Search Results - "CHENARD, Bertrand" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Treatment with HC-070, a potent inhibitor of TRPC4 and TRPC5, leads to anxiolytic and antidepressant effects in mice

Treatment with HC-070, a potent inhibitor of TRPC4 and TRPC5, leads to anxiolytic and antidepressant effects in mice

by Just, Stefan, Chenard, Bertrand L, Ceci, Angelo, Strassmaier, Timothy, Chong, Jayhong A, Blair, Nathaniel T, Gallaschun, Randall J, Del Camino, Donato, Cantin, Susan, D'Amours, Marc, Eickmeier, Christian, Fanger, Christopher M, Hecker, Carsten, Hessler, David P, Hengerer, Bastian, Kroker, Katja S, Malekiani, Sam, Mihalek, Robert, McLaughlin, Joseph, Rast, Georg, Witek, JoAnn, Sauer, Achim, Pryce, Christopher R, Moran, Magdalene M
Published in PloS one (31.01.2018)

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Journal Article

C5a, But Not C3a, Increases VEGF Secretion in ARPE-19 Human Retinal Pigment Epithelial Cells

C5a, But Not C3a, Increases VEGF Secretion in ARPE-19 Human Retinal Pigment Epithelial Cells

by Cortright, Daniel N., Meade, Robin, Waters, Stephen M., Chenard, Bertrand L., Krause, James E.
Published in Current eye research (2009)

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Discovery of Novel 6,6-Heterocycles as Transient Receptor Potential Vanilloid (TRPV1) Antagonists

Discovery of Novel 6,6-Heterocycles as Transient Receptor Potential Vanilloid (TRPV1) Antagonists

by Blum, Charles A, Caldwell, Timothy, Zheng, Xiaozhang, Bakthavatchalam, Rajagopal, Capitosti, Scott, Brielmann, Harry, De Lombaert, Stéphane, Kershaw, Mark T, Matson, David, Krause, James E, Cortright, Daniel, Crandall, Marci, Martin, William J, Murphy, Beth Ann, Boyce, Susan, Jones, A. Brian, Mason, Glenn, Rycroft, Wayne, Perrett, Helen, Conley, Rachael, Burnaby-Davies, Nicola, Chenard, Bertrand L, Hodgetts, Kevin J
Published in Journal of medicinal chemistry (22.04.2010)

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Opportunities and Challenges in the Discovery of New Central Nervous System Drugs

Opportunities and Challenges in the Discovery of New Central Nervous System Drugs

by Krause, James E., Chenard, Bertrand L.
Published in Annals of the New York Academy of Sciences (01.11.2008)

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An Efficient Preparation of β-Aryl-β-ketophosphonates by the TFAA/H3PO4-Mediated Acylation of Arenes with Phosphonoacetic Acids

An Efficient Preparation of β-Aryl-β-ketophosphonates by the TFAA/H3PO4-Mediated Acylation of Arenes with Phosphonoacetic Acids

by Luke, George P, Seekamp, Christopher K, Wang, Zhe-Qing, Chenard, Bertrand L
Published in Journal of organic chemistry (15.08.2008)

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Pyrido[2,3-b]pyrazines, discovery of TRPV1 antagonists with reduced potential for the formation of reactive metabolites

Pyrido[2,3-b]pyrazines, discovery of TRPV1 antagonists with reduced potential for the formation of reactive metabolites

by Hodgetts, Kevin J., Blum, Charles A., Caldwell, Timothy, Bakthavatchalam, Rajagopal, Zheng, Xiaozhang, Capitosti, Scott, Krause, James E., Cortright, Daniel, Crandall, Marci, Murphy, Beth Ann, Boyce, Susan, Brian Jones, A., Chenard, Bertrand L.
Published in Bioorganic & medicinal chemistry letters (01.08.2010)

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Aminoquinazolines as TRPV1 antagonists: Modulation of drug-like properties through the exploration of 2-position substitution

Aminoquinazolines as TRPV1 antagonists: Modulation of drug-like properties through the exploration of 2-position substitution

by Blum, Charles A., Zheng, Xiaozhang, Brielmann, Harry, Hodgetts, Kevin J., Bakthavatchalam, Rajagopal, Chandrasekhar, Jayaraman, Krause, James E., Cortright, Daniel, Matson, David, Crandall, Marci, Ngo, Chu K., Fung, Lawrence, Day, Marta, Kershaw, Mark, De Lombaert, Stéphane, Chenard, Bertrand L.
Published in Bioorganic & medicinal chemistry (15.08.2008)

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1-Benzylbenzimidazoles : The discovery of a novel series of bradykinin B1 receptor antagonists

1-Benzylbenzimidazoles : The discovery of a novel series of bradykinin B1 receptor antagonists

by QIN GUO, CHANDRASEKHAR, Jayaraman, BROOM, Daniel, KERSHAW, Mark T, SIMMERMACHER-MAYER, Jean, YAO PENG, HODGETTS, Kevin J, IHLE, David, WUSTROW, David J, CHENARD, Bertrand L, KRAUSE, James E, HUTCHISON, Alan, ALDERMAN, Dawn, CHENG, Charles, CORTRIGHT, Daniel
Published in Bioorganic & medicinal chemistry letters (15.09.2008)

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Journal Article

Molecular Characterization of the Gerbil C5a Receptor and Identification of a Transmembrane Domain V Amino Acid That Is Crucial for Small Molecule Antagonist Interaction

