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Published in Angewandte Chemie (International ed.) (13.04.2015)
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Imidazopiperidine amides as dipeptidyl peptidase IV inhibitors for the treatment of diabetes
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Published in Bioorganic & medicinal chemistry letters (01.11.2007)
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Electrolytic Macrocyclizations: Scalable Synthesis of a Diazonamide-Based Drug Development Candidate
Ding, Hui, DeRoy, Patrick L., Perreault, Christian, Larivée, Alexandre, Siddiqui, Arshad, Caldwell, Charles G., Harran, Susan, Harran, Patrick G.
Published in Angewandte Chemie (13.04.2015)
Published in Angewandte Chemie (13.04.2015)
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Fluoropyrrolidine amides as dipeptidyl peptidase IV inhibitors
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Published in Bioorganic & medicinal chemistry letters (08.03.2004)
Published in Bioorganic & medicinal chemistry letters (08.03.2004)
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1,3,4-Trisubstituted pyrrolidine CCR5 receptor antagonists: modifications of the arylpropylpiperidine side chains
Lynch, Christopher L., Willoughby, Christopher A., Hale, Jeffrey J., Holson, Edward J., Budhu, Richard J., Gentry, Amy L., Rosauer, Keith G., Caldwell, Charles G., Chen, Ping, Mills, Sander G., MacCoss, Malcolm, Berk, Scott, Chen, Liya, Chapman, Kevin T., Malkowitz, Lorraine, Springer, Martin S., Gould, Sandra L., DeMartino, Julie A., Siciliano, Salvatore J., Cascieri, Margaret A., Carella, Anthony, Carver, Gwen, Holmes, Karen, Schleif, William A., Danzeisen, Renee, Hazuda, Daria, Kessler, Joseph, Lineberger, Janet, Miller, Michael, Emini, Emilio A.
Published in Bioorganic & medicinal chemistry letters (06.01.2003)
Published in Bioorganic & medicinal chemistry letters (06.01.2003)
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Synthesis of analogs of (1,4)-3- and 5-imino oxazepane, thiazepane, and diazepane as inhibitors of nitric oxide synthases
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Published in Bioorganic & medicinal chemistry letters (06.12.2004)
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Design, synthesis, and SAR of heterocycle-containing antagonists of the human CCR5 receptor for the treatment of HIV-1 infection
Kim, Dooseop, Wang, Liping, Caldwell, Charles G., Chen, Ping, Finke, Paul E., Oates, Bryan, MacCoss, Malcolm, Mills, Sander G., Malkowitz, Lorraine, Gould, Sandra L., DeMartino, Julie A., Springer, Martin S., Hazuda, Daria, Miller, Michael, Kessler, Joseph, Danzeisen, Renee, Carver, Gwen, Carella, Anthony, Holmes, Karen, Lineberger, Janet, Schleif, William A., Emini, Emilio A.
