Connexin 30 is expressed in the mouse sino-atrial node and modulates heart rate
Gros, Daniel, Théveniau-Ruissy, Magali, Bernard, Monique, Calmels, Thierry, Kober, Frank, Söhl, Goran, Willecke, Klaus, Nargeot, Joël, Jongsma, Habo J., Mangoni, Matteo E.
Published in Cardiovascular research (01.01.2010)
Published in Cardiovascular research (01.01.2010)
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Refined Docking as a Valuable Tool for Lead Optimization: Application to Histamine H3 Receptor Antagonists
Levoin, Nicolas, Calmels, Thierry, Poupardin-Olivier, Olivia, Labeeuw, Olivier, Danvy, Denis, Robert, Philippe, Berrebi-Bertrand, Isabelle, Ganellin, C. Robin, Schunack, Walter, Stark, Holger, Capet, Marc
Published in Archiv der Pharmazie (Weinheim) (01.10.2008)
Published in Archiv der Pharmazie (Weinheim) (01.10.2008)
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Human p63RhoGEF, a novel RhoA-specific guanine nucleotide exchange factor, is localized in cardiac sarcomere
Souchet, Michel, Portales-Casamar, Elodie, Mazurais, David, Schmidt, Susanne, Léger, Isabelle, Javré, Jean-Luc, Robert, Philippe, Berrebi-Bertrand, Isabelle, Bril, Antoine, Gout, Bernard, Debant, Anne, Calmels, Thierry P G
Published in Journal of cell science (01.02.2002)
Published in Journal of cell science (01.02.2002)
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Hybrid approach for the design of highly affine and selective dopamine D3 receptor ligands using privileged scaffolds of biogenic amine GPCR ligands
SASSE, Britta C, MACH, Ulrich R, LEPPAENEN, Jukka, CALMELS, Thierry, STARK, Holger
Published in Bioorganic & medicinal chemistry (01.12.2007)
Published in Bioorganic & medicinal chemistry (01.12.2007)
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Genomic organization and alternative transcripts of the human Connexin40 gene
Dupays, Laurent, Mazurais, David, Rücker-Martin, Catherine, Calmels, Thierry, Bernot, Denis, Cronier, Laurent, Malassiné, André, Gros, Daniel, Théveniau-Ruissy, Magali
Published in Gene (13.02.2003)
Published in Gene (13.02.2003)
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uDENN, DENN, and dDENN: Indissociable Domains in Rab and MAP Kinases Signaling Pathways
Levivier, Emilie, Goud, Bruno, Souchet, Michel, Calmels, Thierry P.G., Mornon, Jean-Paul, Callebaut, Isabelle
Published in Biochemical and biophysical research communications (28.09.2001)
Published in Biochemical and biophysical research communications (28.09.2001)
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Constitutive expression of the DNA-binding domain of Ets1 increases endothelial cell adhesion and stimulates their organization into capillary-like structures
MATTOT, V, VERCAMER, C, SONCIN, F, CALMELS, T, HUGUET, C, FAFEUR, V, VANDENBUNDER, B
Published in Oncogene (10.02.2000)
Published in Oncogene (10.02.2000)
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Dual Piperidine-Based Histamine H-3 and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain
Szczepanska, Katarzyna, Karcz, Tadeusz, Dichiara, Maria, Mogilski, Szczepan, Kalinowska-Tluscik, Justyna, Pilarski, Boguslaw, Leniak, Arkadiusz, Pietrus, Wojciech, Podlewska, Sabina, Popiolek-Barczyk, Katarzyna, Humphrys, Laura J., Ruiz-Cantero, M. Carmen, Reiner-Link, David, Leitzbach, Luisa, Lazewska, Dorota, Pockes, Steffen, Gorka, Michal, Zmyslowski, Adam, Calmels, Thierry, Cobos, Enrique J., Marrazzo, Agostino, Stark, Holger, Bojarski, Andrzej J., Amata, Emanuele, Kiec-Kononowicz, Katarzyna
Published in Journal of medicinal chemistry (27.07.2023)
Published in Journal of medicinal chemistry (27.07.2023)
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Journal Article
Dual Piperidine-Based Histamine H3 and Sigma‑1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain
