TH1902, a new docetaxel‐peptide conjugate for the treatment of sortilin‐positive triple‐negative breast cancer
Demeule, Michel, Charfi, Cyndia, Currie, Jean‐Christophe, Larocque, Alain, Zgheib, Alain, Kozelko, Sophie, Béliveau, Richard, Marsolais, Christian, Annabi, Borhane
Published in Cancer science (01.10.2021)
Published in Cancer science (01.10.2021)
Get full text
Journal Article
Corrigendum: Sudocetaxel Zendusortide (TH1902) triggers the cGAS/STING pathway and potentiates anti-PD-L1 immune-mediated tumor cell killing
Demeule, Michel, Currie, Jean-Christophe, Charfi, Cyndia, Zgheib, Alain, Cousineau, Isabelle, Lullier, Véronique, Béliveau, Richard, Marsolais, Christian, Annabi, Borhane
Published in Frontiers in immunology (28.02.2024)
Published in Frontiers in immunology (28.02.2024)
Get full text
Journal Article
The TH1902 Docetaxel Peptide-Drug Conjugate Inhibits Xenografts Growth of Human SORT1-Positive Ovarian and Triple-Negative Breast Cancer Stem-like Cells
Demeule, Michel, Charfi, Cyndia, Currie, Jean-Christophe, Zgheib, Alain, Danalache, Bogdan Alexandru, Béliveau, Richard, Marsolais, Christian, Annabi, Borhane
Published in Pharmaceutics (01.09.2022)
Published in Pharmaceutics (01.09.2022)
Get full text
Journal Article
Decreasing stearoyl‐CoA desaturase‐1 expression inhibits β‐catenin signaling in breast cancer cells
Mauvoisin, Daniel, Charfi, Cyndia, Lounis, Amine M, Rassart, Eric, Mounier, Catherine
Published in Cancer science (01.01.2013)
Published in Cancer science (01.01.2013)
Get full text
Journal Article
Sudocetaxel Zendusortide (TH1902) triggers the cGAS/STING pathway and potentiates anti-PD-L1 immune-mediated tumor cell killing
Demeule, Michel, Currie, Jean-Christophe, Charfi, Cyndia, Zgheib, Alain, Cousineau, Isabelle, Lullier, Véronique, Béliveau, Richard, Marsolais, Christian, Annabi, Borhane
Published in Frontiers in immunology (16.02.2024)
Published in Frontiers in immunology (16.02.2024)
Get full text
Journal Article
New Peptide-Drug Conjugates for Precise Targeting of SORT1-Mediated Vasculogenic Mimicry in the Tumor Microenvironment of TNBC-Derived MDA-MB-231 Breast and Ovarian ES-2 Clear Cell Carcinoma Cells
Charfi, Cyndia, Demeule, Michel, Currie, Jean-Christophe, Larocque, Alain, Zgheib, Alain, Danalache, Bogdan Alexandru, Ouanouki, Amira, Béliveau, Richard, Marsolais, Christian, Annabi, Borhane
Published in Frontiers in oncology (22.10.2021)
Published in Frontiers in oncology (22.10.2021)
Get full text
Journal Article
The Peptide-Drug Conjugate TH1902: A New Sortilin Receptor-Mediated Cancer Therapeutic against Ovarian and Endometrial Cancers
Currie, Jean-Christophe, Demeule, Michel, Charfi, Cyndia, Zgheib, Alain, Larocque, Alain, Danalache, Bogdan Alexandru, Ouanouki, Amira, Béliveau, Richard, Marsolais, Christian, Annabi, Borhane
Published in Cancers (08.04.2022)
Published in Cancers (08.04.2022)
Get full text
Journal Article
Binding and Repressive Activities of Apolipoprotein E3 and E4 Isoforms on the Human ApoD Promoter
Levros, Louis-Charles, Labrie, Marilyne, Charfi, Cyndia, Rassart, Eric
Published in Molecular neurobiology (01.12.2013)
Published in Molecular neurobiology (01.12.2013)
Get full text
Journal Article
Characterization and identification of PARM-1 as a new potential oncogene
Charfi, Cyndia, Levros, Jr, Louis-Charles, Edouard, Elsy, Rassart, Eric
Published in Molecular cancer (31.07.2013)
Published in Molecular cancer (31.07.2013)
Get full text
Journal Article
