2,3,8-Trisubstituted Quinolines with Antimalarial Activity
Martinez, Pablo D G, Krake, Susann H, Poggi, Maitia L, Campbell, Simon F, Willis, Paul A, Dias, Luiz C
Published in Anais da Academia Brasileira de Ciências (01.01.2018)
Published in Anais da Academia Brasileira de Ciências (01.01.2018)
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Discovery of a Quinoline-4-carboxamide Derivative with a Novel Mechanism of Action, Multistage Antimalarial Activity, and Potent in Vivo Efficacy
Baragaña, Beatriz, Norcross, Neil R, Wilson, Caroline, Porzelle, Achim, Hallyburton, Irene, Grimaldi, Raffaella, Osuna-Cabello, Maria, Norval, Suzanne, Riley, Jennifer, Stojanovski, Laste, Simeons, Frederick R. C, Wyatt, Paul G, Delves, Michael J, Meister, Stephan, Duffy, Sandra, Avery, Vicky M, Winzeler, Elizabeth A, Sinden, Robert E, Wittlin, Sergio, Frearson, Julie A, Gray, David W, Fairlamb, Alan H, Waterson, David, Campbell, Simon F, Willis, Paul, Read, Kevin D, Gilbert, Ian H
Published in Journal of medicinal chemistry (10.11.2016)
Published in Journal of medicinal chemistry (10.11.2016)
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Identification of potent and reversible piperidine carboxamides that are species-selective orally active proteasome inhibitors to treat malaria
Lawong, Aloysus, Gahalawat, Suraksha, Ray, Sneha, Ho, Nhi, Han, Yan, Ward, Kurt E., Deng, Xiaoyi, Chen, Zhe, Kumar, Ashwani, Xing, Chao, Hosangadi, Varun, Fairhurst, Kate J., Tashiro, Kyuto, Liszczak, Glen, Shackleford, David M., Katneni, Kasiram, Chen, Gong, Saunders, Jessica, Crighton, Elly, Casas, Arturo, Robinson, Joshua J., Imlay, Leah S., Zhang, Xiaoyu, Lemoff, Andrew, Zhao, Zhiyu, Angulo-Barturen, Iñigo, Jiménez-Díaz, María Belén, Wittlin, Sergio, Campbell, Simon F., Fidock, David A., Laleu, Benoît, Charman, Susan A., Ready, Joseph M., Phillips, Margaret A.
Published in Cell chemical biology (15.08.2024)
Published in Cell chemical biology (15.08.2024)
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Trisubstituted Pyrimidines as Efficacious and Fast-Acting Antimalarials
Norcross, Neil R, Baragaña, Beatriz, Wilson, Caroline, Hallyburton, Irene, Osuna-Cabello, Maria, Norval, Suzanne, Riley, Jennifer, Stojanovski, Laste, Simeons, Frederick R. C, Porzelle, Achim, Grimaldi, Raffaella, Wittlin, Sergio, Duffy, Sandra, Avery, Vicky M, Meister, Stephan, Sanz, Laura, Jiménez-Díaz, Belén, Angulo-Barturen, Iñigo, Ferrer, Santiago, Martínez, María Santos, Gamo, Francisco Javier, Frearson, Julie A, Gray, David W, Fairlamb, Alan H, Winzeler, Elizabeth A, Waterson, David, Campbell, Simon F, Willis, Paul, Read, Kevin D, Gilbert, Ian H
Published in Journal of medicinal chemistry (14.07.2016)
Published in Journal of medicinal chemistry (14.07.2016)
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Substituted Aminoacetamides as Novel Leads for Malaria Treatment
Norcross, Neil R., Wilson, Caroline, Baragaña, Beatriz, Hallyburton, Irene, Osuna‐Cabello, Maria, Norval, Suzanne, Riley, Jennifer, Fletcher, Daniel, Sinden, Robert, Delves, Michael, Ruecker, Andrea, Duffy, Sandra, Meister, Stephan, Antonova‐Koch, Yevgeniya, Crespo, Benigno, de Cózar, Cristina, Sanz, Laura M., Gamo, Francisco Javier, Avery, Vicky M., Frearson, Julie A., Gray, David W., Fairlamb, Alan H., Winzeler, Elizabeth A., Waterson, David, Campbell, Simon F., Willis, Paul A., Read, Kevin D., Gilbert, Ian H.
