Discovery of a Highly Selective Glycogen Synthase Kinase-3 Inhibitor (PF-04802367) That Modulates Tau Phosphorylation in the Brain: Translation for PET Neuroimaging
Liang, Steven H., Chen, Jinshan Michael, Normandin, Marc D., Chang, Jeanne S., Chang, George C., Taylor, Christine K., Trapa, Patrick, Plummer, Mark S., Para, Kimberly S., Conn, Edward L., Lopresti-Morrow, Lori, Lanyon, Lorraine F., Cook, James M., Richter, Karl E. G., Nolan, Charlie E., Schachter, Joel B., Janat, Fouad, Che, Ye, Shanmugasundaram, Veerabahu, Lefker, Bruce A., Enerson, Bradley E., Livni, Elijahu, Wang, Lu, Guehl, Nicolas J., Patnaik, Debasis, Wagner, Florence F., Perlis, Roy, Holson, Edward B., Haggarty, Stephen J., El Fakhri, Georges, Kurumbail, Ravi G., Vasdev, Neil
Published in Angewandte Chemie (International ed.) (08.08.2016)
Published in Angewandte Chemie (International ed.) (08.08.2016)
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Journal Article
Ru/Ni Dual Catalytic Desulfinative Photoredox Csp2 –Csp3 Cross‑Coupling of Alkyl Sulfinate Salts and Aryl Halides
Knauber, Thomas, Chandrasekaran, Ramalakshmi, Tucker, Joseph W, Chen, Jinshan Michael, Reese, Matthew, Rankic, Danica A, Sach, Neal, Helal, Christopher
Published in Organic letters (15.12.2017)
Published in Organic letters (15.12.2017)
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Journal Article
Ru/Ni Dual Catalytic Desulfinative Photoredox C-sp(2)-C-sp(3) Cross-Coupling of Alkyl Sulfinate Salts and Aryl Halides
Knauber, Thomas, Chandrasekaran, Ramalakshmi, Tucker, Joseph W., Chen, Jinshan Michael, Reese, Matthew, Rankic, Danica A., Sach, Neal, Helal, Christopher
Published in Organic letters (15.12.2017)
Published in Organic letters (15.12.2017)
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LRRK2 억제제로서의 신규 이미다조[4,5-C]퀴놀린 유도체
BRODNEY MICHAEL AARON, CHAPPIE THOMAS ALLEN, WAGER TRAVIS T, CHEN JINSHAN MICHAEL, GARNSEY MICHELLE RENEE, COFFMAN KAREN JEAN, COE JOTHAM WADSWORTH, REESE MATTHEW RICHARD, VERHOEST PATRICK ROBERT, KURUMBAIL RAVI G, MARTINEZ ALSINA LUIS ANGEL, GALATSIS PAUL, ROSE COLIN RICHARD, WARMUS JOSEPH SCOTT, PETTERSSON MARTIN YOUNGJIN, HELAL CHRISTOPHER JOHN, ZHANG YUAN, KORMOS BETHANY LYN, HENDERSON JACLYN LOUISE, STEPAN ANTONIA FRIEDERIKE
Year of Publication 16.12.2019
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Year of Publication 16.12.2019
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ISOXAZOLE DERIVATIVES USEFUL AS ANTIBATERIAL AGENTS
ABRAMITE JOSEPH A, BROWN MATTHEW F, CHEN JINSHAN MICHAEL, MONTGOMERY JUSTIN I, REILLY USA, MELNICK MICHAEL
Year of Publication 24.12.2013
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Year of Publication 24.12.2013
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IMIDAZOLE, PYRAZOLE, AND TRIAZOLE DERIVATIVES USEFUL AS ANTIBACTERIAL AGENTS
BROWN MATTHEW F, CHEN JINSHAN MICHAEL, MONTGOMERY JUSTIN I, REILLY USA, MELNICK MICHAEL
Year of Publication 23.12.2013
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Year of Publication 23.12.2013
Patent
Structural Basis for Achieving GSK-3β Inhibition with High Potency, Selectivity, and Brain Exposure for Positron Emission Tomography Imaging and Drug Discovery
Bernard-Gauthier, Vadim, Mossine, Andrew V, Knight, Ashley, Patnaik, Debasis, Zhao, Wen-Ning, Cheng, Chialin, Krishnan, Hema S, Xuan, Lucius L, Chindavong, Peter S, Reis, Surya A, Chen, Jinshan Michael, Shao, Xia, Stauff, Jenelle, Arteaga, Janna, Sherman, Phillip, Salem, Nicolas, Bonsall, David, Amaral, Brenda, Varlow, Cassis, Wells, Lisa, Martarello, Laurent, Patel, Shil, Liang, Steven H, Kurumbail, Ravi G, Haggarty, Stephen J, Scott, Peter J. H, Vasdev, Neil
Published in Journal of medicinal chemistry (14.11.2019)
Published in Journal of medicinal chemistry (14.11.2019)
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Journal Article
Ru/Ni Dual Catalytic Desulfinative Photoredox C sp 2 -C sp 3 Cross-Coupling of Alkyl Sulfinate Salts and Aryl Halides
