Process Development of a Suzuki Reaction Used in the Manufacture of Lanabecestat
Ashworth, Ian W, Campbell, Andrew D, Cherryman, Janette H, Clark, Jemma, Crampton, Alex, Eden-Rump, Edward G. B, Evans, Matthew, Jones, Martin F, McKeever-Abbas, Sahar, Meadows, Rebecca E, Skilling, Kathryn, Whittaker, David T. E, Woodward, Robert L, Inglesby, Phillip A
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Published in Organic process research & development (21.12.2018)
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Development and Proof of Concept for a Large-Scale Photoredox Additive-Free Minisci Reaction
Graham, Mark A., Noonan, Gary, Cherryman, Janette H., Douglas, James J., Gonzalez, Miguel, Jackson, Lucinda V., Leslie, Kevin, Liu, Zhi-qing, McKinney, David, Munday, Rachel H., Parsons, Chris D., Whittaker, David T. E., Zhang, En-xuan, Zhang, Jun-wang
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Process Development, Manufacture, and Understanding of the Atropisomerism and Polymorphism of Verinurad
Ring, Oliver T, Hayter, Barry R, Ronson, Thomas O, Agnew, Lauren R, Ashworth, Ian W, Cherryman, Janette, Gall, Malcolm A. Y, Hamilton, Peter R, Inglesby, Phillip A, Jones, Martin F, Lamacraft, Alex L, Leahy, Adam J, McKinney, David, Miller-Potucka, Lucie, Powell, Lyn, Putra, Okky D, Robbins, Andrew J, Tomasi, Simone, Wordsworth, Rosemary A
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Where Has My Acid Gone? Understanding the Self-Catalyzed Esterification of Maleic Acid in Methanol During Salt Formation
Ashworth, Ian W, Bush, Edward, Chan, Lai C, Cherryman, Janette, Cox, Brian G, Muir, James, Korupoju, Srinivasa Rao, Keshwan, Jaikumar
Published in Organic process research & development (19.10.2012)
Published in Organic process research & development (19.10.2012)
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POLYMORPHIC FORM OF 4-[3-(4-CYCLOPROPANECARBONYL-PIPERAZINE-1-CARBONYL)-4-FLUORO-BENZYL]-2H-PHTHALAZIN-1-ONE
ASHWORTH IAN WOODWARD, LAFFAN DAVID DERMOT PATRICK, MULLHOLLAND KEITH RAYMOND, JONES MARTIN FRANCIS, MENEAR KEITH ALLAN, PITTAM JOHN DAVID, OTTRIDGE ANTHONY PETER, HALLETT MICHAEL RAYMOND, CHERRYMAN JANETTE HELEN, LONDESBROUGH DEREK JOHN
Year of Publication 22.01.2015
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Year of Publication 22.01.2015
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PROCESS FOR PREPARING HETEROCYCLIC COMPOUNDS INCLUDING TRANS-7-OXO-6-(SULPHOOXY)-1,6-DIAZABICYCLO[3,2,1]OCTANE-2-CARBOXAMIDE AND SALTS THEREOF
RACHA SAIBABA, ZHOU SHAO HONG, GOLDEN MICHAEL, KALYAN YURIY B, BOYD JOHN ALISTAIR, LAWTON GRAHAM RICHARD, PHILLIPS ANDREW JOHN, CHERRYMAN JANETTE HELEN, RONSHEIM MELANIE SIMONE, TELFORD ALEXANDER, MILNE DAVID, DEDHIYA MAHENDRA G
Year of Publication 03.04.2014
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Year of Publication 03.04.2014
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POLYMORPHIC FORM OF 4-[3-(4-CYCLOPROPANECARBONYL-PIPERAZINE-1-CARBONYL)-4-FLUORO-BENZYL]-2H-PHTHALAZIN-1-ONE
