Search Results - "CANTRELL, BE" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Identification of (3R)-7-Hydroxy-N-((1S)-1-{[(3R,4R)-4-(3-hydroxyphenyl)- 3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl)-1,2,3,4-tetrahydro- 3-isoquinolinecarboxamide as a Novel Potent and Selective Opioid κ Receptor Antagonist

Identification of (3R)-7-Hydroxy-N-((1S)-1-{[(3R,4R)-4-(3-hydroxyphenyl)- 3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl)-1,2,3,4-tetrahydro- 3-isoquinolinecarboxamide as a Novel Potent and Selective Opioid κ Receptor Antagonist

by Thomas, James B, Atkinson, Robert N, Vinson, N. Ariane, Catanzaro, Jennifer L, Perretta, Carin L, Fix, Scott E, Mascarella, S. Wayne, Rothman, Richard B, Xu, Heng, Dersch, Christina M, Cantrell, Buddy E, Zimmerman, Dennis M, Carroll, F. Ivy
Published in Journal of medicinal chemistry (03.07.2003)

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Identification of the First trans-(3R,4R)- Dimethyl-4-(3-hydroxyphenyl)piperidine Derivative To Possess Highly Potent and Selective Opioid κ Receptor Antagonist Activity

Identification of the First trans-(3R,4R)- Dimethyl-4-(3-hydroxyphenyl)piperidine Derivative To Possess Highly Potent and Selective Opioid κ Receptor Antagonist Activity

by Thomas, James B, Atkinson, Robert N, Rothman, Richard B, Fix, Scott E, Mascarella, S. Wayne, Vinson, N. Ariane, Xu, Heng, Dersch, Christina M, Lu, Y. -F, Cantrell, Buddy E, Zimmerman, Dennis M, Carroll, F. Ivy
Published in Journal of medicinal chemistry (16.08.2001)

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Synthesis and Evaluation of a Series of Novel 2-[(4-Chlorophenoxy)methyl]- benzimidazoles as Selective Neuropeptide Y Y1 Receptor Antagonists

Synthesis and Evaluation of a Series of Novel 2-[(4-Chlorophenoxy)methyl]- benzimidazoles as Selective Neuropeptide Y Y1 Receptor Antagonists

by Zarrinmayeh, Hamideh, Nunes, Anne M, Ornstein, Paul L, Zimmerman, Dennis M, Arnold, M. Brian, Schober, Douglas A, Gackenheimer, Susan L, Bruns, Robert F, Hipskind, Philip A, Britton, Thomas C, Cantrell, Buddy E, Gehlert, Donald R
Published in Journal of medicinal chemistry (16.07.1998)

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Structure-activity relationship of a series of diaminoalkyl substituted benzimidazole as neuropeptide Y Y1 receptor antagonists

Structure-activity relationship of a series of diaminoalkyl substituted benzimidazole as neuropeptide Y Y1 receptor antagonists

by Zarrinmayeh, Hamideh, Zimmerman, Dennis M., Cantrell, Buddy E., Schober, Douglas A., Bruns, Robert E., Gackenheimer, Susan L., Ornstein, Paul L., Hipskind, Philip A., Britton, Thomas C., Gehlert, Donald R.
Published in Bioorganic & medicinal chemistry letters (08.03.1999)

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Importance of Phenolic Address Groups in Opioid Kappa Receptor Selective Antagonists

Importance of Phenolic Address Groups in Opioid Kappa Receptor Selective Antagonists

by Thomas, James B, Fix, Scott E, Rothman, Richard B, Mascarella, S. Wayne, Dersch, Christina M, Cantrell, Buddy E, Zimmerman, Dennis M, Carroll, F. Ivy
Published in Journal of medicinal chemistry (12.02.2004)

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Design and Synthesis of a Novel Series of 1,2-Disubstituted Cyclopentanes as Small, Potent Potentiators of 2-Amino-3-(3-hydroxy-5-methyl-isoxazol-4-yl)propanoic Acid (AMPA) Receptors

Design and Synthesis of a Novel Series of 1,2-Disubstituted Cyclopentanes as Small, Potent Potentiators of 2-Amino-3-(3-hydroxy-5-methyl-isoxazol-4-yl)propanoic Acid (AMPA) Receptors

by Shepherd, Timothy A, Aikins, James A, Bleakman, David, Cantrell, Buddy E, Rearick, John P, Simon, Richard L, Smith, Edward C. R, Stephenson, Gregory A, Zimmerman, Dennis M, Mandelzys, Allan, Jarvie, Keith R, Ho, Ken, Deverill, Michelle, Kamboj, Rajender K
Published in Journal of medicinal chemistry (09.05.2002)

