Trifluoromethyl group as a pharmacophore : Effect of replacing a CF3 group on binding and agonist activity of a glucocorticoid receptor ligand
BETAGERI, Raj, YAN ZHANG, PAW, Zofia, SHIH, Daw-Tsun, SHIH, Cheng-Kon, ZUVELA-JELASKA, Ljiljana, NABOZNY, Gerald, THOMSON, David S, ZINDELL, Renee M, KUZMICH, Daniel, KIRRANE, Thomas M, BENTZIEN, Jörg, CARDOZO, Mario, CAPOLINO, Alison J, FADRA, Tazmeen N, NELSON, Richard M
Published in Bioorganic & medicinal chemistry letters (01.11.2005)
Published in Bioorganic & medicinal chemistry letters (01.11.2005)
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Journal Article
Discovery and SAR study of novel dihydroquinoline-containing glucocorticoid receptor agonists
Takahashi, Hidenori, Bekkali, Younes, Capolino, Alison J., Gilmore, Thomas, Goldrick, Susan E., Kaplita, Paul V., Liu, Lisa, Nelson, Richard M., Terenzio, Donna, Wang, Ji, Zuvela-Jelaska, Ljiljana, Proudfoot, John, Nabozny, Gerald, Thomson, David
Published in Bioorganic & medicinal chemistry letters (15.09.2007)
Published in Bioorganic & medicinal chemistry letters (15.09.2007)
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Journal Article
Discovery and SAR study of novel dihydroquinoline containing glucocorticoid receptor ligands
Takahashi, Hidenori, Bekkali, Younes, Capolino, Alison J., Gilmore, Thomas, Goldrick, Susan E., Nelson, Richard M., Terenzio, Donna, Wang, Ji, Zuvela-Jelaska, Ljiljana, Proudfoot, John, Nabozny, Gerald, Thomson, David
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
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Journal Article
Trifluoromethyl group as a pharmacophore: Effect of replacing a CF 3 group on binding and agonist activity of a glucocorticoid receptor ligand
Betageri, Raj, Zhang, Yan, Zindell, Renee M., Kuzmich, Daniel, Kirrane, Thomas M., Bentzien, Jörg, Cardozo, Mario, Capolino, Alison J., Fadra, Tazmeen N., Nelson, Richard M., Paw, Zofia, Shih, Daw-Tsun, Shih, Cheng-Kon, Zuvela-Jelaska, Ljiljana, Nabozny, Gerald, Thomson, David S.
Published in Bioorganic & medicinal chemistry letters (01.11.2005)
Published in Bioorganic & medicinal chemistry letters (01.11.2005)
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Journal Article