ASHWORTH IAN WOODWARD, LAFFAN DAVID DERMOT PATRICK, MULLHOLLAND KEITH RAYMOND, JONES MARTIN FRANCIS, MENEAR KEITH ALLAN, PITTAM JOHN DAVID, OTTRIDGE ANTHONY PETER, HALLETT MICHAEL RAYMOND, CHERRYMAN JANETTE HELEN, LONDESBROUGH DEREK JOHN
Year of Publication 28.01.2014
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Year of Publication 28.01.2014
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PROCESSES FOR PREPARING HETEROCYCLIC COMPOUNDS INCLUDING TRANS-7-OXO-6-(SULPHOOXY)-1,6-DIAZABICYCLO[3,2,1]OCTANE-2-CARBOXAMIDE AND SALTS THEREOF
DEDHIYA, MAHENDRA G, KALYAN, YURIY B, RONSHEIM, MELANIE SIMONE, GOLDEN, MICHAEL, MILNE, DAVID, CHERRYMAN, JANETTE, RACHA, SAIBABA, BOYD, ALISTAIR, ZHOU, SHAO HONG, PHILLIPS, ANDREW, TELFORD, ALEXANDER, LAWTON, GRAHAM RICHARD
Year of Publication 21.04.2020
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Year of Publication 21.04.2020
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PROCESS FOR PREPARING HETEROCYCLIC COMPOUNDS INCLUDING TRANS-7-OXO-6-(SULPHOOXY)-1,6-DIAZABICYCLO[3,2,1]OCTANE-2-CARBOXAMIDE AND SALTS THEREOF
DEDHIYA, MAHENDRA G, BOYD, JOHN ALISTAIR, KALYAN, YURIY B, GOLDEN, MICHAEL, MILNE, DAVID, RONSHEIM, MELANIE SIMONE, RACHA, SAIBABA, ZHOU, SHAO HONG, CHERRYMAN, JANETTE HELEN, TELFORD, ALEXANDER, LAWTON, GRAHAM RICHARD, PHILLIPS, ANDREW JOHN
Year of Publication 20.04.2018
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Year of Publication 20.04.2018
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Processes for preparing heterocyclic compounds including trans-7-oxo-6-(sulphooxy)-1,6-diazabicyclo[3,2,1]octane-2-carboxamide and salts thereof
Kalyan Yuriy B, Ronsheim Melanie Simone, Golden Michael, Cherryman Janette, Dedhiya Mahendra G, Racha Saibaba, Zhou Shao Hong, Lawton Graham Richard, Telford Alexander, Boyd Alistair, Phillips Andrew, Milne David
Year of Publication 04.07.2017
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Year of Publication 04.07.2017
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PROCESSES FOR PREPARING HETEROCYCLIC COMPOUNDS INCLUDING TRANS-7-OXO-6-(SULPHOOXY)-1,6-DIAZABICYCLO[3,2,1]OCTANE-2-CARBOXAMIDE AND SALTS THEREOF
Kalyan Yuriy B, Ronsheim Melanie Simone, Golden Michael, Cherryman Janette, Dedhiya Mahendra G, Racha Saibaba, Zhou Shao Hong, Lawton Graham Richard, Telford Alexander, Boyd Alistair, Phillips Andrew, Milne David
Year of Publication 26.01.2017
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Year of Publication 26.01.2017
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Process for preparing heterocyclic compounds including trans-7-oxo-6-(sulphooxy)-1,6-diazabicyclo[3,2,1]octane-2-carboxamide and salts thereof
Cherryman, Janette Helen, Boyd, John Alistair, Ronsheim, Melanie Simone, Telford, Alexander, Kalyan, Yuriy B, Lawton, Graham Richard, Dedhiya, Mahendra G, Phillips, Andrew John, Zhou, Shao Hong, Golden, Michael, Milne, David, Racha, Saibaba
Year of Publication 22.12.2016
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Year of Publication 22.12.2016
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METHOD OF PREPARING CRYSTALLINE FORM PHTHALAZINONE DERIVATIVE FOR USE IN CANCER TREATMENT