Szczepańska, Katarzyna, Karcz, Tadeusz, Dichiara, Maria, Mogilski, Szczepan, Kalinowska-Tłuścik, Justyna, Pilarski, Bogusław, Leniak, Arkadiusz, Pietruś, Wojciech, Podlewska, Sabina, Popiołek-Barczyk, Katarzyna, Humphrys, Laura J., Ruiz-Cantero, M. Carmen, Reiner-Link, David, Leitzbach, Luisa, Łażewska, Dorota, Pockes, Steffen, Górka, Michał, Zmysłowski, Adam, Calmels, Thierry, Cobos, Enrique J., Marrazzo, Agostino, Stark, Holger, Bojarski, Andrzej J., Amata, Emanuele, Kieć-Kononowicz, Katarzyna
Published in Journal of medicinal chemistry (27.07.2023)
Published in Journal of medicinal chemistry (27.07.2023)
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Synthesis and evaluation of a 2-benzothiazolylphenylmethyl ether class of histamine H4 receptor antagonists
Labeeuw, Olivier, Levoin, Nicolas, Billot, Xavier, Danvy, Denis, Calmels, Thierry, Krief, Stéphane, Ligneau, Xavier, Berrebi-Bertrand, Isabelle, Robert, Philippe, Lecomte, Jeanne-Marie, Schwartz, Jean-Charles, Capet, Marc
Published in Bioorganic & medicinal chemistry letters (01.11.2016)
Published in Bioorganic & medicinal chemistry letters (01.11.2016)
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Journal Article
Discovery of nanomolar ligands with novel scaffolds for the histamine H4 receptor by virtual screening
Levoin, Nicolas, Labeeuw, Olivier, Billot, Xavier, Calmels, Thierry, Danvy, Denis, Krief, Stéphane, Berrebi-Bertrand, Isabelle, Lecomte, Jeanne-Marie, Schwartz, Jean-Charles, Capet, Marc
Published in European journal of medicinal chemistry (05.01.2017)
Published in European journal of medicinal chemistry (05.01.2017)
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Journal Article
Improving selectivity of dopamine D3 receptor ligands
Capet, Marc, Calmels, Thierry, Levoin, Nicolas, Danvy, Denis, Berrebi-Bertrand, Isabelle, Stark, Holger, Schwartz, Jean-Charles, Lecomte, Jeanne-Marie
Published in Bioorganic & medicinal chemistry letters (01.02.2016)
Published in Bioorganic & medicinal chemistry letters (01.02.2016)
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Journal Article
Novel and highly potent histamine H3 receptor ligands. Part 1: withdrawing of hERG activity
Levoin, Nicolas, Labeeuw, Olivier, Calmels, Thierry, Poupardin-Olivier, Olivia, Berrebi-Bertrand, Isabelle, Lecomte, Jeanne-Marie, Schwartz, Jean-Charles, Capet, Marc
Published in Bioorganic & medicinal chemistry letters (15.09.2011)
Published in Bioorganic & medicinal chemistry letters (15.09.2011)
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Journal Article
Determination of the binding mode and interacting amino-acids for dibasic H3 receptor antagonists
Levoin, Nicolas, Labeeuw, Olivier, Krief, Stéphane, Calmels, Thierry, Poupardin-Olivier, Olivia, Berrebi-Bertrand, Isabelle, Lecomte, Jeanne-Marie, Schwartz, Jean-Charles, Capet, Marc
Published in Bioorganic & medicinal chemistry (01.08.2013)
Published in Bioorganic & medicinal chemistry (01.08.2013)
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Journal Article
Novel and highly potent histamine H-3 receptor ligands. Part 3: An alcohol function to improve the pharmacokinetic profile
Labeeuw, Olivier, Levoin, Nicolas, Poupardin-Olivier, Olivia, Calmels, Thierry, Ligneau, Xavier, Berrebi-Bertrand, Isabelle, Robert, Philippe, Lecomte, Jeanne-Marie, Schwartz, Jean-Charles, Capet, Marc
Published in Bioorganic & medicinal chemistry letters (01.05.2013)
Published in Bioorganic & medicinal chemistry letters (01.05.2013)
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Journal Article
Hybrid approach for the design of highly affine and selective dopamine D 3 receptor ligands using privileged scaffolds of biogenic amine GPCR ligands
Sasse, Britta C., Mach, Ulrich R., Leppaenen, Jukka, Calmels, Thierry, Stark, Holger
Published in Bioorganic & medicinal chemistry (01.12.2007)
Published in Bioorganic & medicinal chemistry (01.12.2007)
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