Knauber, Thomas, Chandrasekaran, Ramalakshmi, Tucker, Joseph W, Chen, Jinshan Michael, Reese, Matthew, Rankic, Danica A, Sach, Neal, Helal, Christopher
Published in Organic letters (15.12.2017)
Published in Organic letters (15.12.2017)
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Pyridone Methylsulfone Hydroxamate LpxC Inhibitors for the Treatment of Serious Gram-Negative Infections
Montgomery, Justin I, Brown, Matthew F, Reilly, Usa, Price, Loren M, Abramite, Joseph A, Arcari, Joel, Barham, Rose, Che, Ye, Chen, Jinshan Michael, Chung, Seung Won, Collantes, Elizabeth M, Desbonnet, Charlene, Doroski, Matthew, Doty, Jonathan, Engtrakul, Juntyma J, Harris, Thomas M, Huband, Michael, Knafels, John D, Leach, Karen L, Liu, Shenping, Marfat, Anthony, McAllister, Laura, McElroy, Eric, Menard, Carol A, Mitton-Fry, Mark, Mullins, Lisa, Noe, Mark C, O’Donnell, John, Oliver, Robert, Penzien, Joseph, Plummer, Mark, Shanmugasundaram, Veerabahu, Thoma, Christy, Tomaras, Andrew P, Uccello, Daniel P, Vaz, Alfin, Wishka, Donn G
Published in Journal of medicinal chemistry (23.02.2012)
Published in Journal of medicinal chemistry (23.02.2012)
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Potent Inhibitors of LpxC for the Treatment of Gram-Negative Infections
Brown, Matthew F, Reilly, Usa, Abramite, Joseph A, Arcari, Joel T, Oliver, Robert, Barham, Rose A, Che, Ye, Chen, Jinshan Michael, Collantes, Elizabeth M, Chung, Seung Won, Desbonnet, Charlene, Doty, Jonathan, Doroski, Matthew, Engtrakul, Juntyma J, Harris, Thomas M, Huband, Michael, Knafels, John D, Leach, Karen L, Liu, Shenping, Marfat, Anthony, Marra, Andrea, McElroy, Eric, Melnick, Michael, Menard, Carol A, Montgomery, Justin I, Mullins, Lisa, Noe, Mark. C, O’Donnell, John, Penzien, Joseph, Plummer, Mark S, Price, Loren M, Shanmugasundaram, Veerabahu, Thoma, Christy, Uccello, Daniel P, Warmus, Joseph S, Wishka, Donn G
Published in Journal of medicinal chemistry (26.01.2012)
Published in Journal of medicinal chemistry (26.01.2012)
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SUBSTITUTED HETEROCYCLIC DERIVATIVES AND COMPOSITIONS AND THEIR PHARMACEUTICAL USE AS ANTIBACTERIALS
CHEN JINSHAN MICHAEL, LI ZHENGONG BRYAN, ZHANG ZHIJUN, BRICKNER STEVEN JOSEPH, ROBINSON SHAUGHNESSY, MARFAT ANTHONY, REILLY USA, MITTON FRY MARK JOSEPH, SUBRAMANYAM CHAKRAPANI, PLOTKIN MICHAEL AARON
Year of Publication 06.02.2012
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Year of Publication 06.02.2012
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Discovery of Dap‑3 Polymyxin Analogues for the Treatment of Multidrug-Resistant Gram-Negative Nosocomial Infections
Magee, Thomas V, Brown, Matthew F, Starr, Jeremy T, Ackley, David C, Abramite, Joseph A, Aubrecht, Jiri, Butler, Andrew, Crandon, Jared L, Dib-Hajj, Fadia, Flanagan, Mark E, Granskog, Karl, Hardink, Joel R, Huband, Michael D, Irvine, Rebecca, Kuhn, Michael, Leach, Karen L, Li, Bryan, Lin, Jian, Luke, David R, MacVane, Shawn H, Miller, Alita A, McCurdy, Sandra, McKim, James M, Nicolau, David P, Nguyen, Thuy-Trinh, Noe, Mark C, O’Donnell, John P, Seibel, Scott B, Shen, Yue, Stepan, Antonia F, Tomaras, Andrew P, Wilga, Paul C, Zhang, Li, Xu, Jinfeng, Chen, Jinshan Michael
Published in Journal of medicinal chemistry (27.06.2013)
Published in Journal of medicinal chemistry (27.06.2013)
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Novel 3-O-carbamoyl erythromycin A derivatives (carbamolides) with activity against resistant staphylococcal and streptococcal isolates
Magee, Thomas V., Han, Seungil, McCurdy, Sandra P., Nguyen, Thuy-Trinh, Granskog, Karl, Marr, Eric S., Maguire, Bruce A., Huband, Michael D., Chen, Jinshan Michael, Subashi, Timothy A., Shanmugasundaram, Veerabahu
Published in Bioorganic & medicinal chemistry letters (15.03.2013)
Published in Bioorganic & medicinal chemistry letters (15.03.2013)
