Allosteric modulation of metabotropic glutamate receptor 4 activates IDO1-dependent, immunoregulatory signaling in dendritic cells
Volpi, Claudia, Mondanelli, Giada, Pallotta, Maria T., Vacca, Carmine, Iacono, Alberta, Gargaro, Marco, Albini, Elisa, Bianchi, Roberta, Belladonna, Maria L., Celanire, Sylvain, Mordant, Céline, Heroux, Madeleine, Royer-Urios, Isabelle, Schneider, Manfred, Vitte, Pierre-Alain, Cacquevel, Mathias, Galibert, Laurent, Poli, Sonia-Maria, Solari, Aldo, Bicciato, Silvio, Calvitti, Mario, Antognelli, Cinzia, Puccetti, Paolo, Orabona, Ciriana, Fallarino, Francesca, Grohmann, Ursula
Published in Neuropharmacology (01.03.2016)
Published in Neuropharmacology (01.03.2016)
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Characterization of an mGluR2/3 Negative Allosteric Modulator in Rodent Models of Depression
Campo, Brice, Kalinichev, Mikhail, Lambeng, Nathalie, Yacoubi, M. El, Royer-Urios, Isabelle, Schneider, Manfred, Legrand, Coline, Parron, Delphine, Girard, Francoise, Bessif, Abdelhak, Poli, Sonia, Vaugeois, Jean-Marie, Poul, Emmanuel Le, Celanire, Sylvain
Published in Journal of neurogenetics (01.12.2011)
Published in Journal of neurogenetics (01.12.2011)
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Characterization of the novel positive allosteric modulator of the metabotropic glutamate receptor 4 ADX88178 in rodent models of neuropsychiatric disorders
Kalinichev, Mikhail, Le Poul, Emmanuel, Boléa, Christelle, Girard, Françoise, Campo, Brice, Fonsi, Massimiliano, Royer-Urios, Isabelle, Browne, Susan E, Uslaner, Jason M, Davis, Matthew J, Raber, Jacob, Duvoisin, Robert, Bate, Simon T, Reynolds, Ian J, Poli, Sonia, Celanire, Sylvain
Published in The Journal of pharmacology and experimental therapeutics (01.09.2014)
Published in The Journal of pharmacology and experimental therapeutics (01.09.2014)
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Journal Article
HDAC6 억제제로서의 화합물 및 이의 용도
REIS PEDRO JOANA CATARINA, CELANIRE SYLVAIN, ROMBOUTS FREDERIK JAN RITA, SENNHENN PETER CHRISTIAN, CURCIO MICHELE, DOS SANTOS CARVALHO JOAO FERNANDO
Year of Publication 19.08.2024
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Year of Publication 19.08.2024
Patent
Novel metabotropic glutamate receptor 2/3 antagonists and their therapeutic applications: a patent review (2005 - present)
Celanire, Sylvain, Sebhat, Iyassu, Wichmann, Juergen, Mayer, Stanislas, Schann, Stephan, Gatti, Silvia
Published in Expert opinion on therapeutic patents (01.01.2015)
Published in Expert opinion on therapeutic patents (01.01.2015)
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Journal Article
A convenient synthesis of cyclopenta[b]pyridin-2,5-dione as a non- glycosidic cardiotonic agent
Robert, Nicolas, Verrier, Cécile, Hoarau, Christophe, Célanire, Sylvain, Marsais, Francis
Published in ARKIVOC (01.01.2008)
Published in ARKIVOC (01.01.2008)
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Web Resource
NADPH 산화효소 저해제로서의 신규한 화합물
MACHIN PETER, CELANIRE SYLVAIN, SHARPE ANDREW, WISHART GRANT, PERRY BENJAMIN, CHAMBERS MARK, HEITZ FREDDY, HODGES ALASTAIR
Year of Publication 11.06.2021
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Year of Publication 11.06.2021
Patent
Lead Optimization of Thiazolo[5,4-c]piperidines: 3-Cyclobutoxy Linker as a Key Spacer for H3R Inverse Agonists
