Targeted kinase degradation via the KLHDC2 ubiquitin E3 ligase
Kim, Younghoon, Seo, Pooreum, Jeon, Eunhye, You, Inchul, Hwang, Kyubin, Kim, Namkyoung, Tse, Jason, Bae, Juhyeon, Choi, Ha-Soon, Hinshaw, Stephen M, Gray, Nathanael S, Sim, Taebo
Published in Cell chemical biology (16.11.2023)
Published in Cell chemical biology (16.11.2023)
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Journal Article
Design and synthesis of 7H-pyrrolo[2,3-d]pyrimidines as focal adhesion kinase inhibitors. Part 2
Choi, Ha-Soon, Wang, Zhicheng, Richmond, Wendy, He, Xiaohui, Yang, Kunyong, Jiang, Tao, Karanewsky, Donald, Gu, Xiang-ju, Zhou, Vicki, Liu, Yi, Che, Jianwei, Lee, Christian C., Caldwell, Jeremy, Kanazawa, Takanori, Umemura, Ichiro, Matsuura, Naoko, Ohmori, Osamu, Honda, Toshiyuki, Gray, Nathanael, He, Yun
Published in Bioorganic & medicinal chemistry letters (15.05.2006)
Published in Bioorganic & medicinal chemistry letters (15.05.2006)
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Journal Article
Total Synthesis of the CP Molecules CP-263,114 and CP-225,917- Part 1: Synthesis of Key Intermediates and Intelligence Gathering
Nicolaou, K. C., Baran, Phil S., Zhong, Yong-Li, Choi, Ha-Soon, Yoon, Won Hyung, He, Yun, Fong, Kin Chiu
Published in Angewandte Chemie (International ed.) (01.06.1999)
Published in Angewandte Chemie (International ed.) (01.06.1999)
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Journal Article
Total Synthesis of the CP Molecules CP-225,917 and CP-263,114- Part 2: Evolution of the Final Strategy
Nicolaou, K. C., Baran, Phil S., Zhong, Yong-Li, Fong, Kin Chiu, He, Yun, Yoon, Won Hyung, Choi, Ha-Soon
Published in Angewandte Chemie (International ed.) (01.06.1999)
Published in Angewandte Chemie (International ed.) (01.06.1999)
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Journal Article
(R)‑2-Phenylpyrrolidine Substituted Imidazopyridazines: A New Class of Potent and Selective Pan-TRK Inhibitors
Choi, Ha-Soon, Rucker, Paul V, Wang, Zhicheng, Fan, Yi, Albaugh, Pamela, Chopiuk, Greg, Gessier, Francois, Sun, Fangxian, Adrian, Francisco, Liu, Guoxun, Hood, Tami, Li, Nanxin, Jia, Yong, Che, Jianwei, McCormack, Susan, Li, Allen, Li, Jie, Steffy, Auzon, Culazzo, AnneMarie, Tompkins, Celine, Phung, Van, Kreusch, Andreas, Lu, Min, Hu, Bin, Chaudhary, Apurva, Prashad, Mahavir, Tuntland, Tove, Liu, Bo, Harris, Jennifer, Seidel, H. Martin, Loren, Jon, Molteni, Valentina
Published in ACS medicinal chemistry letters (14.05.2015)
Published in ACS medicinal chemistry letters (14.05.2015)
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Journal Article
A Novel Route to the Fused Maleic Anhydride Moiety of CP Molecules
Nicolaou, K. C., Baran, Phil S., Jautelat, Rolf, He, Yun, Fong, Kin Chiu, Choi, Ha-Soon, Yoon, Won Hyung, Zhong, Yong-Li
Published in Angewandte Chemie (International ed.) (15.02.1999)
Published in Angewandte Chemie (International ed.) (15.02.1999)
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Journal Article
Crystal structures of human HSP90α-complexed with dihydroxyphenylpyrazoles
Kreusch, Andreas, Han, Shulin, Brinker, Achim, Zhou, Vicki, Choi, Ha-soon, He, Yun, Lesley, Scott A., Caldwell, Jeremy, Gu, Xiang-ju
Published in Bioorganic & medicinal chemistry letters (01.03.2005)
Published in Bioorganic & medicinal chemistry letters (01.03.2005)
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Journal Article
Design and synthesis of 7H-pyrrolo[2,3-d]pyrimidines as focal adhesion kinase inhibitors. Part 1
CHOI, Ha-Soon, ZHICHENG WANG, YI LIU, OHMORI, Osamu, CALDWELL, Jeremy, GRAY, Nathanael, YUN HE, RICHMOND, Wendy, XIAOHUI HE, KUNYONG YANG, TAO JIANG, SIM, Taebo, KARANEWSKY, Donald, GU, Xiang-Ju, ZHOU, Vicki
Published in Bioorganic & medicinal chemistry letters (15.04.2006)
Published in Bioorganic & medicinal chemistry letters (15.04.2006)
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Journal Article
2,7-SUBSTITUTED PYRROLO[2,1-F][1,2,4]TRIAZINE COMPOUND HAVING PROTEIN KINASE INHIBITORY ACTIVITY
SHIN, In Jae, KIM, Young Hoon, SIM, Tae Bo, SANDIP, Sengupta, KIM, Nam Kyoung, CHOI, Ha Soon
Year of Publication 08.06.2023
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Year of Publication 08.06.2023
Patent
Targeted degradation of METTL3 against acute myeloid leukemia and gastric cancer
Hwang, Kyubin, Bae, Juhyeon, Jhe, Yoo-Lim, Kim, Jungmin, Cheong, Jae-Ho, Choi, Ha-Soon, Sim, Taebo
Published in European journal of medicinal chemistry (05.12.2024)
Published in European journal of medicinal chemistry (05.12.2024)
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Journal Article
Catalytic asymmetric allylation of aldehydes with BINOL-Ti(IV) complex accelerated by i-PrSSiMe3
Yu, Chan-Mo, Choi, Ha-Soon, Jung, Won-Hyuk, Lee, Sung-Soo
Published in Tetrahedron letters (23.09.1996)
Published in Tetrahedron letters (23.09.1996)
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Journal Article
New Synthetic Technology for the Synthesis of Hindered α-Diazoketones via Acyl Mesylates
Nicolaou, K. C, Baran, Phil S, Zhong, Yong-Li, Choi, Ha-Soon, Fong, Kin Chiu, He, Yun, Yoon, Won Hyung
Published in Organic letters (23.09.1999)
Published in Organic letters (23.09.1999)
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Journal Article
(R)-2-Phenylpyrrolidine Substituted Imidazopyridazines: A New Class of Potent and Selective Pan-IRK Inhibitors
Choi, Ha-Soon, Rucker, Paul V., Wang, Zhicheng, Fan, Yi, Albaugh, Pamela, Chopiuk, Greg, Gessier, Francois, Sun, Fangxian, Adrian, Francisco, Liu, Guoxun, Hood, Tami, Li, Nanxin, Jia, Yong, Che, Jianwei, McCormack, Susan, Li, Allen, Li, Jie, Steffy, Auzon, Culazzo, AnneMarie, Tompkins, Celine, Van Phung, Kreusch, Andreas, Lu, Min, Hu, Bin, Chaudhary, Apurva, Prashad, Mahavir, Tuntland, Tove, Liu, Bo, Harris, Jennifer, Seidel, H. Martin, Loren, Jon, Molteni, Valentina
Published in ACS medicinal chemistry letters (01.05.2015)
Published in ACS medicinal chemistry letters (01.05.2015)
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Journal Article