Dolutegravir (S/GSK1349572) Exhibits Significantly Slower Dissociation than Raltegravir and Elvitegravir from Wild-Type and Integrase Inhibitor-Resistant HIV-1 Integrase-DNA Complexes
HIGHTOWER, Kendra E, WANG, Ruolan, SEKI, Takahiro, KOBAYASHI, Masanori, UNDERWOOD, Mark R, DEANDA, Felix, JOHNS, Brian A, WEAVER, Kurt, YINGNIAN SHEN, TOMBERLIN, Ginger H, LUKE CARTER, H, BRODERICK, Timothy, SIGETHY, Scott
Published in Antimicrobial Agents and Chemotherapy (01.10.2011)
Published in Antimicrobial Agents and Chemotherapy (01.10.2011)
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A pre-steady state and steady state kinetic analysis of the N-ribosyl hydrolase activity of hCD157
Preugschat, Frank, Carter, Luke H., Boros, Eric E., Porter, David J.T., Stewart, Eugene L., Shewchuk, Lisa M.
Published in Archives of biochemistry and biophysics (15.12.2014)
Published in Archives of biochemistry and biophysics (15.12.2014)
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Impact of Common Epidermal Growth Factor Receptor and HER2 Variants on Receptor Activity and Inhibition by Lapatinib
GILMER, Tona M, CABLE, Louann, WOOD, Edgar R, ALLIGOOD, Krystal, RUSNAK, David, SPEHAR, Glenn, GALLAGHER, Kathleen T, WOLDU, Ermias, CARTER, H. Luke, TRUESDALE, Anne T, SHEWCHUK, Lisa
Published in Cancer research (Chicago, Ill.) (15.01.2008)
Published in Cancer research (Chicago, Ill.) (15.01.2008)
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TIMP-3 Inhibition of ADAMTS-4 (Aggrecanase-1) Is Modulated by Interactions between Aggrecan and the C-terminal Domain of ADAMTS-4
Wayne, Gareth J., Deng, Su-Jun, Amour, Augustin, Borman, Satty, Matico, Rosalie, Carter, H. Luke, Murphy, Gillian
Published in The Journal of biological chemistry (20.07.2007)
Published in The Journal of biological chemistry (20.07.2007)
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Crystallization of protein-ligand complexes
Hassell, Anne M., An, Gang, Bledsoe, Randy K., Bynum, Jane M., Carter III, H. Luke, Deng, Su-Jun J., Gampe, Robert T., Grisard, Tamara E., Madauss, Kevin P., Nolte, Robert T., Rocque, Warren J., Wang, Liping, Weaver, Kurt L., Williams, Shawn P., Wisely, G. Bruce, Xu, Robert, Shewchuk, Lisa M.
Published in Acta crystallographica. Section D, Biological crystallography. (01.01.2007)
Published in Acta crystallographica. Section D, Biological crystallography. (01.01.2007)
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Potent Inhibitors of HIV-1 Integrase Display a Two-Step, Slow-Binding Inhibition Mechanism Which Is Absent in a Drug-Resistant T66I/M154I Mutant
Garvey, Edward P, Schwartz, Benjamin, Gartland, Margaret J, Lang, Scott, Halsey, Wendy, Sathe, Ganesh, Carter, H. Luke, Weaver, Kurt L
Published in Biochemistry (Easton) (24.02.2009)
Published in Biochemistry (Easton) (24.02.2009)
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Journal Article
Substrate Specificity of Human Collagenase 3 Assessed Using a Phage-displayed Peptide Library
Deng, Su-Jun, Bickett, D. Mark, Mitchell, Justin L., Lambert, Millard H., Blackburn, R. Kevin, Carter, H. Luke, Neugebauer, Jennifer, Pahel, Gregory, Weiner, Michael P., Moss, Marcia L.
