A Phase I, Open-Label, Multicenter, Dose-escalation Study of the Oral Selective FGFR Inhibitor Debio 1347 in Patients with Advanced Solid Tumors Harboring FGFR Gene Alterations
Voss, Martin H, Hierro, Cinta, Heist, Rebecca S, Cleary, James M, Meric-Bernstam, Funda, Tabernero, Josep, Janku, Filip, Gandhi, Leena, Iafrate, A John, Borger, Darrell R, Ishii, Nobuya, Hu, Youyou, Kirpicheva, Yulia, Nicolas-Metral, Valerie, Pokorska-Bocci, Anna, Vaslin Chessex, Anne, Zanna, Claudio, Flaherty, Keith T, Baselga, Jose
Published in Clinical cancer research (01.05.2019)
Published in Clinical cancer research (01.05.2019)
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Journal Article
FGFR2 Extracellular Domain In-Frame Deletions Are Therapeutically Targetable Genomic Alterations That Function as Oncogenic Drivers in Cholangiocarcinoma
Cleary, James M, Raghavan, Srivatsan, Wu, Qibiao, Li, Yvonne Y, Spurr, Liam F, Gupta, Hersh V, Rubinson, Douglas A, Fetter, Isobel J, Hornick, Jason L, Nowak, Jonathan A, Siravegna, Giulia, Goyal, Lipika, Shi, Lei, Brais, Lauren K, Loftus, Maureen, Shinagare, Atul B, Abrams, Thomas A, Clancy, Thomas E, Wang, Jiping, Patel, Anuj K, Brichory, Franck, Vaslin Chessex, Anne, Sullivan, Ryan J, Keller, Rachel B, Denning, Sarah, Hill, Emma R, Shapiro, Geoffrey I, Pokorska-Bocci, Anna, Zanna, Claudio, Ng, Kimmie, Schrag, Deborah, Jänne, Pasi A, Hahn, William C, Cherniack, Andrew D, Corcoran, Ryan B, Meyerson, Matthew, Daina, Antoine, Zoete, Vincent, Bardeesy, Nabeel, Wolpin, Brian M
Published in Cancer discovery (01.10.2021)
Published in Cancer discovery (01.10.2021)
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Journal Article
Debio 0617B Inhibits Growth of STAT3-Driven Solid Tumors through Combined Inhibition of JAK, SRC, and Class III/V Receptor Tyrosine Kinases
Murone, Maximilien, Vaslin Chessex, Anne, Attinger, Antoine, Ramachandra, Raghuveer, Shetty, Shankar J, Daginakatte, Girish, Sengupta, Saumitra, Marappan, Sivapriya, Dhodheri, Samiulla, Rigotti, Stefania, Bachhav, Yogeshwar, Brienza, Silvano, Traxler, Peter, Lang, Marc, Aguet, Michel, Zoete, Vincent, Michielin, Olivier, Nicholas, Courtney, Johnson, Faye M, Ramachandra, Murali, McAllister, Andres
Published in Molecular cancer therapeutics (01.10.2016)
Published in Molecular cancer therapeutics (01.10.2016)
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Journal Article
FGFR FGFR FUSIONS
TANAKA HIROAKI, MOULON CORINNE, WOJCIK JEROME, CHESSEX ANNE VASLIN, ARMENISE CLAUDIA
Year of Publication 05.12.2016
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Year of Publication 05.12.2016
Patent
Towards a translational computational model of allergen challenge in mild asthma to support clinical development of an intranasal administration of a bacterial lysate
Arsène, Simon, Faddeenkov, Igor, Galland, Théo, Leon, Cristhyne, Lehr, Lorenz, Sansone, Caterina, Vaslin-Chessex, Anne, Pasquali, Christian, Kulesza, Alexander
Published in Journal of allergy and clinical immunology (01.02.2023)
Published in Journal of allergy and clinical immunology (01.02.2023)
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Journal Article
Truncated FGFR2 is a clinically actionable oncogene in multiple cancers
Zingg, Daniel, Bhin, Jinhyuk, Yemelyanenko, Julia, Kas, Sjors M., Rolfs, Frank, Lutz, Catrin, Lee, Jessica K., Klarenbeek, Sjoerd, Silverman, Ian M., Annunziato, Stefano, Chan, Chang S., Piersma, Sander R., Eijkman, Timo, Badoux, Madelon, Gogola, Ewa, Siteur, Bjørn, Sprengers, Justin, de Klein, Bim, de Goeij-de Haas, Richard R., Riedlinger, Gregory M., Ke, Hua, Madison, Russell, Drenth, Anne Paulien, van der Burg, Eline, Schut, Eva, Henneman, Linda, van Miltenburg, Martine H., Proost, Natalie, Zhen, Huiling, Wientjens, Ellen, de Bruijn, Roebi, de Ruiter, Julian R., Boon, Ute, de Korte-Grimmerink, Renske, van Gerwen, Bastiaan, Féliz, Luis, Abou-Alfa, Ghassan K., Ross, Jeffrey S., van de Ven, Marieke, Rottenberg, Sven, Cuppen, Edwin, Chessex, Anne Vaslin, Ali, Siraj M., Burn, Timothy C., Jimenez, Connie R., Ganesan, Shridar, Wessels, Lodewyk F. A., Jonkers, Jos
Published in Nature (London) (18.08.2022)
Published in Nature (London) (18.08.2022)
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Journal Article
Abstract 4703: The inhibitor of apoptosis protein (IAP) antagonist Debio 1143 enhances the immune response to anti-PD1/L1 inhibitors in vitro and in vivo
