Imidazopyridine-5,6,7,8-tetrahydro-8-quinolinamine derivatives with potent activity against HIV-1
Gudmundsson, Kristjan S., Boggs, Sharon D., Catalano, John G., Svolto, Angilique, Spaltenstein, Andrew, Thomson, Michael, Wheelan, Pat, Jenkinson, Stephen
Published in Bioorganic & medicinal chemistry letters (15.11.2009)
Published in Bioorganic & medicinal chemistry letters (15.11.2009)
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Journal Article
Hepatitis C Replication Inhibitors That Target the Viral NS4B Protein
Miller, John F., Chong, Pek Y., Shotwell, J. Brad, Catalano, John G., Tai, Vincent W.-F., Fang, Jing, Banka, Anna L., Roberts, Christopher D., Youngman, Michael, Zhang, Huichang, Xiong, Zhiping, Mathis, Amanda, Pouliot, Jeffery J., Hamatake, Robert K., Price, Daniel J., Seal, John W., Stroup, Lisa L., Creech, Katrina L., Carballo, Luz H., Todd, Dan, Spaltenstein, Andrew, Furst, Sylvia, Hong, Zhi, Peat, Andrew J.
Published in Journal of medicinal chemistry (13.03.2014)
Published in Journal of medicinal chemistry (13.03.2014)
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Journal Article
Amine substituted N-(1 H-benzimidazol-2ylmethyl)-5,6,7,8-tetrahydro-8-quinolinamines as CXCR4 antagonists with potent activity against HIV-1
Gudmundsson, Kristjan S., Sebahar, Paul R., Richardson, Leah D’Aurora, Miller, John F., Turner, Elizabeth M., Catalano, John G., Spaltenstein, Andrew, Lawrence, Wendell, Thomson, Michael, Jenkinson, Stephen
Published in Bioorganic & medicinal chemistry letters (01.09.2009)
Published in Bioorganic & medicinal chemistry letters (01.09.2009)
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Journal Article
Substituted tetrahydrocarbazoles with potent activity against human papillomaviruses
Gudmundsson, Kristjan S., Sebahar, Paul R., Richardson, Leah D’Aurora, Catalano, John G., Boggs, Sharon D., Spaltenstein, Andrew, Sethna, Phiroze B., Brown, Kevin W., Harvey, Robert, Romines, Karen R.
Published in Bioorganic & medicinal chemistry letters (01.07.2009)
Published in Bioorganic & medicinal chemistry letters (01.07.2009)
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Journal Article
Synthesis of a novel tricyclic 1,2,3,4,4a,5,6,10b-octahydro-1,10-phenanthroline ring system and CXCR4 antagonists with potent activity against HIV-1
Catalano, John G., Gudmundsson, Kristjan S., Svolto, Angilique, Boggs, Sharon D., Miller, John F., Spaltenstein, Andrew, Thomson, Michael, Wheelan, Pat, Minick, Doug J., Phelps, Dean P., Jenkinson, Stephen
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
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Journal Article
화학적 화합물
DICKSON HAMILTON D, WEATHERHEAD JASON GORDON, CHONG PEK YOKE, CATALANO JOHN G, LEIVERS MARTIN R
Year of Publication 08.06.2020
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Year of Publication 08.06.2020
Patent
Acyclic, orally bioavailable ketone-based cathepsin K inhibitors
Barrett, David G., Catalano, John G., Deaton, David N., Long, Stacey T., McFadyen, Robert B., Miller, Aaron B., Miller, Larry R., Samano, Vicente, Tavares, Francis X., Wells-Knecht, Kevin J., Wright, Lois L., Zhou, Hui-Qiang Q.
Published in Bioorganic & medicinal chemistry letters (2007)
Published in Bioorganic & medicinal chemistry letters (2007)
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Journal Article
Design of small molecule ketoamide-based inhibitors of cathepsin K
Catalano, John G., Deaton, David N., Long, Stacey T., McFadyen, Robert B., Miller, Larry R., Payne, J.Alan, Wells-Knecht, Kevin J., Wright, Lois L.
Published in Bioorganic & medicinal chemistry letters (09.02.2004)
Published in Bioorganic & medicinal chemistry letters (09.02.2004)
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Journal Article
A structural screening approach to ketoamide-based inhibitors of cathepsin K
Barrett, David G., Catalano, John G., Deaton, David N., Long, Stacey T., McFadyen, Robert B., Miller, Aaron B., Miller, Larry R., Wells-Knecht, Kevin J., Wright, Lois L.
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
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Journal Article
Orally bioavailable small molecule ketoamide-based inhibitors of cathepsin K
Barrett, David G., Catalano, John G., Deaton, David N., Long, Stacey T., Miller, Larry R., Tavares, Francis X., Wells-Knecht, Kevin J., Wright, Lois L., Zhou, Hui-Qiang Q.
Published in Bioorganic & medicinal chemistry letters (17.05.2004)
Published in Bioorganic & medicinal chemistry letters (17.05.2004)
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Journal Article
Novel, potent P2–P3 pyrrolidine derivatives of ketoamide-based cathepsin K inhibitors
Barrett, David G., Catalano, John G., Deaton, David N., Hassell, Anne M., Long, Stacey T., Miller, Aaron B., Miller, Larry R., Ray, John A., Samano, Vicente, Shewchuk, Lisa M., Wells-Knecht, Kevin J., Willard, Derril H., Wright, Lois L.