Published in The Journal of biological chemistry (06.10.2000)
Published in The Journal of biological chemistry (06.10.2000)
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Journal Article
Inhibition of Wild-Type and Mutant Human Immunodeficiency Virus Type 1 Proteases by GW0385 and Other Arylsulfonamides
Hanlon, Mary H, Porter, David J. T, Furfine, Eric S, Spaltenstein, Andrew, Carter, H. Luke, Danger, Dana, Shu, Arthur Y. L, Kaldor, Istvan W, Miller, John F, Samano, Vicente A
Published in Biochemistry (Easton) (16.11.2004)
Published in Biochemistry (Easton) (16.11.2004)
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Journal Article
Effectors of HIV-1 Protease Peptidolytic Activity
Porter, David J. T, Hanlon, Mary H, Carter, Luke H, Danger, Dana P, Furfine, Eric S
Published in Biochemistry (Easton) (18.09.2001)
Published in Biochemistry (Easton) (18.09.2001)
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Pyrrolidinyl pyridone and pyrazinone analogues as potent inhibitors of prolyl oligopeptidase (POP)
Haffner, Curt D., Diaz, Caroline J., Miller, Aaron B., Reid, Robert A., Madauss, Kevin P., Hassell, Annie, Hanlon, Mary H., Porter, David J.T., Becherer, J. David, Carter, Luke H.
Published in Bioorganic & medicinal chemistry (01.08.2008)
Published in Bioorganic & medicinal chemistry (01.08.2008)
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Anthranilimide based glycogen phosphorylase inhibitors for the treatment of type 2 diabetes. Part 3: X-ray crystallographic characterization, core and urea optimization and in vivo efficacy
Thomson, Stephen A., Banker, Pierette, Bickett, D. Mark, Boucheron, Joyce A., Carter, H. Luke, Clancy, Daphne C., Cooper, Joel P., Dickerson, Scott H., Garrido, Dulce M., Nolte, Robert T., Peat, Andrew J., Sheckler, Lauren R., Sparks, Steven M., Tavares, Francis X., Wang, Liping, Wang, Tony Y., Weiel, James E.
Published in Bioorganic & medicinal chemistry letters (15.02.2009)
Published in Bioorganic & medicinal chemistry letters (15.02.2009)
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Journal Article
Discovery of an inhibitor of insulin-like growth factor 1 receptor activation: Implications for cellular potency and selectivity over insulin receptor
Wood, Edgar R., Shewchuk, Lisa, Hassel, Anne, Nichols, Jim, Truesdale, Anne T., Smith, Danielle, Carter, H. Luke, Weaver, Kurt, Barrett, George, Leesnitzer, Tony, Alvarez, Emilio, Bardera, Ana Isabel, Alamillo, Amelia, Cantizani, Juan, Martin, Julio, Smith, Gary K., Jensen, David E., Xie, Hongbo, Mook, Robert, Kumar, Rakesh, Kuntz, Kevin
Published in Biochemical pharmacology (15.12.2009)
Published in Biochemical pharmacology (15.12.2009)
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Specific Sequence Elements Are Required for the Expression of Functional Tumor Necrosis Factor-α-converting Enzyme (TACE)
Milla, Marcos E., Leesnitzer, M. Anthony, Moss, Marcia L., Clay, William C., Carter, H. Luke, Miller, Ann B., Su, Jui-Lan, Lambert, Millard H., Willard, Derril H., Sheeley, Douglas M., Kost, Thomas A., Burkhart, William, Moyer, Mary, Blackburn, R. Kevin, Pahel, Gregory L., Mitchell, Justin L., Hoffman, Christine R., Becherer, J. David
Published in The Journal of biological chemistry (22.10.1999)
Published in The Journal of biological chemistry (22.10.1999)
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Comparison of the biochemical and kinetic properties of the type 1 receptor tyrosine kinase intracellular domains. Demonstration of differential sensitivity to kinase inhibitors
Brignola, Perry S, Lackey, Karen, Kadwell, Sue H, Hoffman, Christine, Horne, Earnest, Carter, H Luke, Stuart, J Darren, Blackburn, Kevin, Moyer, Mary B, Alligood, Krystal J, Knight, Wilson B, Wood, Edgar R
Published in The Journal of biological chemistry (11.01.2002)
Published in The Journal of biological chemistry (11.01.2002)
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Journal Article
Anthranilimide-based glycogen phosphorylase inhibitors for the treatment of type 2 diabetes: 1. Identification of 1-amino-1-cycloalkyl carboxylic acid headgroups
Sparks, Steven M., Banker, Pierette, Bickett, David M., Carter, H. Luke, Clancy, Daphne C., Dickerson, Scott H., Dwornik, Kate A., Garrido, Dulce M., Golden, Pamela L., Nolte, Robert T., Peat, Andrew J., Sheckler, Lauren R., Tavares, Francis X., Thomson, Stephen A., Wang, Liping, Weiel, James E.
