Ivacaftor Is Associated with Reduced Lung Infection by Key Cystic Fibrosis Pathogens. A Cohort Study Using National Registry Data
Frost, Freddy J, Nazareth, Dilip S, Charman, Susan C, Winstanley, Craig, Walshaw, Martin J
Published in Annals of the American Thoracic Society (01.11.2019)
Published in Annals of the American Thoracic Society (01.11.2019)
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System-wide biochemical analysis reveals ozonide antimalarials initially act by disrupting Plasmodium falciparum haemoglobin digestion
Giannangelo, Carlo, Siddiqui, Ghizal, De Paoli, Amanda, Anderson, Bethany M, Edgington-Mitchell, Laura E, Charman, Susan A, Creek, Darren J
Published in PLoS pathogens (01.06.2020)
Published in PLoS pathogens (01.06.2020)
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Disease progression in patients with cystic fibrosis treated with ivacaftor: Data from national US and UK registries
Volkova, Nataliya, Moy, Kristin, Evans, Jennifer, Campbell, Daniel, Tian, Simon, Simard, Christopher, Higgins, Mark, Konstan, Michael W., Sawicki, Gregory S., Elbert, Alexander, Charman, Susan C., Marshall, Bruce C., Bilton, Diana
Published in Journal of cystic fibrosis (01.01.2020)
Published in Journal of cystic fibrosis (01.01.2020)
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A Multicentre Study of 5-year Outcomes Following Focal Therapy in Treating Clinically Significant Nonmetastatic Prostate Cancer
Guillaumier, Stephanie, Peters, Max, Arya, Manit, Afzal, Naveed, Charman, Susan, Dudderidge, Tim, Hosking-Jervis, Feargus, Hindley, Richard G., Lewi, Henry, McCartan, Neil, Moore, Caroline M., Nigam, Raj, Ogden, Chris, Persad, Raj, Shah, Karishma, van der Meulen, Jan, Virdi, Jaspal, Winkler, Mathias, Emberton, Mark, Ahmed, Hashim U.
Published in European urology (01.10.2018)
Published in European urology (01.10.2018)
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Transperineal Magnetic Resonance Image Targeted Prostate Biopsy Versus Transperineal Template Prostate Biopsy in the Detection of Clinically Significant Prostate Cancer
Kasivisvanathan, Veeru, Dufour, Robert, Moore, Caroline M, Ahmed, Hashim U, Abd-Alazeez, Mohamed, Charman, Susan C, Freeman, Alex, Allen, Clare, Kirkham, Alex, van der Meulen, Jan, Emberton, Mark
Published in The Journal of urology (01.03.2013)
Published in The Journal of urology (01.03.2013)
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Malarial dihydrofolate reductase as a paradigm for drug development against a resistance-compromised target
Yuthavong, Yongyuth, Tarnchompoo, Bongkoch, Vilaivan, Tirayut, Chitnumsub, Penchit, Kamchonwongpaisan, Sumalee, Charman, Susan A., McLennan, Danielle N., White, Karen L., Vivas, Livia, Bongard, Emily, Thongphanchang, Chawanee, Taweechai, Supannee, Vanichtanankul, Jarunee, Rattanajak, Roonglawan, Arwon, Uthai, Fantauzzi, Pascal, Yuvaniyama, Jirundon, Charman, William N., Matthews, David
Published in Proceedings of the National Academy of Sciences - PNAS (16.10.2012)
Published in Proceedings of the National Academy of Sciences - PNAS (16.10.2012)
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Journal Article
Determinants of Patient Mobility for Prostate Cancer Surgery: A Population-based Study of Choice and Competition
Aggarwal, Ajay, Lewis, Daniel, Charman, Susan C., Mason, Malcolm, Clarke, Noel, Sullivan, Richard, van der Meulen, Jan
Published in European urology (01.06.2018)
Published in European urology (01.06.2018)
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Journal Article
Fluorine Modulates Species Selectivity in the Triazolopyrimidine Class of Plasmodium falciparum Dihydroorotate Dehydrogenase Inhibitors
Deng, Xiaoyi, Kokkonda, Sreekanth, El Mazouni, Farah, White, John, Burrows, Jeremy N, Kaminsky, Werner, Charman, Susan A, Matthews, David, Rathod, Pradipsinh K, Phillips, Margaret A
Published in Journal of medicinal chemistry (26.06.2014)
Published in Journal of medicinal chemistry (26.06.2014)
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Journal Article
The Development Process for Discovery and Clinical Advancement of Modern Antimalarials
Ashton, Trent D, Devine, Shane M, Möhrle, Jörg J, Laleu, Benoît, Burrows, Jeremy N, Charman, Susan A, Creek, Darren J, Sleebs, Brad E
Published in Journal of medicinal chemistry (12.12.2019)
Published in Journal of medicinal chemistry (12.12.2019)
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Journal Article
Synthetic ozonide drug candidate OZ439 offers new hope for a single-dose cure of uncomplicated malaria
Charman, Susan A., Arbe-Barnes, Sarah, Bathurst, Ian C., Brun, Reto, Campbell, Michael, Charman, William N., Chiu, Francis C. K., Chollet, Jacques, Craft, J. Carl, Creek, Darren J., Dong, Yuxiang, Matile, Hugues, Maurer, Melanie, Morizzi, Julia, Nguyen, Tien, Papastogiannidis, Petros, Scheurer, Christian, Shackleford, David M., Sriraghavan, Kamaraj, Stingelin, Lukas, Tang, Yuanqing, Urwyler, Heinrich, Wang, Xiaofang, White, Karen L., Wittlin, Sergio, Zhou, Lin, Vennerstrom, Jonathan L., Wellems, Thomas E.
