Antitumor activity of a kinesin inhibitor
SAKOWICZ, Roman, FINER, Jeffrey T, CHABALA, John C, GONZALES, Paul, ROTH, Stephanie, WEITMAN, Steve, WOOD, Kenneth W, BERAUD, Christophe, CROMPTON, Anne, LEWIS, Evan, FRITSCH, Alex, LEE, Yan, MAK, John, MOODY, Robert, TURINCIO, Rebecca
Published in Cancer research (Chicago, Ill.) (01.05.2004)
Published in Cancer research (Chicago, Ill.) (01.05.2004)
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Avermectins. Structure determination
Albers-Schoenberg, G, Arison, B. H, Chabala, J. C, Douglas, A. W, Eskola, P, Fisher, M. H, Lusi, A, Mrozik, H, Smith, J. L, Tolman, R. L
Published in Journal of the American Chemical Society (01.07.1981)
Published in Journal of the American Chemical Society (01.07.1981)
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Inhibition of Hydroxymethylglutaryl-Coenzyme A Synthase by L-659,699
Greenspan, Michael D., Yudkovitz, Joel B., Lo, Chia-Yee L., Chen, Julie S., Alberts, Alfred W., Hunt, Vincent M., Chang, Michael N., Yang, Shu Shu, Thompson, Kathryn L., Chiang, Yuan-Ching P., Chabala, John C., Monaghan, Richard L., Schwartz, Robert L.
Published in Proceedings of the National Academy of Sciences - PNAS (01.11.1987)
Published in Proceedings of the National Academy of Sciences - PNAS (01.11.1987)
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(±)-Trans-2-(3-methoxy-5-methylsulfonyl-4-propoxyphenyl)-5-(3,4,5-trimethoxyphenyl)tetrahydrofuran (L-659,989), a novel, potent PAF receptor antagonist
Ponpipom, Mitree M., Hwang, San-Bao, Doebber, Thomas W., Acton, John J., Alberts, Alfred W., Biftu, Tesfaye, Brooker, David R., Bugianesi, Robert L., Chabala, John C., Gamble, Nancy L., Graham, Donald W., Lam, My-Hanh, Wu, Margaret S.
Published in Biochemical and biophysical research communications (15.02.1988)
Published in Biochemical and biophysical research communications (15.02.1988)
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DEVELOPMENT, SYNTHESIS, AND BIOLOGICAL EVALUATION OF (-)-TRANS-(2S,5S)-2-[3-[(2-OXOPROPYL)SULFONYL]-4-NORMAL-PROPOXY-5-(3-HYDROXYPROPOXY)-PHENYL]-5-(3,4,5-TRIMETHOXYPHENYL)TETRAHYDROFURAN, A POTENT ORALLY ACTIVE PLATELET-ACTIVATING-FACTOR (PAF) ANTAGONIST AND ITS WATER-SOLUBLE PRODRUG PHOSPHATE ESTER
GIROTRA, NN, BIFTU, T, PONPIPOM, MM, ACTON, JJ, ALBERTS, AW, BACH, TN, BALL, RG, BUGIANESI, RL, PARSONS, WH, CHABALA, JC, DAVIES, P, DOEBBER, TW, DOHERTY, J, GRAHAM, DW, HWANG, SB, KUO, CH, LAM, MH, LUELL, S, MACINTYRE, DE, MEURER, R, ROBERTS, CD, SAHOO, SP, WU, MS
Published in Journal of medicinal chemistry (18.09.1992)
Published in Journal of medicinal chemistry (18.09.1992)
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Biochemical and pharmacological characterization of L-659,989: an extremely potent, selective and competitive receptor antagonist of platelet-activating factor
SAN-BAO HWANG, MY-HANH LAM, ALBERTS, A. W, BUGIANESI, R. L, CHABALA, J. C, PONPIPOM, M. M
Published in The Journal of pharmacology and experimental therapeutics (01.08.1988)
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Published in The Journal of pharmacology and experimental therapeutics (01.08.1988)
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Benzylated 1,2,3-triazoles as anticoccidiostats
Bochis, Richard J, Chabala, John C, Harris, Ellwood, Peterson, Louis H, Barash, Louis, Beattie, Thomas, Brown, Jeannette E, Graham, Donald W, Waksmunski, Frank S
Published in Journal of medicinal chemistry (01.09.1991)
Published in Journal of medicinal chemistry (01.09.1991)
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Total synthesis of L-659,699, a novel inhibitor of cholesterol biosynthesis
Chiang, Yuan Ching P, Yang, Shu Shu, Heck, James V, Chabala, John C, Chang, Michael N
Published in Journal of organic chemistry (01.11.1989)
Published in Journal of organic chemistry (01.11.1989)
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Journal Article
Absolute configuration of L-659,699, a novel inhibitor of cholesterol biosynthesis
CHIANG, Y.-C. P, CHANG, M. N, SHU SHU YANG, CHABALA, J. C, HECK, J. V
Published in Journal of organic chemistry (16.09.1988)
Published in Journal of organic chemistry (16.09.1988)
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Synthesis and biological activity of MK 287 (L-680,573): a potent, specific and orally active paf receptor antagonist
Sahoo, Soumya P., Graham, Donald W., Acton, John, Biftu, Tesfaye, Bugianesi, Robert L., Girotra, Narindar N., Kuo, Chan-Hwa, Ponpipom, Mitree M., Doebber, Thomas W., Wu, Margaret S., Hwang, San-Bao, Lam, My-Hanh, MacIntyre, D.Euan, Bach, Thomas J., Luell, Silvi, Meurer, Roger, Davies, Philip, Alberts, Alfred W., Chabala, John C.