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
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Journal Article
Kinetic Analysis of the Effects of Mutagenesis of W501 and V432 of the Hepatitis C Virus NS3 Helicase Domain on ATPase and Strand-Separating Activity
Preugschat, Frank, Danger, Dana P, Carter, Luke H, Davis, Roderick G, Porter, David J. T
Published in Biochemistry (Easton) (02.05.2000)
Published in Biochemistry (Easton) (02.05.2000)
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Journal Article
Comparison of the Biochemical and Kinetic Properties of the Type 1 Receptor Tyrosine Kinase Intracellular Domains
Brignola, Perry S., Lackey, Karen, Kadwell, Sue H., Hoffman, Christine, Horne, Earnest, Carter, H. Luke, Stuart, J. Darren, Blackburn, Kevin, Moyer, Mary B., Alligood, Krystal J., Knight, Wilson B., Wood, Edgar R.
Published in The Journal of biological chemistry (11.01.2002)
Published in The Journal of biological chemistry (11.01.2002)
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Journal Article
Erratum: Cloning of a disintegrin metalloproteinase that processes precursor tumour-necrosis factor-α
Moss, Marcia L., Jin, S.-L. Catherine, Milla, Marcos E., Bickett, D. Mark, Burkhart, William, Carter, H. Luke, Chen, Wen-Ji, William, C., Didsbury, John R., Hassler, Daniel, Hoffman, Christine R., Kost, Thomas A., Lambert, Millard H., Leesnitzer, M. Anthony, McCauley, Philip, McGeehan, Gerard, Mitchell, Justin, Moyer, Mary, Pahel, Gregory, Rocque, Warren, Overton, Laurie K., Schoenen, Frank, Seaton, Theresa, Su, Jui-Lan, Warner, Janet, Willard, Derril, Becherer, J. David
Published in Nature (London) (17.04.1997)
Published in Nature (London) (17.04.1997)
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Journal Article
Cloning of a disintegrin metalloproteinase that processes precursor tumour-necrosis factor-α
Moss, Marcia L, Jin, S.-L. Catherine, Milla, Marcos E, Burkhart, William, Carter, H. Luke, Chen, Wen-Ji, Clay, William C, Didsbury, John R, Hassler, Daniel, Hoffman, Christine R, Kost, Thomas A, Lambert, Millard H, Leesnitzer, M. Anthony, McCauley, Philip, McGeehan, Gerard, Mitchell, Justin, Moyer, Mary, Pahel, Gregory, Rocque, Warren, Overton, Laurie K, Schoenen, Frank, Seaton, Theresa, Su, Jui-Lan, Warner, Janet, Willard, Derril, Becherer, J. David
Published in Nature (London) (20.02.1997)
Published in Nature (London) (20.02.1997)
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Syntheses and Biological Activities of a Novel Group of Steroidal Derived Inhibitors for Human CDC25A Protein Phosphatase
Peng, Hairuo, Xie, Wenge, Otterness, Diane M, Cogswell, John P, McConnell, Randy T, Carter, H. Luke, Powis, Garth, Abraham, Robert T, Zalkow, Leon H
Published in Journal of medicinal chemistry (01.03.2001)
Published in Journal of medicinal chemistry (01.03.2001)
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