrecl, Milka, Schwartz, Thue W., Elling, Christian E.
Published in The Journal of pharmacology and experimental therapeutics (01.07.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2007)
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