Published in Bioorganic & medicinal chemistry letters (1991)
Published in Bioorganic & medicinal chemistry letters (1991)
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Synthesis and biological activity of the platelet-activating factor antagonist (±)- trans-2-(3-methoxy-4-phenylsulfonylethoxy-5- n-propylsulfonylphenyl)-5-(3,4,5-trimethoxyphenyl)tetrahydrofuran (L-671,284) and its analogs
Bugianesi, Robert L., Ponpipom, Mitree M., Parsons, William H., Hwang, San-Bao, Doebber, Thomas W., Lam, My-Hanh, Wu, Margaret S., Alberts, Alfred W., Chabala, John C.
Published in Bioorganic & medicinal chemistry letters (1992)
Published in Bioorganic & medicinal chemistry letters (1992)
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The inhibition of cytoplasmic acetoacetyl-CoA thiolase by a triyne carbonate (L-660,631)
Greenspan, Michael D., Yudkovitz, Joel B., Chen, Julie S., Hanf, Darlene P., Chang, Michael N., Chiang, Phoebe Y.C., Chabala, John C., Alberts, Alfred W.
Published in Biochemical and biophysical research communications (30.08.1989)
Published in Biochemical and biophysical research communications (30.08.1989)
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Metabolism of the platelet-activating factor antagonist (+/-)-trans-2-(3'-methoxy-5'-methylsulphonyl-4'-propoxyphenyl)-5-(3",4" ,5"- trimethoxyphenyl)tetrahydrofuran (L-659,989) in rhesus monkeys
Thomson, K L, Chang, M N, Bugianesi, R L, Ponpipom, M M, Arison, B H, Hucker, H B, Sweeney, B M, White, S D, Chabala, J C
Published in Xenobiotica (01.05.1991)
Published in Xenobiotica (01.05.1991)
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Metabolism of kadsurenone and 9,10-dihydrokadsurenone in rhesus monkeys and rat liver microsomes
Thompson, K L, Chang, M N, Chabala, J C, Chiu, S H, Eline, D, Hucker, H B, Sweeney, B M, White, S D, Arison, B H, Smith, J L
Published in Drug metabolism and disposition (01.09.1988)
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Published in Drug metabolism and disposition (01.09.1988)
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1-(substituted)benzyl-5-aminoimidazole-4-carboxamides are potent orally active inhibitors of Trypanosoma cruzi in mice
Chabala, J C, Waits, V B, Ikeler, T, Patchett, A A, Payne, L, Peterson, L H, Reamer, R A, Hoogsteen, K, Wyvratt, M, Hanson, W L
Published in Experientia (15.01.1991)
Published in Experientia (15.01.1991)
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POTENT INHIBITORY EFFECT OF ANTIBIOTIC 1233A ON CHOLESTEROL BIOSYNTHESIS WHICH SPECIFICALLY BLOCKS 3-HYDROXY-3-METHYLGLUTARYL COENZYME A SYNTHASE
OMURA, SATOSHI, TOMODA, HIROSHI, KUMAGAI, HIDETOSHI, GREENSPAN, MICHAEL D., YODKOVITZ, JOEL B., CHEN, JULIE S., ALBERTS, ALFRED W., MARTIN, ISOBEL, MOCHALES, SAGRARIO, MONAGHAN, RICHARD L., CHABALA, JOHN C., SCHWARTZ, ROBERT E., PATCHETT, ARTHUR A.
Published in The Journal of Antibiotics (25.09.1987)
Published in The Journal of Antibiotics (25.09.1987)
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MK 287: a potent, specific, and orally active receptor antagonist of platelet-activating factor
Hwang, S B, Lam, M H, Szalkowski, D M, MacIntyre, D E, Bach, T J, Luell, S, Meuer, R, Sahoo, S P, Alberts, A W, Chabala, J C
Published in Journal of lipid mediators (01.06.1993)
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Published in Journal of lipid mediators (01.06.1993)
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PERI-CARBINOLS
JORDAN, Thomas, A. TA, CHABALA, John, Clifford JC, LING, Ke-Qing, KINNEY, William, A. WA
Year of Publication 06.01.2017
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Year of Publication 06.01.2017
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