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
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Journal Article
P2-P3 conformationally constrained ketoamide-based inhibitors of cathepsin K
BARRETT, David G, BONCEK, Virginia M, PAYNE, J. Alan, RAY, John A, SAMANO, Vicente, SHEWCHUK, Lisa M, TAVARES, Francis X, WELLS-KNECHT, Kevin J, WILLARD, Derril H, WRIGHT, Lois L, ZHOU, Hui-Qiang Q, CATALANO, John G, DEATON, David N, HASSELL, Anne M, JURGENSEN, Cynthia H, LONG, Stacey T, MCFADYEN, Robert B, MILLER, Aaron B, MILLER, Larry R
Published in Bioorganic & medicinal chemistry letters (01.08.2005)
Published in Bioorganic & medicinal chemistry letters (01.08.2005)
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Journal Article
Potent and selective P2-P3 ketoamide inhibitors of cathepsin K with good pharmacokinetic properties via favorable P1', P1, and/or P3 substitutions
BARRETT, David G, CATALANO, John G, WRIGHT, Lois L, DEATON, David N, HASSELL, Anne M, LONG, Stacey T, MILLER, Aaron B, MILLER, Larry R, SHEWCHUK, Lisa M, WELLS-KNECHT, Kevin J, WILLARD, Derril H
Published in Bioorganic & medicinal chemistry letters (04.10.2004)
Published in Bioorganic & medicinal chemistry letters (04.10.2004)
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Journal Article
Exploration of the P1 SAR of aldehyde cathepsin K inhibitors
CATALANO, John G, DEATON, David N, FURFINE, Eric S, HASSELL, Annie M, MCFADYEN, Robert B, MILLER, Aaron B, MILLER, Larry R, SHEWCHUK, Lisa M, WILLARD, Derril H, WRIGHT, Lois L
Published in Bioorganic & medicinal chemistry letters (05.01.2004)
Published in Bioorganic & medicinal chemistry letters (05.01.2004)
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Journal Article
Phenoxide leaving group SNAr strategy for the facile preparation of 7-amino-3-aryl pyrazolo[1,5-a]pyrimidines from a 3-bromo-7-phenoxypyrazolo[1,5-a]pyrimidine intermediate
Catalano, John G., Gaitonde, Vishwanath, Beesu, Mallesh, Leivers, Anna L., Shotwell, J. Brad
Published in Tetrahedron letters (28.10.2015)
Published in Tetrahedron letters (28.10.2015)
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Journal Article
Structure/Activity Relationships in Lysophosphatidic Acid: The 2-Hydroxyl Moiety
Lynch, K R, Hopper, D W, Carlisle, S J, Catalano, J G, Zhang, M, MacDonald, T L
Published in Molecular pharmacology (01.07.1997)
Published in Molecular pharmacology (01.07.1997)
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Journal Article
ChemInform Abstract: Phenoxide Leaving Group SNAr Strategy for the Facile Preparation of 7‐Amino‐3‐aryl Pyrazolo[1,5‐a]pyrimidines from a 3‐Bromo‐7‐phenoxypyrazolo[1,5‐a]pyrimidine Intermediate
Catalano, John G., Gaitonde, Vishwanath, Beesu, Mallesh, Leivers, Anna L., Shotwell, J. Brad
Published in ChemInform (01.02.2016)
Published in ChemInform (01.02.2016)
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Journal Article
Facile synthesis of lysophospholipids containing unsaturated fatty acid chains
Hopper, Darrin W., Catalano, John G., Macdonald, Timothy L.
Published in Tetrahedron letters (28.10.1996)
Published in Tetrahedron letters (28.10.1996)
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Journal Article
Amine substituted N-(1H-benzimidazol-2ylmethyl)-5,6,7,8-tetrahydro-8-quinolin amines as CXCR4 antagonists with potent activity against HIV-1
Gudmundsson, Kristjan S, Sebahar, Paul R, Richardson, Leah DAurora, Miller, John F, Turner, Elizabeth M, Catalano, John G, Spaltenstein, Andrew, Lawrence, Wendell, Thomson, Michael, Jenkinson, Stephen
Published in Bioorganic & medicinal chemistry letters (01.09.2009)
Published in Bioorganic & medicinal chemistry letters (01.09.2009)
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Journal Article
P 2–P 3 conformationally constrained ketoamide-based inhibitors of cathepsin K
Barrett, David G., Boncek, Virginia M., Catalano, John G., Deaton, David N., Hassell, Anne M., Jurgensen, Cynthia H., Long, Stacey T., McFadyen, Robert B., Miller, Aaron B., Miller, Larry R., Payne, J. Alan, Ray, John A., Samano, Vicente, Shewchuk, Lisa M., Tavares, Francis X., Wells-Knecht, Kevin J., Willard, Derril H., Wright, Lois L., Zhou, Hui-Qiang Q.
Published in Bioorganic & medicinal chemistry letters (01.08.2005)
Published in Bioorganic & medicinal chemistry letters (01.08.2005)
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Journal Article