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Discovery of the First N-Substituted 4β-Methyl-5-(3-hydroxyphenyl)morphan To Possess Highly Potent and Selective Opioid δ Receptor Antagonist Activity

Discovery of the First N-Substituted 4β-Methyl-5-(3-hydroxyphenyl)morphan To Possess Highly Potent and Selective Opioid δ Receptor Antagonist Activity

by Carroll, F. Ivy, Zhang, Li, Mascarella, S. Wayne, Navarro, Hernán A, Rothman, Richard B, Cantrell, Buddy E, Zimmerman, Dennis M, Thomas, James B
Published in Journal of medicinal chemistry (15.01.2004)

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Discovery of a Potent, Peripherally Selective trans-3,4-Dimethyl-4-(3-hydroxyphenyl)piperidine Opioid Antagonist for the Treatment of Gastrointestinal Motility Disorders

Discovery of a Potent, Peripherally Selective trans-3,4-Dimethyl-4-(3-hydroxyphenyl)piperidine Opioid Antagonist for the Treatment of Gastrointestinal Motility Disorders

by Zimmerman, Dennis M, Gidda, Jaswant S, Cantrell, Buddy E, Schoepp, Darryle D, Johnson, Bryan G, Leander, J. David
Published in Journal of medicinal chemistry (01.07.1994)

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Discovery of an Opioid κ Receptor Selective Pure Antagonist from a Library of N-Substituted 4β-Methyl-5-(3-hydroxyphenyl)morphans

Discovery of an Opioid κ Receptor Selective Pure Antagonist from a Library of N-Substituted 4β-Methyl-5-(3-hydroxyphenyl)morphans

by Thomas, James B, Atkinson, Robert N, Namdev, Nivedita, Rothman, Richard B, Gigstad, Kenneth M, Fix, Scott E, Mascarella, S. Wayne, Burgess, Jason P, Vinson, N. Ariane, Xu, Heng, Dersch, Christina M, Cantrell, Buddy E, Zimmerman, Dennis M, Carroll, F. Ivy
Published in Journal of medicinal chemistry (01.08.2002)

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Identification of an Opioid κ Receptor Subtype-Selective N-Substituent for (+)-(3R,4R)-Dimethyl-4-(3-hydroxyphenyl)piperidine

Identification of an Opioid κ Receptor Subtype-Selective N-Substituent for (+)-(3R,4R)-Dimethyl-4-(3-hydroxyphenyl)piperidine

by Thomas, James B, Fall, Michael J, Cooper, Julie B, Rothman, Richard B, Mascarella, S. Wayne, Xu, Heng, Partilla, John S, Dersch, Christina M, McCullough, Karen B, Cantrell, Buddy E, Zimmerman, Dennis M, Carroll, F. Ivy
Published in Journal of medicinal chemistry (17.12.1998)

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Investigation of the N-Substituent Conformation Governing Potency and μ Receptor Subtype-Selectivity in (+)-(3R,4R)-Dimethyl-4-(3-hydroxyphenyl)- piperidine Opioid Antagonists

Investigation of the N-Substituent Conformation Governing Potency and μ Receptor Subtype-Selectivity in (+)-(3R,4R)-Dimethyl-4-(3-hydroxyphenyl)- piperidine Opioid Antagonists

by Thomas, James B, Mascarella, S. Wayne, Rothman, Richard B, Partilla, John S, Xu, Heng, McCullough, Karen B, Dersch, Christina M, Cantrell, Buddy E, Zimmerman, Dennis M, Carroll, F. Ivy
Published in Journal of medicinal chemistry (21.05.1998)

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STRUCTURE-ACTIVITY-RELATIONSHIPS OF TRANS-3,4-DIMETHYL-4-(3-HYDROXYPHENYL)PIPERIDINE ANTAGONISTS FOR MU-OPIOID AND KAPPA-OPIOID RECEPTORS

STRUCTURE-ACTIVITY-RELATIONSHIPS OF TRANS-3,4-DIMETHYL-4-(3-HYDROXYPHENYL)PIPERIDINE ANTAGONISTS FOR MU-OPIOID AND KAPPA-OPIOID RECEPTORS

by ZIMMERMAN, DM, LEANDER, JD, CANTRELL, BE, REEL, JK, SNODDY, J, MENDELSOHN, LG, JOHNSON, BG, MITCH, CH
Published in Journal of medicinal chemistry (01.10.1993)

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N-Substituted 9β-Methyl-5-(3-hydroxyphenyl)morphans Are Opioid Receptor Pure Antagonists