Characterization of nuclear factors modulating the apolipoprotein D promoter during growth arrest: Implication of PARP-1, APEX-1 and ERK1/2 catalytic activities
Levros, Louis-Charles, Carmo, Sonia Do, Edouard, Elsy, Legault, Philippe, Charfi, Cyndia, Rassart, Eric
Published in Biochimica et biophysica acta (01.09.2010)
Published in Biochimica et biophysica acta (01.09.2010)
Get full text
Journal Article
A Role for the Cavin-3/Matrix Metalloproteinase-9 Signaling Axis in the Regulation of PMA-Activated Human HT1080 Fibrosarcoma Cell Neoplastic Phenotype
Toufaily, Chirine, Charfi, Cyndia, Annabi, Bayader, Annabi, Borhane
Published in Cancer Growth and Metastasis (01.01.2014)
Published in Cancer Growth and Metastasis (01.01.2014)
Get full text
Journal Article
Abstract 1313: TH1902, a docetaxel peptide-drug conjugate, shows pre-clinical efficacy in several Sortilin-positive (SORT1+) cancers
Marsolais, Christian, Currie, Jean-Christophe, Demeule, Michel, Charfi, Cyndia, Larocque, Alain, Zgheib, Alain, Béliveau, Richard, Annabi, Borhane
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Get full text
Journal Article
Abstract 1439: Increasing potency of anticancer drugs through SORT1+ technology: A new targeted approach for the treatment of ovarian and endometrial cancers
Demeule, Michel, Currie, Jean-Christophe, Charfi, Cyndia, Larocque, Alain, Zgheib, Alain, Béliveau, Richard, Marsolais, Christian, Annabi, Borhane
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Get full text
Journal Article
Increasing potency and safety of anticancer drugs through sortilin receptor-mediated cancer therapy: A new targeted approach for the treatment of ovarian cancer
Annabi, Borhane, Demeule, Michel, Currie, Jean-Christophe, Larocque, Alain, Charfi, Cyndia, Béliveau, Richard
Published in Journal of clinical oncology (20.05.2019)
Published in Journal of clinical oncology (20.05.2019)
Get full text
Journal Article
Abstract 1061: Increasing potency of anticancer drugs through Sortilin receptor-mediated cancer therapy: A new targeted approach for the treatment of ovarian cancer
Demeule, Michel, Currie, Jean-Christophe, Charfi, Cyndia, Larocque, Alain, Zgheib, Alain, Kozelko, Sophie, Béliveau, Richard, Marsolais, Christian, Annabi, Borhane
Published in Cancer research (Chicago, Ill.) (15.08.2020)
Published in Cancer research (Chicago, Ill.) (15.08.2020)
Get full text
Journal Article
Abstract 2910: A novel Sortilin-targeted docetaxel peptide conjugate (TH1902), for the treatment of Sortilin-positive (SORT1+) triple-negative breast cancer
Marsolais, Christian, Charfi, Cyndia, Demeule, Michel, Currie, Jean-Christophe, Larocque, Alain, Zgheib, Alain, Duquette, Natacha, Béliveau, Richard, Annabi, Borhane
Published in Cancer research (Chicago, Ill.) (15.08.2020)
Published in Cancer research (Chicago, Ill.) (15.08.2020)
Get full text
Journal Article
Abstract P3-10-07: Receptor-mediated chemotherapy using a new Docetaxel-peptide conjugate for Sortilin-positive triple-negative breast cancer
Demeule, Michel, Charfi, Cyndia, Currie, Jean-Christophe C, Larocque, Alain, Zgheib, Alain, Marsolais, Christian, Béliveau, Richard, Annabi, Borhane
Published in Cancer research (Chicago, Ill.) (15.02.2020)
Published in Cancer research (Chicago, Ill.) (15.02.2020)
Get full text
Journal Article
Abstract 3364: Adaptive mechanisms upon LRP1 repression: Impact on sphingosine-1-phosphate-mediated signalling and migration of brain endothelial cells
Vézina, Amélie, Charfi, Cyndia, Zgheib, Alain, Annabi, Borhane
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Get full text
Journal Article