Published in Proceedings of the National Academy of Sciences - PNAS (15.03.2011)
Published in Proceedings of the National Academy of Sciences - PNAS (15.03.2011)
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Inhibitors of histone acetyltransferases KAT6A/B induce senescence and arrest tumour growth
Baell, Jonathan B, Leaver, David J, Hermans, Stefan J, Kelly, Gemma L, Brennan, Margs S, Downer, Natalie L, Nguyen, Nghi, Wichmann, Johannes, McRae, Helen M, Yang, Yuqing, Cleary, Ben, Lagiakos, H Rachel, Mieruszynski, Stephen, Pacini, Guido, Vanyai, Hannah K, Bergamasco, Maria I, May, Rose E, Davey, Bethany K, Morgan, Kimberly J, Sealey, Andrew J, Wang, Beinan, Zamudio, Natasha, Wilcox, Stephen, Garnham, Alexandra L, Sheikh, Bilal N, Aubrey, Brandon J, Doggett, Karen, Chung, Matthew C, de Silva, Melanie, Bentley, John, Pilling, Pat, Hattarki, Meghan, Dolezal, Olan, Dennis, Matthew L, Falk, Hendrik, Ren, Bin, Charman, Susan A, White, Karen L, Rautela, Jai, Newbold, Andrea, Hawkins, Edwin D, Johnstone, Ricky W, Huntington, Nicholas D, Peat, Thomas S, Heath, Joan K, Strasser, Andreas, Parker, Michael W, Smyth, Gordon K, Street, Ian P, Monahan, Brendon J, Voss, Anne K, Thomas, Tim
Published in Nature (London) (01.08.2018)
Published in Nature (London) (01.08.2018)
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The PICTURE study: diagnostic accuracy of multiparametric MRI in men requiring a repeat prostate biopsy
Simmons, Lucy A M, Kanthabalan, Abi, Arya, Manit, Briggs, Tim, Barratt, Dean, Charman, Susan C, Freeman, Alex, Gelister, James, Hawkes, David, Hu, Yipeng, Jameson, Charles, McCartan, Neil, Moore, Caroline M, Punwani, Shonit, Ramachandran, Navin, van der Meulen, Jan, Emberton, Mark, Ahmed, Hashim U
Published in British journal of cancer (25.04.2017)
Published in British journal of cancer (25.04.2017)
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Journal Article
Endochin-like quinolones are highly efficacious against acute and latent experimental toxoplasmosis
Doggett, J. Stone, Nilsen, Aaron, Forquer, Isaac, Wegmann, Keith W, Jones-Brando, Lorraine, Yolken, Robert H, Bordón, Claudia, Charman, Susan A, Katneni, Kasiram, Schultz, Tracey, Burrows, Jeremy N, Hinrichs, David J, Meunier, Brigitte, Carruthers, Vern B, Riscoe, Michael K
Published in Proceedings of the National Academy of Sciences - PNAS (25.09.2012)
Published in Proceedings of the National Academy of Sciences - PNAS (25.09.2012)
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Journal Article
Ozonide Antimalarial Activity in the Context of Artemisinin-Resistant Malaria
Giannangelo, Carlo, Fowkes, Freya J.I., Simpson, Julie A., Charman, Susan A., Creek, Darren J.
Published in Trends in parasitology (01.07.2019)
Published in Trends in parasitology (01.07.2019)
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Journal Article
The accuracy of multiparametric MRI in men with negative biopsy and elevated PSA level—Can it rule out clinically significant prostate cancer?
Abd-Alazeez, Mohamed, M.Sc. (UROL), M.R.C.S, Ahmed, Hashim U., F.R.C.S. (UROL), Arya, Manit, M.D., F.R.C.S. (UROL), Charman, Susan C., B.Sc. (Hons), M.Sc, Anastasiadis, Eleni, M.R.C.S, Freeman, Alex, F.R.C.Path, Emberton, Mark, M.D, F.R.C.S. (UROL), Kirkham, Alex, M.D., F.R.C.R
Published in Urologic oncology (2014)
Published in Urologic oncology (2014)
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Transformation of Poorly Water-Soluble Drugs into Lipophilic Ionic Liquids Enhances Oral Drug Exposure from Lipid Based Formulations
Sahbaz, Yasemin, Williams, Hywel D, Nguyen, Tri-Hung, Saunders, Jessica, Ford, Leigh, Charman, Susan A, Scammells, Peter J, Porter, Christopher J. H
Published in Molecular pharmaceutics (01.06.2015)
Published in Molecular pharmaceutics (01.06.2015)
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Journal Article
Relationship between Antimalarial Activity and Heme Alkylation for Spiro- and Dispiro-1,2,4-Trioxolane Antimalarials
Creek, Darren J, Charman, William N, Chiu, Francis C K, Prankerd, Richard J, Dong, Yuxiang, Vennerstrom, Jonathan L, Charman, Susan A
Published in Antimicrobial Agents and Chemotherapy (01.04.2008)
Published in Antimicrobial Agents and Chemotherapy (01.04.2008)
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