Published in Bioorganic & medicinal chemistry letters (17.12.2001)
Published in Bioorganic & medicinal chemistry letters (17.12.2001)
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2,3-Dihydro-5-benzofuranols as antioxidant-based inhibitors of leukotriene biosynthesis
Hammond, Milton L, Kopka, Ihor E, Zambias, Robert A, Caldwell, Charles G, Boger, Joshua, Baker, Florence, Bach, Tom, Luell, Silvi, MacIntyre, D. Euan
Published in Journal of medicinal chemistry (01.05.1989)
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Sulfur-substituted dienes and the silylene protecting group in synthesis. Deoxypillaromycinone
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Published in Journal of organic chemistry (01.09.1983)
Published in Journal of organic chemistry (01.09.1983)
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CCR5 Antagonists: 3-(Pyrrolidin-1-yl)propionic Acid Analogues with Potent Anti-HIV Activity
Lynch, Christopher L, Hale, Jeffrey J, Budhu, Richard J, Gentry, Amy L, Finke, Paul E, Caldwell, Charles G, Mills, Sander G, MacCoss, Malcolm, Shen, Dong-Ming, Chapman, Kevin T, Malkowitz, Lorraine, Springer, Martin S, Gould, Sandra L, DeMartino, Julie A, Siciliano, Salvatore J, Cascieri, Margaret A, Carella, Anthony, Carver, Gwen, Holmes, Karen, Schleif, William A, Danzeisen, Renee, Hazuda, Daria, Kessler, Joseph, Lineberger, Janet, Miller, Michael, Emini, Emilio
Published in Organic letters (10.07.2003)
Published in Organic letters (10.07.2003)
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Syntheses and biological evaluation of 5-(piperidin-1-yl)-3-phenyl-pentylsulfones as CCR5 antagonists
Shankaran, K., Donnelly, Karla L., Shah, Shrenik K., Caldwell, Charles G., Chen, Ping, Finke, Paul E., Oates, Bryan, MacCoss, Malcolm, Mills, Sander G., DeMartino, Julie A., Gould, Sandra L., Malkowitz, Lorraine, Siciliano, Salvatore J., Springer, Martin S., Kwei, Gloria, Carella, Anthony, Carver, Gwen, Danzeisen, Renee, Hazuda, Daria, Holmes, Karen, Kessler, Joseph, Lineberger, Janet, Miller, Michael D., Emini, Emilio A., Schleif, William A.
Published in Bioorganic & medicinal chemistry letters (05.07.2004)
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Inhibition of Stromelysin-1 (MMP-3) by P1‘-Biphenylylethyl Carboxyalkyl Dipeptides
Esser, Craig K, Bugianesi, Robert L, Caldwell, Charles G, Chapman, Kevin T, Durette, Philippe L, Girotra, Narindar N, Kopka, Ihor E, Lanza, Thomas J, Levorse, Dorothy A, MacCoss, Malcolm, Owens, Karen A, Ponpipom, Mitree M, Simeone, Joseph P, Harrison, Richard K, Niedzwiecki, Lisa, Becker, Joseph W, Marcy, Alice I, Axel, Melinda G, Christen, Amy J, McDonnell, Joseph, Moore, Vernon L, Olszewski, Julie M, Saphos, Cheryl, Visco, Denise M, Shen, Frank, Colletti, Adria, Krieter, Philip A, Hagmann, William K
Published in Journal of medicinal chemistry (14.03.1997)
Published in Journal of medicinal chemistry (14.03.1997)
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Caldwell, Charles G., Sahoo, Soumya P., Polo, Scott A., Eversole, Randall R., Lanza, Thomas J., Mills, Sander G., Niedzwiecki, Lisa M., Izquierdo-Martin, Maria, Chang, Benedict C., Harrison, Richard K., Kuo, David W., Lin, T.-Y., Stein, Ross L., Durette, Philippe L., Hagmann, William K.
Published in Bioorganic & medicinal chemistry letters (01.02.1996)
Published in Bioorganic & medicinal chemistry letters (01.02.1996)
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Photoisomerization Mechanism of the Rhodopsin Chromophore: Picosecond Photolysis of Pigment Containing 11-Cis-Locked Eight-Membered Ring Retinal
Mizukami, Taku, Kandori, Hideki, Shichida, Yoshinori, Chen, Arh-Hwang, Derguini, Fadila, Caldwell, Charles G., Bigge, Christopher F., Nakanishi, Koji, Yoshizawa, Toru
Published in Proceedings of the National Academy of Sciences - PNAS (01.05.1993)
Published in Proceedings of the National Academy of Sciences - PNAS (01.05.1993)
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Substituted 4,6-diaminoquinolines as inhibitors of C5a receptor binding
Lanza, Thomas J, Durette, Philippe L, Rollins, Thomas, Siciliano, Salvatore, Cianciarulo, Dana N, Kobayashi, Sumire V, Caldwell, Charles G, Springer, Martin S, Hagmann, William K
Published in Journal of medicinal chemistry (01.01.1992)
Published in Journal of medicinal chemistry (01.01.1992)
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