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Discovery of a Highly Selective Glycogen Synthase Kinase-3 Inhibitor (PF-04802367) That Modulates Tau Phosphorylation in the Brain: Translation for PET Neuroimaging
Liang, Steven H., Chen, Jinshan Michael, Normandin, Marc D., Chang, Jeanne S., Chang, George C., Taylor, Christine K., Trapa, Patrick, Plummer, Mark S., Para, Kimberly S., Conn, Edward L., Lopresti-Morrow, Lori, Lanyon, Lorraine F., Cook, James M., Richter, Karl E. G., Nolan, Charlie E., Schachter, Joel B., Janat, Fouad, Che, Ye, Shanmugasundaram, Veerabahu, Lefker, Bruce A., Enerson, Bradley E., Livni, Elijahu, Wang, Lu, Guehl, Nicolas J., Patnaik, Debasis, Wagner, Florence F., Perlis, Roy, Holson, Edward B., Haggarty, Stephen J., El Fakhri, Georges, Kurumbail, Ravi G., Vasdev, Neil
Published in Angewandte Chemie (08.08.2016)
Published in Angewandte Chemie (08.08.2016)
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NOVEL IMIDAZO[4,5-C]QUINOLINE DERIVATIVES AS LRRK2 INHIBITORS
ZHANG, Yuan, BRODNEY, Michael Aaron, HELAL, Christopher John, REESE, Matthew Richard, WAGER, Travis T, CHAPPIE, Thomas Allen, PETTERSSON, Martin Youngjin, MARTINEZ-ALSINA, Luis Angel, COE, Jotham Wadsworth, COFFMAN, Karen Jean, CHEN, Jinshan Michael, ROSE, Colin Richard, GARNSEY, Michelle Renee, KORMOS, Bethany Lyn, GALATSIS, Paul, VERHOEST, Patrick Robert, WARMUS, Joseph Scott, STEPAN, Antonia Friederike, HENDERSON, Jaclyn Louise, KURUMBAIL, Ravi G
Year of Publication 15.02.2023
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Year of Publication 15.02.2023
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Novel imidazo[4,5-c]quinoline derivatives as LRRK2 inhibitors
Verhoest, Patrick Robert, Brodney, Michael Aaron, Wager, Travis T, Zhang, Yuan, Chen, Jinshan Michael, Reese, Matthew Richard, Coffman, Karen Jean, Stepan, Antonia Friederike, Garnsey, Michelle Renee, Henderson, Jaclyn Louise, Kormos, Bethany Lyn, Rose, Colin Richard, Kurumbail, Ravi G, Galatsis, Paul, Coe, Jotham Wadsworth, Chappie, Thomas Allen, Pettersson, Martin Youngjin, Helal, Christopher John, Martinez-Alsina, Luis Angel, Warmus, Joseph Scott
Year of Publication 19.05.2022
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Year of Publication 19.05.2022
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Imidazo[4,5-C]quinoline derivatives as LRRK2 inhibitors
Verhoest, Patrick Robert, Brodney, Michael Aaron, Wager, Travis T, Zhang, Yuan, Chen, Jinshan Michael, Reese, Matthew Richard, Coffman, Karen Jean, Stepan, Antonia Friederike, Garnsey, Michelle Renee, Henderson, Jaclyn Louise, Kormos, Bethany Lyn, Rose, Colin Richard, Kurumbail, Ravi G, Galatsis, Paul, Coe, Jotham Wadsworth, Chappie, Thomas Allen, Pettersson, Martin Youngjin, Helal, Christopher John, Martinez-Alsina, Luis Angel, Warmus, Joseph Scott
Year of Publication 26.04.2022
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Year of Publication 26.04.2022
Patent
NOVEL IMIDAZO[4,5-C]QUINOLINE DERIVATIVES AS LRRK2 INHIBITORS
ZHANG, Yuan, BRODNEY, Michael Aaron, HELAL, Christopher John, REESE, Matthew Richard, WAGER, Travis T, CHAPPIE, Thomas Allen, PETTERSSON, Martin Youngjin, MARTINEZ-ALSINA, Luis Angel, COE, Jotham Wadsworth, COFFMAN, Karen Jean, CHEN, Jinshan Michael, ROSE, Colin Richard, GARNSEY, Michelle Renee, KORMOS, Bethany Lyn, GALATSIS, Paul, Henderson, Jaclyn Louise, VERHOEST, Patrick Robert, WARMUS, Joseph Scott, STEPAN, Antonia Friederike, KURUMBAIL, Ravi G
Year of Publication 18.11.2021
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Year of Publication 18.11.2021
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IMIDAZOLE, PYRAZOLE, AND TRIAZOLE DERIVATIVES USEFUL AS ANTIBACTERIAL AGENTS
REILLY, USA, MONTGOMERY, JUSTIN I, MELNICK, MICHAEL, CHEN, JINSHAN MICHAEL, BROWN, MATTHEW F
Year of Publication 30.12.2015
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Year of Publication 30.12.2015
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