Novel Class of Benzoic Acid Ester Derivatives as Potent PDE4 Inhibitors for Inhaled Administration in the Treatment of Respiratory Diseases
Armani, Elisabetta, Amari, Gabriele, Rizzi, Andrea, Fanti, Renato De, Ghidini, Eleonora, Capaldi, Carmelida, Carzaniga, Laura, Caruso, Paola, Guala, Matilde, Peretto, Ilaria, La Porta, Elena, Bolzoni, Pier T, Facchinetti, Fabrizio, Carnini, Chiara, Moretto, Nadia, Patacchini, Riccardo, Bassani, Franco, Cenacchi, Valentina, Volta, Roberta, Amadei, Francesco, Capacchi, Silvia, Delcanale, Maurizio, Puccini, Paola, Catinella, Silvia, Civelli, Maurizio, Villetti, Gino
Published in Journal of medicinal chemistry (13.02.2014)
Published in Journal of medicinal chemistry (13.02.2014)
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Microwave-assisted solid phase synthesis of Imatinib, a blockbuster anticancer drug
Leonetti, Francesco, Capaldi, Carmelida, Carotti, Angelo
Published in Tetrahedron letters (01.05.2007)
Published in Tetrahedron letters (01.05.2007)
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Design, Synthesis, and Biological Characterization of Inhaled p38?/? MAPK Inhibitors for the Treatment of Lung Inflammatory Diseases
Armani, Elisabetta, Capaldi, Carmelida, Bagnacani, Valentina, Saccani, Francesca, Aquino, Giancarlo, Puccini, Paola, Facchinetti, Fabrizio, Martucci, Cataldo, Moretto, Nadia, Villetti, Gino, Patacchini, Riccardo, Civelli, Maurizio, Hurley, Chris, Jennings, Andrew, Alcaraz, Lilian, Bloomfield, Dawn, Briggs, Michael, Daly, Stephen, Panchal, Terry, Russell, Vince, Wicks, Sharon, Finch, Harry, Fitzgerald, Mary, Fox, Craig, Delcanale, Maurizio
Published in Journal of medicinal chemistry (26.05.2022)
Published in Journal of medicinal chemistry (26.05.2022)
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Discovery of M-3 Antagonist-PDE4 Inhibitor Dual Pharmacology Molecules for the Treatment of Chronic Obstructive Pulmonary Disease
Armani, Elisabetta, Rizzi, Andrea, Capaldi, Carmelida, De Fanti, Renato, Delcanale, Maurizio, Villetti, Gino, Marchini, Gessica, Pisano, Anna Rita, Pitozzi, Vanessa, Pittelli, Maria Gloria, Trevisani, Marcello, Salvadori, Michela, Cenacchi, Valentina, Puccini, Paola, Amadei, Francesco, Pappani, Alice, Civelli, Maurizio, Patacchini, Riccardo, Baker-Glenn, Charles A. G., Van de Poel, Herve, Blackaby, Wesley P., Nash, Kevin, Amari, Gabriele
Published in Journal of medicinal chemistry (08.07.2021)
Published in Journal of medicinal chemistry (08.07.2021)
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CHF6001 I: a novel highly potent and selective phosphodiesterase 4 inhibitor with robust anti-inflammatory activity and suitable for topical pulmonary administration
Moretto, Nadia, Caruso, Paola, Bosco, Raffaella, Marchini, Gessica, Pastore, Fiorella, Armani, Elisabetta, Amari, Gabriele, Rizzi, Andrea, Ghidini, Eleonora, De Fanti, Renato, Capaldi, Carmelida, Carzaniga, Laura, Hirsch, Emilio, Buccellati, Carola, Sala, Angelo, Carnini, Chiara, Patacchini, Riccardo, Delcanale, Maurizio, Civelli, Maurizio, Villetti, Gino, Facchinetti, Fabrizio
Published in The Journal of pharmacology and experimental therapeutics (01.03.2015)
Published in The Journal of pharmacology and experimental therapeutics (01.03.2015)
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Journal Article