Attinger, Antoine, Gavillet, Bruno, Chessex, Anne Vaslin, Wiedemann, Norbert, Vuagniaux, Gregoire
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Abstract 2303: The WEE1 inhibitor Debio 0123 enhances the efficacy of standard of care DNA damaging agents in lung cancer models
Piggott, Luke, Vaslin-Chessex, Anne, Luong, Noemie, Tschumi, Benjamin, Vuagniaux, Gregoire
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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Abstract 4423: Antitumor activity of the novel oral highly selective Wee1 inhibitor Debio 0123
O'Dowd, Colin, Gavory, Gerald, Burkamp, Frank, Treder, Adam, Boyd, Caroline, Harrison, Tim, Massière, Frederic, Glück, Astrid, Chardonnens, Christophe, Zaffalon, Andrea, Rigotti, Stefania, Mader, Robert, Vuagniaux, Grégoire, Chessex, Anne Vaslin
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
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Journal Article
Publisher Correction: Truncated FGFR2 is a clinically actionable oncogene in multiple cancers
Zingg, Daniel, Bhin, Jinhyuk, Yemelyanenko, Julia, Kas, Sjors M., Rolfs, Frank, Lutz, Catrin, Lee, Jessica K., Klarenbeek, Sjoerd, Silverman, Ian M., Annunziato, Stefano, Chan, Chang S., Piersma, Sander R., Eijkman, Timo, Badoux, Madelon, Gogola, Ewa, Siteur, Bjørn, Sprengers, Justin, de Klein, Bim, de Goeij-de Haas, Richard R., Riedlinger, Gregory M., Ke, Hua, Madison, Russell, Drenth, Anne Paulien, van der Burg, Eline, Schut, Eva, Henneman, Linda, van Miltenburg, Martine H., Proost, Natalie, Zhen, Huiling, Wientjens, Ellen, de Bruijn, Roebi, de Ruiter, Julian R., Boon, Ute, de Korte-Grimmerink, Renske, van Gerwen, Bastiaan, Féliz, Luis, Abou-Alfa, Ghassan K., Ross, Jeffrey S., van de Ven, Marieke, Rottenberg, Sven, Cuppen, Edwin, Chessex, Anne Vaslin, Ali, Siraj M., Burn, Timothy C., Jimenez, Connie R., Ganesan, Shridar, Wessels, Lodewyk F. A., Jonkers, Jos
Published in Nature (London) (29.09.2022)
Published in Nature (London) (29.09.2022)
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Journal Article
FGFR FUSIONS
ARMENISE, CLAUDIA, TANAKA, HIROAKI, CHESSEX, ANNE VASLIN, WOJCIK, JÉRÔME, VASLIN CHESSEX, ANNE, MOULON, CORINNE
Year of Publication 28.10.2016
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Year of Publication 28.10.2016
Patent
The Multi-kinase Inhibitor Debio 0617B Reduces Maintenance and Self-renewal of Primary Human AML CD34 + Stem/Progenitor Cells
Murone, Maximilien, Radpour, Ramin, Attinger, Antoine, Chessex, Anne Vaslin, Huguenin, Anne-Laure, Schürch, Christian M, Banz, Yara, Sengupta, Saumitra, Aguet, Michel, Rigotti, Stefania, Bachhav, Yogeshwar, Massière, Frédéric, Ramachandra, Murali, McAllister, Andres, Riether, Carsten
Published in Molecular cancer therapeutics (01.08.2017)
Published in Molecular cancer therapeutics (01.08.2017)
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Journal Article
METHODS OF TREATING SMALL CELL LUNG CANCER
ZANNA, Claudio, NICOLAS, Valerie, DAMSTRUP, Lars, RODRIGO IMEDIO, Esteban, PIGGOTT, Luke, BELLON, Anne, VASLIN CHESSEX, Anne
Year of Publication 14.09.2023
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Year of Publication 14.09.2023
Patent
FGFR expression and susceptibility to an FGFR inhibitor
Vaslin-Chessex, Anne, Moulon, Corinne, Brichory, Franck, Pokorska-Bocci, Anna
Year of Publication 01.03.2018
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Year of Publication 01.03.2018
Patent
MÉTODOS PARA TRATAR CARCINOMA MICROCÍTICO DE PULMÓN
RODRIGO IMEDIO, ESTEBAN, DAMSTRUP, LARS, NICOLAS, VALERIE, ZANNA, CLAUDIO, BELLON, ANNE, VASLIN CHESSEX, ANNE, PIGGOTT, LUKE
Year of Publication 05.06.2024
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Year of Publication 05.06.2024
Patent
FGFR-FUSIONER
TANAKA, Hiroaki, MOULON, Corinne, CHESSEX, Anne Vaslin, WOJCIK, Jérôme, ARMENISE, Claudia
Year of Publication 05.08.2019
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Year of Publication 05.08.2019
Patent
FGFR FUSIONS
TANAKA, Hiroaki, MOULON, Corinne, CHESSEX, Anne Vaslin, WOJCIK, Jérôme, ARMENISE, Claudia
Year of Publication 08.05.2019
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Year of Publication 08.05.2019
Patent
Methods of treating small cell lung cancer
RODRIGO IMEDIO, ESTEBAN, DAMSTRUP, LARS, NICOLAS, VALERIE, ZANNA, CLAUDIO, BELLON, ANNE, VASLIN CHESSEX, ANNE, PIGGOTT, LUKE
Year of Publication 01.10.2023
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Year of Publication 01.10.2023
Patent