Published in ChemMedChem (17.07.2019)
Published in ChemMedChem (17.07.2019)
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A highly stereoselective synthesis of the racemic juvenile hormone
Johnson, William S, Li, Tsung-tee, Faulkner, D. John, Campbell, Simon F
Published in Journal of the American Chemical Society (01.10.1968)
Published in Journal of the American Chemical Society (01.10.1968)
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Journal Article
Long-acting dihydropyridine calcium antagonists. 4. Synthesis and structure-activity relationships for a series of basic and nonbasic derivatives of 2[(2-aminoethoxy)methyl]-1,4-dihydropyridine calcium antagonists
Alker, David, Campbell, Simon F, Cross, Peter E, Burges, Roger A, Carter, Anthony J, Gardiner, Donald G
Published in Journal of medicinal chemistry (01.02.1990)
Published in Journal of medicinal chemistry (01.02.1990)
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Long-acting dihydropyridine calcium antagonists. 6. Structure-activity relationships around 4-(2,3-dichlorophenyl)-3-(ethoxycarbonyl)-2-[(2-hydroxyethoxy)methyl]-5-(methoxycarbonyl)-6-methyl-1,4-dihydropyridine
Alker, David, Campbell, Simon F, Cross, Peter E
Published in Journal of medicinal chemistry (01.01.1991)
Published in Journal of medicinal chemistry (01.01.1991)
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2,4-Diamino-6,7-dimethoxyquinazolines. 1. 2-[4-(1,4-Benzodioxan-2-ylcarbonyl)piperazin-1-yl] derivatives as .alpha.1-adrenoceptor antagonists and antihypertensive agents
Campbell, Simon F, Davey, Michael J, Hardstone, J. David, Lewis, Brian N, Palmer, Michael J
Published in Journal of medicinal chemistry (01.01.1987)
Published in Journal of medicinal chemistry (01.01.1987)
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Journal Article
2(1H)-Quinolinones with cardiac stimulant activity. 2. Synthesis and biological activities of 6-(N-linked, five-membered heteroaryl) derivatives
Alabaster, Colin T, Bell, Andrew S, Campbell, Simon F, Ellis, Peter, Henderson, Christopher G, Morris, David S, Roberts, David A, Ruddock, Keith S, Samuels, Gillian M. R, Stefaniak, Mark H
Published in Journal of medicinal chemistry (01.03.1989)
Published in Journal of medicinal chemistry (01.03.1989)
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Journal Article
Long-acting dihydropyridine calcium antagonists. 1. 2-Alkoxymethyl derivatives incorporating basic substituents
Arrowsmith, John E, Campbell, Simon F, Cross, Peter E, Stubbs, John K, Burges, Roger A, Gardiner, Donald G, Blackburn, Kenneth J
Published in Journal of medicinal chemistry (01.09.1986)
Published in Journal of medicinal chemistry (01.09.1986)
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Journal Article
2(1H)-Quinolinones with cardiac stimulant activity. 1. Synthesis and biological activities of (six-membered heteroaryl)-substituted derivatives
Alabaster, Colin T, Bell, Andrew S, Campbell, Simon F, Ellis, Peter, Henderson, Christopher G, Roberts, David A, Ruddock, Keith S, Samuels, Gillian M. R, Stefaniak, Mark H
Published in Journal of medicinal chemistry (01.10.1988)
Published in Journal of medicinal chemistry (01.10.1988)
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