Ribose-Modified Nucleosides as Ligands for Adenosine Receptors: Synthesis, Conformational Analysis, and Biological Evaluation of 1‘-C-Methyl Adenosine Analogues
Cappellacci, Loredana, Barboni, Grazia, Palmieri, Micaela, Pasqualini, Michela, Grifantini, Mario, Costa, Barbara, Martini, Claudia, Franchetti, Palmarisa
Published in Journal of medicinal chemistry (14.03.2002)
Published in Journal of medicinal chemistry (14.03.2002)
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Synthesis and potency of novel uracil nucleotides and derivatives as P2Y 2 and P2Y 6 receptor agonists
Ko, Hyojin, Carter, Rhonda L., Cosyn, Liesbet, Petrelli, Riccardo, de Castro, Sonia, Besada, Pedro, Zhou, Yixing, Cappellacci, Loredana, Franchetti, Palmarisa, Grifantini, Mario, Van Calenbergh, Serge, Harden, T. Kendall, Jacobson, Kenneth A.
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
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Exploring the Role of N 6‑Substituents in Potent Dual Acting 5′‑C‑Ethyltetrazolyladenosine Derivatives: Synthesis, Binding, Functional Assays, and Antinociceptive Effects in Mice
Petrelli, Riccardo, Scortichini, Mirko, Kachler, Sonja, Boccella, Serena, Cerchia, Carmen, Torquati, Ilaria, Del Bello, Fabio, Salvemini, Daniela, Novellino, Ettore, Luongo, Livio, Maione, Sabatino, Jacobson, Kenneth A, Lavecchia, Antonio, Klotz, Karl-Norbert, Cappellacci, Loredana
Published in Journal of medicinal chemistry (25.05.2017)
Published in Journal of medicinal chemistry (25.05.2017)
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The synergistic apoptotic effects of thiophenfurin, an inosine monophosphate dehydrogenase inhibitor, in combination with retinoids in HL60 cells
MELI, Maria, TOLOMEO, Manlio, GRIFANTINI, Mario, FRANCHETTI, Palmarisa, CAPPELLACCI, Loredana, SIMONI, Daniele, INVIDIATA, Francesco P, AIELLO, Stefania, DUSONCHET, Luisa
Published in Oncology reports (2007)
Published in Oncology reports (2007)
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Erythrocyte-mediated delivery of a new homodinucleotide active against human immunodeficiency virus and herpes simplex virus
Rossi, Luigia, Serafini, Sonja, Cappellacci, Loredana, Balestra, Emanuela, Brandi, Giorgio, Schiavano, Giuditta F., Franchetti, Palmarisa, Grifantini, Mario, Perno, Carlo-Federico, Magnani, Mauro
Published in Journal of antimicrobial chemotherapy (01.06.2001)
Published in Journal of antimicrobial chemotherapy (01.06.2001)
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Furanfurin and Thiophenfurin: Two Novel Tiazofurin Analogs. Synthesis, Structure, Antitumor Activity, and Interactions with Inosine Monophosphate Dehydrogenase
Franchetti, Palmarisa, Cappellacci, Loredana, Grifantini, Mario, Barzi, Anna, Nocentini, Giuseppe, Yang, Hongyoan, O'Connor, Ayrn, Jayaram, Hiremagalur N, Carrell, Christopher, Goldstein, Barry M
Published in Journal of medicinal chemistry (01.09.1995)
Published in Journal of medicinal chemistry (01.09.1995)
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2‘-C-Methyl Analogues of Selective Adenosine Receptor Agonists: Synthesis and Binding Studies
Franchetti, Palmarisa, Cappellacci, Loredana, Marchetti, Stefano, Trincavelli, Letizia, Martini, Claudia, Mazzoni, Maria R, Lucacchini, Antonio, Grifantini, Mario
Published in Journal of medicinal chemistry (07.05.1998)
Published in Journal of medicinal chemistry (07.05.1998)
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5′‑C‑Ethyl-tetrazolyl‑N 6‑Substituted Adenosine and 2‑Chloro-adenosine Derivatives as Highly Potent Dual Acting A1 Adenosine Receptor Agonists and A3 Adenosine Receptor Antagonists
Petrelli, Riccardo, Torquati, Ilaria, Kachler, Sonja, Luongo, Livio, Maione, Sabatino, Franchetti, Palmarisa, Grifantini, Mario, Novellino, Ettore, Lavecchia, Antonio, Klotz, Karl-Norbert, Cappellacci, Loredana
Published in Journal of medicinal chemistry (12.03.2015)
Published in Journal of medicinal chemistry (12.03.2015)
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A new C-nucleoside analogue of tiazofurin : synthesis and biological evaluation of 2-β- d-ribofuranosylimidazole-4-carboxamide (imidazofurin)
Franchetti, Palmarisa, Marchetti, Stefano, Cappellacci, Loredana, Yalowitz, Joel A, Jayaram, Hiremagalur N, Goldstein, Barry M, Grifantini, Mario
Published in Bioorganic & medicinal chemistry letters (08.01.2001)
Published in Bioorganic & medicinal chemistry letters (08.01.2001)
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Purine and pyrimidine nucleoside analogs of 3 '-C-methyladenosine as antitumor agents
Cappellacci, Loredana, Franchetti, Palmarisa, Petrelli, Riccardo, Riccioni, Sara, Vita, Patrizia, Jayaram, Hiremagalur N., Grifantini, Mario