Design, Synthesis, and Biological Characterization of Inhaled p38α/β MAPK Inhibitors for the Treatment of Lung Inflammatory Diseases
Armani, Elisabetta, Capaldi, Carmelida, Bagnacani, Valentina, Saccani, Francesca, Aquino, Giancarlo, Puccini, Paola, Facchinetti, Fabrizio, Martucci, Cataldo, Moretto, Nadia, Villetti, Gino, Patacchini, Riccardo, Civelli, Maurizio, Hurley, Chris, Jennings, Andrew, Alcaraz, Lilian, Bloomfield, Dawn, Briggs, Michael, Daly, Stephen, Panchal, Terry, Russell, Vince, Wicks, Sharon, Finch, Harry, Fitzgerald, Mary, Fox, Craig, Delcanale, Maurizio
Published in Journal of medicinal chemistry (26.05.2022)
Published in Journal of medicinal chemistry (26.05.2022)
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Journal Article
Discovery of M3 Antagonist-PDE4 Inhibitor Dual Pharmacology Molecules for the Treatment of Chronic Obstructive Pulmonary Disease
Armani, Elisabetta, Rizzi, Andrea, Capaldi, Carmelida, De Fanti, Renato, Delcanale, Maurizio, Villetti, Gino, Marchini, Gessica, Pisano, Anna Rita, Pitozzi, Vanessa, Pittelli, Maria Gloria, Trevisani, Marcello, Salvadori, Michela, Cenacchi, Valentina, Puccini, Paola, Amadei, Francesco, Pappani, Alice, Civelli, Maurizio, Patacchini, Riccardo, Baker-Glenn, Charles A.G, Van de Poël, Hervé, Blackaby, Wesley P, Nash, Kevin, Amari, Gabriele
Published in Journal of medicinal chemistry (08.07.2021)
Published in Journal of medicinal chemistry (08.07.2021)
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Journal Article
Discovery and Optimization of Thiazolidinyl and Pyrrolidinyl Derivatives as Inhaled PDE4 Inhibitors for Respiratory Diseases
Carzaniga, Laura, Amari, Gabriele, Rizzi, Andrea, Capaldi, Carmelida, De Fanti, Renato, Ghidini, Eleonora, Villetti, Gino, Carnini, Chiara, Moretto, Nadia, Facchinetti, Fabrizio, Caruso, Paola, Marchini, Gessica, Battipaglia, Loredana, Patacchini, Riccardo, Cenacchi, Valentina, Volta, Roberta, Amadei, Francesco, Pappani, Alice, Capacchi, Silvia, Bagnacani, Valentina, Delcanale, Maurizio, Puccini, Paola, Catinella, Silvia, Civelli, Maurizio, Armani, Elisabetta
Published in Journal of medicinal chemistry (28.12.2017)
Published in Journal of medicinal chemistry (28.12.2017)
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Journal Article
Solid-Phase Synthesis and Insights into Structure−Activity Relationships of Safinamide Analogues as Potent and Selective Inhibitors of Type B Monoamine Oxidase
Leonetti, Francesco, Capaldi, Carmelida, Pisani, Leonardo, Nicolotti, Orazio, Muncipinto, Giovanni, Stefanachi, Angela, Cellamare, Saverio, Caccia, Carla, Carotti, Angelo
Published in Journal of medicinal chemistry (04.10.2007)
Published in Journal of medicinal chemistry (04.10.2007)
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Journal Article
1-PHENYL-2-PYRIDINYL ALKYL ALCOHOL DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS
CARZANIGA, LAURA, ESPOSITO, ORIANA, ARMANI, ELISABETTA, AMARI, GABRIELE, CAPALDI, CARMELIDA
Year of Publication 30.11.2021
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Year of Publication 30.11.2021
Patent
IMIDAZOLONE COMPOUNDS AS HUMAN NEUTROPHIL ELASTASE INHIBITORS
CARMELIDA CAPALDI, ANDREW STEPHEN ROBERT JENNINGS, ALISABETTA ARMANI, ROBERT ANDREW HEALD, JONATHAN MARK SUTTON
Year of Publication 11.01.2023
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Year of Publication 11.01.2023
Patent