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Published in MedChemComm (21.07.2021)
Published in MedChemComm (21.07.2021)
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Published in Bioorganic & medicinal chemistry letters (01.01.2017)
Published in Bioorganic & medicinal chemistry letters (01.01.2017)
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MARK inhibitors: Declaring a No-Go decision on a chemical series based on extensive DMPK experimentation
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Published in Bioorganic & medicinal chemistry letters (01.01.2017)
Published in Bioorganic & medicinal chemistry letters (01.01.2017)
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Thiophene carboxamide inhibitors of JAK2 as potential treatments for myleoproliferative neoplasms
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Published in Bioorganic & medicinal chemistry letters (15.04.2014)
Published in Bioorganic & medicinal chemistry letters (15.04.2014)
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Thiazole-substituted aminoheteroaryls as spleen tyrosine kinase inhibitors
Ellis John Michael, Wang Liping, Andresen Brian M, Anthony Neville J, Altman Michael D, Lebrun Marie-Eve, Donofrio Anthony, Northrup Alan B, Spencer Kerrie B, Machacek Michelle R, Childers Kaleen K, Woo Hyun Chong, DuBois Byron, Miller Thomas A, Robichaud Joel S, Romeo Eric T, Deng Qiaolin, Liu Yuan, Guay Daniel, Grimm Jonathan
Year of Publication 29.08.2017
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Year of Publication 29.08.2017
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THIAZOLE-SUBSTITUTED AMINOHETEROARYLS AS SPLEEN TYROSINE KINASE INHIBITORS
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Year of Publication 02.11.2016
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Year of Publication 02.11.2016
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THIAZOLE-SUBSTITUTED AMINOHETEROARYLS AS SPLEEN TYROSINE KINASE INHIBITORS
DONOFRIO ANTHONY, GUAY DANIEL, MACHACEK MICHELLE R, WANG LIPING, WOO HYUN CHONG, GRIMM JONATHAN, ANTHONY NEVILLE J, ROBICHAUD JOEL S, ROMEO ERIC T, DENG QIAOLIN, SPENCER KERRIE B, ALTMAN MICHAEL D, LEBRUN MARIE-EVE, ANDRESEN BRIAN M, LIU YUAN, CHILDERS KALEEN K, MILLER THOMAS A, ELLIS JOHN MICHAEL, DUBOIS BYRON, NORTHRUP ALAN B
Year of Publication 03.03.2016
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Year of Publication 03.03.2016
Patent
THIAZOLE-SUBSTITUTED AMINOHETEROARYLS AS SPLEEN TYROSINE KINASE INHIBITORS
SPENCER, KERRIE, B, ANDRESEN, BRIAN, M, MILLER, THOMAS, A, LIU, YUAN, WOO, HYUN CHONG, ROBICHAUD, JOEL, S, GUAY, DANIEL, DUBOIS, BYRON, WANG, LIPING, ELLIS, JOHN MICHAEL, ALTMAN, MICHAEL, D, DENG, QIAOLIN, ANTHONY, NEVILLE, J, CHILDERS, KALEEN, K, MACHACEK, MICHELLE, R, LEBRUN, MARIE-EVE, DONOFRIO, ANTHONY, ROMEO, ERIC, T, NORTHRUP, ALAN, B, GRIMM, JONATHAN
Year of Publication 02.03.2016
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Year of Publication 02.03.2016
Patent
THIAZOLE-SUBSTITUTED AMINOHETEROARYLS AS SPLEEN TYROSINE KINASE INHIBITORS
SPENCER, KERRIE, B, ANDRESEN, BRIAN, M, MILLER, THOMAS, A, LIU, YUAN, WOO, HYUN CHONG, ROBICHAUD, JOEL, S, GUAY, DANIEL, DUBOIS, BYRON, WANG, LIPING, ELLIS, JOHN MICHAEL, ALTMAN, MICHAEL, D, DENG, QIAOLIN, ANTHONY, NEVILLE, J, CHILDERS, KALEEN, K, MACHACEK, MICHELLE, R, LEBRUN, MARIE-EVE, DONOFRIO, ANTHONY, ROMEO, ERIC, T, NORTHRUP, ALAN, B, GRIMM, JONATHAN
Year of Publication 30.10.2014
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Year of Publication 30.10.2014
Patent