In Vitro Resistance Study of AG-021541, a Novel Nonnucleoside Inhibitor of the Hepatitis C Virus RNA-Dependent RNA Polymerase
SHI, Stephanie T, HERLIHY, Koleen J, GONZALEZ, Javier, HUI LI, LEWIS, Cristina, PATICK, Amy K, DUGGAL, Rohit, GRAHAM, Joanne P, FUHRMAN, Shella A, DOAN, Chau, PARGE, Hans, HICKEY, Michael, JINGJIN GAO, XIU YU, CHAU, Fannie
Published in Antimicrobial Agents and Chemotherapy (01.02.2008)
Published in Antimicrobial Agents and Chemotherapy (01.02.2008)
Get full text
Journal Article
Discovery of (R)-6-Cyclopentyl-6-(2-(2,6-diethylpyridin-4-yl)ethyl)-3-((5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)methyl)-4-hydroxy-5,6-dihydropyran-2-one (PF-00868554) as a Potent and Orally Available Hepatitis C Virus Polymerase Inhibitor
Li, Hui, Tatlock, John, Linton, Angelica, Gonzalez, Javier, Jewell, Tanya, Patel, Leena, Ludlum, Sarah, Drowns, Matthew, Rahavendran, Sadayappan V, Skor, Heather, Hunter, Robert, Shi, Stephanie T, Herlihy, Koleen J, Parge, Hans, Hickey, Michael, Yu, Xiu, Chau, Fannie, Nonomiya, Jim, Lewis, Cristina
Published in Journal of medicinal chemistry (12.03.2009)
Published in Journal of medicinal chemistry (12.03.2009)
Get full text
Journal Article
Enzymatic Characterization of c-Met Receptor Tyrosine Kinase Oncogenic Mutants and Kinetic Studies with Aminopyridine and Triazolopyrazine Inhibitors
Timofeevski, Sergei L, McTigue, Michele A, Ryan, Kevin, Cui, Jean, Zou, Helen Y, Zhu, Jeff X, Chau, Fannie, Alton, Gordon, Karlicek, Shannon, Christensen, James G, Murray, Brion W
Published in Biochemistry (Easton) (16.06.2009)
Published in Biochemistry (Easton) (16.06.2009)
Get full text
Journal Article
Clinical Pharmacokinetics of Apto-253 Support Its Use As a Novel Agent for the Treatment of Relapsed or Refractory Hematologic Malignancies
Rice, William G., Lightfoot, Jeff, Zhang, Hongying, Cheng, Tiffany, Vellanki, Avanish, Peralta, Robert, Howell, Stephen B, Local, Andrea, Chau, Fannie, Esquivies, Luis
Published in Blood (03.12.2015)
Published in Blood (03.12.2015)
Get full text
Journal Article