MENEAR, KEITH ALLAN, PITTAM, JOHN DAVID, MULLHOLLAND, KEITH RAYMOND, HALLETT, MICHAEL RAYMOND, JONES, MARTIN FRANCIS, LAFFAN, DAVID DERMOT PATRICK, CHERRYMAN, JANETTE HELEN, LONDESBROUGH, DEREK JOHN, OTTRIDGE, ANTHONY PETER, ASHWORTH, IAN WOODWARD
Year of Publication 06.09.2016
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Year of Publication 06.09.2016
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Processes for preparing heterocyclic compounds including trans-7-oxo-6-(sulphooxy)-1,6-diazabicyclo[3,2,1]octane-2-carboxamide and salts thereof
RACHA SAIBABA, CHERRYMAN JANETTE, BOYD ALISTAIR, ZHOU SHAO HONG, KALYAN YURIY B, GOLDEN MICHAEL, LAWTON GRAHAM RICHARD, RONSHEIM MELANIE SIMONE, TELFORD ALEXANDER, MILNE DAVID, DEDHIYA MAHENDRA G, PHILLIPS ANDREW
Year of Publication 15.03.2016
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Year of Publication 15.03.2016
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PROCESSES FOR PREPARING HETEROCYCLIC COMPOUNDS INCLUDING TRANS-7-OXO-6-(SULPHOOXY)-1,6-DIAZABICYCLO[3,2,1]OCTANE-2-CARBOXAMIDE AND SALTS THEREOF
RACHA SAIBABA, CHERRYMAN JANETTE, BOYD ALISTAIR, ZHOU SHAO HONG, KALYAN YURIY B, GOLDEN MICHAEL, LAWTON GRAHAM RICHARD, RONSHEIM MELANIE SIMONE, TELFORD ALEXANDER, MILNE DAVID, DEDHIYA MAHENDRA G, PHILLIPS ANDREW
Year of Publication 03.02.2016
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Year of Publication 03.02.2016
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PROCESS FOR PREPARING HETEROCYCLIC COMPOUNDS INCLUDING TRANS-7-OXO-6-(SULPHOOXY)-1,6-DIAZABICYCLO[3,2,1]OCTANE-2-CARBOXAMIDE AND SALTS THEREOF
DEDHIYA, MAHENDRA G, KALYAN, YURIY B, GOLDEN, MICHAEL, MILNE, DAVID, RONSHEIM, MELANIE SIMONE, RACHA, SAIBABA, ZHOU, SHAO HONG, CHERRYMAN, JANETTE HELEN, BOYD, ALISTAIR JOHN, TELFORD, ALEXANDER, LAWTON, GRAHAM RICHARD, PHILLIPS, ANDREW JOHN
Year of Publication 25.11.2015
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Year of Publication 25.11.2015
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Polymorphic form of 4-[3-(4-cyclopropanecarbonyl-piperazine-1-carbonyl)-4-fluorobenzyl]-2H-phthalazin-1-one
MENEAR, KEITH ALLAN, PITTAM, JOHN DAVID, MULLHOLLAND, KEITH RAYMOND, HALLETT, MICHAEL RAYMOND, JONES, MARTIN FRANCIS, LAFFAN, DAVID DERMOT PATRICK, CHERRYMAN, JANETTE HELEN, LONDESBROUGH, DEREK JOHN, OTTRIDGE, ANTHONY PETER, ASHWORTH, IAN WOODWARD
Year of Publication 25.06.2015
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Year of Publication 25.06.2015
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Polymorphic form of 4-[3-(4-cyclopropanecarbonyl-piperazine-1-carbonyl)-4-fluoro-benzyl]-2H-phthalazin-1-one
ASHWORTH IAN WOODWARD, LAFFAN DAVID DERMOT PATRICK, MULLHOLLAND KEITH RAYMOND, JONES MARTIN FRANCIS, MENEAR KEITH ALLAN, PITTAM JOHN DAVID, OTTRIDGE ANTHONY PETER, HALLETT MICHAEL RAYMOND, CHERRYMAN JANETTE HELEN, LONDESBROUGH DEREK JOHN
Year of Publication 27.05.2015
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Year of Publication 27.05.2015
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