Published in Collection of Czechoslovak chemical communications (01.07.2006)
Published in Collection of Czechoslovak chemical communications (01.07.2006)
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Synthesis, Conformational Analysis, and Biological Activity of C-Thioribonucleosides Related to Tiazofurin
Franchetti, Palmarisa, Marchetti, Stefano, Cappellacci, Loredana, Jayaram, Hiremagalur N, Yalowitz, Joel Aaron, Goldstein, Barry M, Barascut, Jean-Louis, Dukhan, David, Imbach, Jean-Louis, Grifantini, Mario
Published in Journal of medicinal chemistry (06.04.2000)
Published in Journal of medicinal chemistry (06.04.2000)
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Decomposition Pathways and in Vitro HIV Inhibitory Effects of IsoddA Pronucleotides: Toward a Rational Approach for Intracellular Delivery of Nucleoside 5‘-Monophosphates
Valette, Gilles, Pompon, Alain, Girardet, Jean-Luc, Cappellacci, Loredana, Franchetti, Palmarisa, Grifantini, Mario, La Colla, Paolo, Loi, Anna Giulia, Périgaud, Christian, Gosselin, Gilles, Imbach, Jean-Louis
Published in Journal of medicinal chemistry (10.05.1996)
Published in Journal of medicinal chemistry (10.05.1996)
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Synthesis, Structure, and Antiproliferative Activity of Selenophenfurin, an Inosine 5‘-Monophosphate Dehydrogenase Inhibitor Analogue of Selenazofurin
Franchetti, Palmarisa, Cappellacci, Loredana, Sheikha, Ghassan Abu, Jayaram, Hiremagalur N, Gurudutt, Vivek V, Sint, Thaw, Schneider, Bryan P, Jones, William D, Goldstein, Barry M, Perra, Graziella, De Montis, Antonella, Loi, Anna Giulia, La Colla, Paolo, Grifantini, Mario
Published in Journal of medicinal chemistry (23.05.1997)
Published in Journal of medicinal chemistry (23.05.1997)
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Isosteric Analogues of Nicotinamide Adenine Dinucleotide Derived from Furanfurin, Thiophenfurin, and Selenophenfurin as Mammalian Inosine Monophosphate Dehydrogenase (Type I and II) Inhibitors
Franchetti, Palmarisa, Cappellacci, Loredana, Perlini, Paolo, Jayaram, Hiremagalur N, Butler, Adrian, Schneider, Bryan P, Collart, Frank R, Huberman, Eliezer, Grifantini, Mario
Published in Journal of medicinal chemistry (07.05.1998)
Published in Journal of medicinal chemistry (07.05.1998)
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Journal Article
Ribose-modified Mizoribine Analogues: Synthesis and Biological Evaluation
Franchetti, Palmarisa, Pasqualini, Michela, Cappellacci, Loredana, Petrelli, Riccardo, Vita, Patrizia, Grifantini, Mario, Jayaram, Hiremagalur N.
Published in Nucleosides, nucleotides & nucleic acids (01.09.2005)
Published in Nucleosides, nucleotides & nucleic acids (01.09.2005)
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Journal Article
C-nucleoside analogues of furanfurin as ligands to A1 adenosine receptors
FRANCHETTI, Palmarisa, CAPPELLACCI, Loredana, MARCHETTI, Stefano, MARTINI, Claudia, COSTA, Barbara, VARANI, Katia, BOREA, Pier Andrea, GRIFANTINI, Mario
Published in Bioorganic & medicinal chemistry (01.09.2000)
Published in Bioorganic & medicinal chemistry (01.09.2000)
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Pharmacokinetic and antiretroviral activity in mice of oral [P1,P2-bis[2-(adenin-9-yl)ethoxymethyl]phosphonate], a prodrug of 9-(2-phosphonylmethoxyethyl)adenine
Rossi, Luigia, Dominici, Sabrina, Serafini, Sonja, Casabianca, Anna, Cerasi, Aurora, Chiarantini, Laura, Celeste, Angela Gabriela, Cappellacci, Loredana, Franchetti, Palmarisa, Grifantini, Mario, Magnani, Mauro
Published in Journal of antimicrobial chemotherapy (01.09.2002)
Published in Journal of antimicrobial chemotherapy (01.09.2002)
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Journal Article
A new acyclic heterodinucleotide active against Human Immunodeficiency Virus and Herpes Simplex Virus
Franchetti, Palmarisa, Abu Sheikha, Ghassan, Cappellacci, Loredana, Marchetti, Stefano, Grifantini, Mario, Balestra, Emanuela, Perno, Carlo-Federico, Benatti, Umberto, Brandi, Giorgio, Rossi, Luigia, Magnani, Mauro
Published in Antiviral research (01.09.2000)
Published in Antiviral research (01.09.2000)
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Journal Article
c-nucleoside analogues of furanfurin as ligands to a 1 adenosine receptors
Franchetti, Palmarisa, Cappellacci, Loredana, Marchetti, Stefano, Martini, Claudia, Costa, Barbara, Varani, Katia, Borea, Pier Andrea, Grifantini, Mario
Published in Bioorganic & medicinal chemistry (2000)
Published in Bioorganic & medicinal chemistry (2000)
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