Provins, Laurent, Denonne, Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie-Laure, Demaude, Thierry, Durieu, Véronique, Gillard, Michel, Hubert, Delphine, Lamberty, Yves, Lorent, Geneviève, Valade, Anne, Vanbellinghen, Alain, Van houtvin, Nathalie
Published in ChemMedChem (01.12.2012)
Published in ChemMedChem (01.12.2012)
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Targeting type-2 metabotropic glutamate receptors to protect vulnerable hippocampal neurons against ischemic damage
Motolese, Marta, Mastroiacovo, Federica, Cannella, Milena, Bucci, Domenico, Gaglione, Anderson, Riozzi, Barbara, Lütjens, Robert, Poli, Sonia M, Celanire, Sylvain, Bruno, Valeria, Battaglia, Giuseppe, Nicoletti, Ferdinando
Published in Molecular brain (24.10.2015)
Published in Molecular brain (24.10.2015)
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Journal Article
Acetamide Scanning around Bicyclic Thiazoles: SAR at the H 3 Receptor
Denonne , Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie‐Laure, Detrait, Eric, Durieu, Véronique, Gillard, Michel, Lamberty, Yves, Lorent, Geneviève, Nicolas, Jean‐Marie, Vanbellinghen, Alain, Van Houtvin, Nathalie, Provins, Laurent
Published in ChemMedChem (05.09.2011)
Published in ChemMedChem (05.09.2011)
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Journal Article
Phenyl‐oxazoles, a New Family of Inverse Agonists at the H 3 Histamine Receptor
Denonne, Frédéric, Atienzar, Franck, Célanire, Sylvain, Christophe, Bernard, Delannois, Frédérique, Delaunoy, Christel, Delporte, Marie‐Laure, Durieu, Véronique, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lorent, Geneviève, Vanbellinghen, Alain, Van houtvin, Nathalie, Verbois, Valérie, Provins, Laurent
Published in ChemMedChem (01.02.2010)
Published in ChemMedChem (01.02.2010)
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Journal Article
Keynote review: Histamine H3 receptor antagonists reach out for the clinic
Celanire, Sylvain, Wijtmans, Maikel, Talaga, Patrice, Leurs, Rob, de Esch, Iwan J.P.
Published in Drug discovery today (01.12.2005)
Published in Drug discovery today (01.12.2005)
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Journal Article
Discovery of a New Class of Non‐imidazole Oxazoline‐Based Histamine H 3 Receptor (H 3 R) Inverse Agonists
Célanire, Sylvain, Wijtmans, Maikel, Christophe, Bernard, Collart, Philippe, de Esch, Iwan, Dassesse, Donald, Delaunoy, Christel, Denonne, Frédéric, Durieu, Véronique, Gelens, Edith, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lebon, Florence, Nicolas, Jean‐Marie, Quéré, Luc, Snip, Erwin, Vanbellinghen, Alain, Van houtvin, Nathalie, Verbois, Valérie, Timmerman, Henk, Talaga, Patrice, Leurs, Rob, Provins, Laurent
Published in ChemMedChem (06.07.2009)
Published in ChemMedChem (06.07.2009)
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Journal Article
4-benzyl-1H-imidazoles with oxazoline termini as histamine H-3 receptor agonists
Wijtmans, Maikel, Celanire, Sylvain, Snip, Erwin, Gillard, Michel R., Gelens, Edith, Collart, Philippe P., Venhuis, Bastiaan J., Christophe, Bernard, Hulscher, Saskia, van der Goot, Henk, Lebon, Florence, Timmerman, Henk, Bakker, Remko A., Lallemand, Benedicte I. L. F., Leurs, Rob, Talaga, Patrice E., de Esch, Iwan J. P.
Published in Journal of medicinal chemistry (22.05.2008)
Published in Journal of medicinal chemistry (22.05.2008)
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