N-Substituted 9β-Methyl-5-(3-hydroxyphenyl)morphans Are Opioid Receptor Pure Antagonists

by Thomas, James B, Zheng, Xiaoling, Mascarella, S. Wayne, Rothman, Richard B, Dersch, Christina M, Partilla, John S, Flippen-Anderson, Judith L, George, Clifford F, Cantrell, Buddy E, Zimmerman, Dennis M, Carroll, F. Ivy
Published in Journal of medicinal chemistry (08.10.1998)

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A stereoselective synthetic approach to N-alkyl-4β-methyl-5-phenylmorphans

A stereoselective synthetic approach to N-alkyl-4β-methyl-5-phenylmorphans

by Thomas, James B., Gigstad, Kenneth M., Fix, Scott E., Burgess, Jason P., Cooper, Julie B., Mascarella, S.Wayne, Cantrell, Buddy E., Zimmerman, Dennis M., Carroll, F.Ivy
Published in Tetrahedron letters (15.01.1999)

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Rapid parallel synthesis applied to the optimization of a series of potent nonpeptide neuropeptide Y-1 receptor antagonists

Rapid parallel synthesis applied to the optimization of a series of potent nonpeptide neuropeptide Y-1 receptor antagonists

by Siegel, Miles G., Chaney, Michael O., Bruns, Robert F., Clay, Michael P., Schober, Douglas A., Van Abbema, Anne M., Johnson, Douglas W., Cantrell, Buddy E., Hahn, Patric J., Hunden, David C., Gehlert, Donald R., Zarrinmayeh, Hamideh, Ornstein, Paul L., Zimmerman, Dennis M., Koppel, Gary A.
Published in Tetrahedron (24.09.1999)

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Synthesis of a Series of Aryl Kainic Acid Analogs and Evaluation in Cells Stably Expressing the Kainate Receptor humGluR6

Synthesis of a Series of Aryl Kainic Acid Analogs and Evaluation in Cells Stably Expressing the Kainate Receptor humGluR6

by Cantrell, Buddy E, Zimmerman, Dennis M, Monn, James A, Kamboj, Rajender K, Hoo, Ken H, Tizzano, Joseph P, Pullar, Ian A, Farrell, Louise N, Bleakman, David
Published in Journal of medicinal chemistry (13.09.1996)

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3,4-Dimethyl-4-(3-hydroxyphenyl)piperidines: opioid antagonists with potent anorectant activity

3,4-Dimethyl-4-(3-hydroxyphenyl)piperidines: opioid antagonists with potent anorectant activity

by Mitch, Charles H, Leander, J. David, Mendelsohn, Laurane G, Shaw, Walter N, Wong, David T, Cantrell, Buddy E, Johnson, Bryan G, Reel, John K, Snoddy, John D
Published in Journal of medicinal chemistry (01.10.1993)

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Structure-activity relationships of a series of 1-substituted-4-methylbenzimidazole neuropeptide Y-1 receptor antagonists

Structure-activity relationships of a series of 1-substituted-4-methylbenzimidazole neuropeptide Y-1 receptor antagonists

by Zimmerman, Dennis M., Cantrell, Buddy E., Smith, Edward C.R., Nixon, James A., Bruns, Robert F., Gitter, Bruce, Hipskind, Philip A., Ornstein, Paul L., Zarrinmayeh, Hamideh, Britton, Thomas C., Schober, Douglas A., Gehlert, Donald R.
Published in Bioorganic & medicinal chemistry letters (03.03.1998)

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Synthesis of 9β-methyl-2-alkyl-7-oxo-5-arylmorphans

Synthesis of 9β-methyl-2-alkyl-7-oxo-5-arylmorphans

by Thomas, James B., Zheng, Xiaoling, Brieaddy, Lawrence E., Burgess, Jason P., Wayne Mascarella, S., Fix, Scott E., Cantrell, Buddy E., Zimmerman, Dennis M., Ivy Carroll, F.
Published in Tetrahedron letters (24.09.1998)

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CHARACTERIZATION OF THE NEUROTOXIC POTENTIAL OF META-METHOXY-MPTP AND THE USE OF ITS N-ETHYL ANALOG AS A MEANS OF AVOIDING EXPOSURE TO A POSSIBLE PARKINSONISM-CAUSING AGENT

CHARACTERIZATION OF THE NEUROTOXIC POTENTIAL OF META-METHOXY-MPTP AND THE USE OF ITS N-ETHYL ANALOG AS A MEANS OF AVOIDING EXPOSURE TO A POSSIBLE PARKINSONISM-CAUSING AGENT

by ZIMMERMAN, DM, CANTRELL, BE, REEL, JK, HEMRICKLUECKE, SK, FULLER, RW
Published in Journal of medicinal chemistry (01.08.1986)

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