Molecular Characterization of the Gerbil C5a Receptor and Identification of a Transmembrane Domain V Amino Acid That Is Crucial for Small Molecule Antagonist Interaction

by Waters, Stephen M., Brodbeck, Robbin M., Steflik, Jeremy, Yu, Jianying, Baltazar, Carolyn, Peck, Amy E., Severance, Daniel, Zhang, Lu Yan, Currie, Kevin, Chenard, Bertrand L., Hutchison, Alan J., Maynard, George, Krause, James E.
Published in The Journal of biological chemistry (09.12.2005)

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Journal Article

Aminopyrazine CB1 receptor inverse agonists

Aminopyrazine CB1 receptor inverse agonists

by Wustrow, David J., Maynard, George D., Yuan, Jun, Zhao, He, Mao, Jianmin, Guo, Qin, Kershaw, Mark, Hammer, Jack, Brodbeck, Robbin M., Near, Kristen E., Zhou, Dan, Beers, David S., Chenard, Bertrand L., Krause, James E., Hutchison, Alan J.
Published in Bioorganic & medicinal chemistry (01.06.2008)

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Journal Article

Transient receptor potential ion channels as targets for the discovery of pain therapeutics

Transient receptor potential ion channels as targets for the discovery of pain therapeutics

by Krause, James E, Chenard, Bertrand L, Cortright, Daniel N
Published in Current opinion in investigational drugs (London, England : 2000) (01.01.2005)

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Development of a Scaleable Synthesis of NDT 9533750, a Key Intermediate to a Series of Novel Subtype Preferring GABAA Partial Agonists

Development of a Scaleable Synthesis of NDT 9533750, a Key Intermediate to a Series of Novel Subtype Preferring GABAA Partial Agonists

by Xu, Yuelian, Han, Bingsong, Wang, Zhe-Qing, Shaw, Kenneth R, Chenard, Bertrand L, Maynard, George, Xie, Linghong
Published in Organic process research & development (20.07.2007)

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Quinazolin-4-one α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor Antagonists: Structure−Activity Relationship of the C-2 Side Chain Tether

Quinazolin-4-one α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor Antagonists: Structure−Activity Relationship of the C-2 Side Chain Tether

by Chenard, Bertrand L, Welch, Willard M, Blake, James F, Butler, Todd W, Reinhold, Anthony, Ewing, Frank E, Menniti, Frank S, Pagnozzi, Martin J
Published in Journal of medicinal chemistry (24.05.2001)

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CP-101,606, an NR2B subunit selective NMDA receptor antagonist, inhibits NMDA and injury induced c-fos expression and cortical spreading depression in rodents

CP-101,606, an NR2B subunit selective NMDA receptor antagonist, inhibits NMDA and injury induced c-fos expression and cortical spreading depression in rodents

by Menniti, Frank S, Pagnozzi, Martin J, Butler, Paul, Chenard, Bertrand L, Jaw-Tsai, Sarah S, Frost White, W
Published in Neuropharmacology (01.06.2000)

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CP-465,022, a selective noncompetitive AMPA receptor antagonist, blocks AMPA receptors but is not neuroprotective in vivo

CP-465,022, a selective noncompetitive AMPA receptor antagonist, blocks AMPA receptors but is not neuroprotective in vivo

by MENNITI, Frank S, BUCHAN, Alistair M, CHENARD, Bertrand L, CRITCHETT, Donald J, GANONG, Alan H, GUANOWSKY, Victor, SEYMOUR, Patricia A, WELCH, Willard M
Published in Stroke (1970) (2003)

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Journal Article

SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF

SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF

by CHENARD BERTRAND, GALLASCHUN RANDALL
Year of Publication 27.11.2015

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Patent

피부 장애 치료에서 사용을 위한 화합물 및 조성물

피부 장애 치료에서 사용을 위한 화합물 및 조성물

by WU XINYUAN, TERKIELTAUB DOV, SCHUTZ NILI CLAUDIA, CHENARD BERTRAND L
Year of Publication 14.10.2022

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Patent

(3R,4S)-3-[4-(4-Fluorophenyl)-4-hydroxypiperidin-1-yl]chroman-4,7-diol: A Conformationally Restricted Analogue of the NR2B Subtype-Selective NMDA Antagonist (1S,2S)-1-(4-Hydroxyphenyl)-2- (4-hydroxy-4-phenylpiperidino)-1-propanol

(3R,4S)-3-[4-(4-Fluorophenyl)-4-hydroxypiperidin-1-yl]chroman-4,7-diol: A Conformationally Restricted Analogue of the NR2B Subtype-Selective NMDA Antagonist (1S,2S)-1-(4-Hydroxyphenyl)-2- (4-hydroxy-4-phenylpiperidino)-1-propanol

by Butler, Todd W, Blake, James F, Bordner, Jon, Butler, Paul, Chenard, Bertrand L, Collins, Mary A, DeCosta, Debra, Ducat, Mary J, Eisenhard, Michael E, Menniti, Frank S, Pagnozzi, Martin J, Sands, Steven B, Segelstein, Barbara E, Volberg, Walter, White, W. Frost, Zhao, Dayao
Published in Journal of medicinal chemistry (26.03.1998)

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Journal Article

치료 화합물 및 조성물

치료 화합물 및 조성물

by TENG ZHIYAO, XU YUELIAN, STASSEN FRANS L, HAYWARD NEIL J, CHENARD BERTRAND L
Year of Publication 14.10.2020

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Patent

치료 화합물 및 조성물

치료 화합물 및 조성물

by FORNICOLA RICHARD, MATISON MICHAEL E, XU YUELIAN, HAYWARD NEIL J, CHENARD BERTRAND L, DOROW ROBERTA L, KOLCHINSKI ALEXANDER
Year of Publication 12.07.2021

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Patent

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