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Published in Brain (London, England : 1878) (01.05.2013)
Published in Brain (London, England : 1878) (01.05.2013)
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Proteasome-based mechanisms of intrinsic and acquired bortezomib resistance in non-small cell lung cancer
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Published in Biochemical pharmacology (15.01.2012)
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The next generation proteasome inhibitors carfilzomib and oprozomib activate prosurvival autophagy via induction of the unfolded protein response and ATF4
Zang, Yan, Thomas, Sufi M., Chan, Elena T., Kirk, Christopher J., Freilino, Maria L., DeLancey, Hannah M., Grandis, Jennifer R., Li, Changyou, Johnson, Daniel E.
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Carfilzomib and ONX 0912 Inhibit Cell Survival and Tumor Growth of Head and Neck Cancer and Their Activities Are Enhanced by Suppression of Mcl-1 or Autophagy
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Inactivating PSMB5 mutations and P-glycoprotein (multidrug resistance-associated protein/ATP-binding cassette B1) mediate resistance to proteasome inhibitors: ex vivo efficacy of (immuno)proteasome inhibitors in mononuclear blood cells from patients with rheumatoid arthritis
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Published in The Journal of pharmacology and experimental therapeutics (01.04.2012)
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Overcoming bortezomib resistance in human B cells by anti-CD20/rituximab-mediated complement-dependent cytotoxicity and epoxyketone-based irreversible proteasome inhibitors
Verbrugge, Sue Ellen, Al, Marjon, Assaraf, Yehuda G, Niewerth, Denise, van Meerloo, Johan, Cloos, Jacqueline, van der Veer, Michael, Scheffer, George L, Peters, Godefridus J, Chan, Elena T, Anderl, Janet L, Kirk, Christopher J, Zweegman, Sonja, Dijkmans, Ben Ac, Lems, Willem F, Scheper, Rik J, de Gruijl, Tanja D, Jansen, Gerrit
Published in Experimental hematology & oncology (10.01.2013)
Published in Experimental hematology & oncology (10.01.2013)
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Abstract 1022: Carfilzomib demonstrates broad antitumor activity in preclinical lung cancer models
Baker, Amanda F., Sands, Barbara, Carbajal, Lilliana, Anderl, Janet, Chan, Elena T., Kirk, Christopher J., Garland, Linda L.
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Published in Cancer research (Chicago, Ill.) (15.04.2013)
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Sensitivity of Pediatric Acute Leukemia Cells to Bortezomib and Epoxyketone-Based Proteasome Inhibitors: Correlations with Proteasome Subunit Expression
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Published in Blood (18.11.2011)
Published in Blood (18.11.2011)
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Liposomal compositions of epoxyketone-based proteasome inhibitors
Jamaa, Mouhannad, Muchamuel, Tony, Wang, Zhengping, Chan, Elena T, Fang, Ying, Jones, Jeffrey Joseph, Chu, Katherine A, Kirk, Christopher Justin, Jiang, Jing
Year of Publication 17.07.2018
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Year of Publication 17.07.2018
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LIPOSOMAL COMPOSITIONS OF EPOXYKETONE-BASED PROTEASOME INHIBITORS
CHU KATHERINE A, JAMAA MOUHANNAD, WANG ZHENGPING, FANG YING, KIRK CHRISTOPHER JUSTIN, JONES JEFFREY JOSEPH, CHAN ELENA T, MUCHAMUEL TONY, JIANG JING
Year of Publication 30.07.2015
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Year of Publication 30.07.2015
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LIPOSOMAL COMPOSITIONS OF EPOXYKETONE-BASED PROTEASOME INHIBITORS
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Year of Publication 30.07.2015
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Year of Publication 30.07.2015
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