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ZHANG, Han-Zhong, CLAASSEN, Gisela, CROGRAN-GRUNDY, Candace, TSENG, Ben, DREWE, John, SUI XIONG CAI
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Published in Bioorganic & medicinal chemistry (2008)
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MX1013, a dipeptide caspase inhibitor with potent in vivo antiapoptotic activity
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Published in British journal of pharmacology (01.09.2003)
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The discovery and mechanism of action of novel tumor-selective and apoptosis-inducing 3,5-diaryl-1,2,4-oxadiazole series using a chemical genetics approach
Jessen, Katayoun A, English, Nicole M, Yu Wang, Jean, Maliartchouk, Sergei, Archer, Shannon P, Qiu, Ling, Brand, Regina, Kuemmerle, Jared, Zhang, Han-Zhong, Gehlsen, Kurt, Drewe, John, Tseng, Ben, Cai, Sui Xiong, Kasibhatla, Shailaja
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Published in Molecular cancer therapeutics (01.05.2005)
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Dipeptidyl aspartyl fluoromethylketones as potent caspase inhibitors : Peptidomimetic replacement of the P2 amino acid by 2-aminoaryl acids and other non-natural amino acids
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Published in Bioorganic & medicinal chemistry letters (15.11.2007)
Published in Bioorganic & medicinal chemistry letters (15.11.2007)
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Discovery of 5-(4-hydroxy-6-methyl-2-oxo-2 H-pyran-3-yl)-7-phenyl-( E)-2,3,6,7-tetrahydro-1,4-thiazepines as a new series of apoptosis inducers using a cell- and caspase-based HTS assay
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Published in Bioorganic & medicinal chemistry letters (01.09.2007)
Published in Bioorganic & medicinal chemistry letters (01.09.2007)
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V102862 (Co 102862): a potent, broad‐spectrum state‐dependent blocker of mammalian voltage‐gated sodium channels
Ilyin, Victor I, Hodges, Dianne D, Whittemore, Edward R, Carter, Richard B, Cai, Sui Xiong, Woodward, Richard M
Published in British journal of pharmacology (01.03.2005)
Published in British journal of pharmacology (01.03.2005)
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Design and synthesis of Rhodamine 110 derivative and Caspase-3 substrate for enzyme and cell-based fluorescent assay
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Published in Bioorganic & medicinal chemistry letters (08.01.2001)
Published in Bioorganic & medicinal chemistry letters (08.01.2001)
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Dipeptidyl aspartyl fluoromethylketones as potent caspase inhibitors: peptidomimetic replacement of the P2 α-amino acid by a α-hydroxy acid
YAN WANG, LUFENG GUAN, SHAOJUAN JIA, BEN TSENG, DREWE, John, SUI XIONG CAI
Published in Bioorganic & medicinal chemistry letters (01.03.2005)
Published in Bioorganic & medicinal chemistry letters (01.03.2005)
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Dipeptidyl aspartyl fluoromethylketones as potent caspase inhibitors: SAR of the N-protecting group
SUI XIONG CAI, LUFENG GUAN, SHAOJUAN JIA, YAN WANG, WU YANG, TSENG, Ben, DREWE, John
Published in Bioorganic & medicinal chemistry letters (01.11.2004)
Published in Bioorganic & medicinal chemistry letters (01.11.2004)
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Discovery and structure–activity relationship of 2-phenyl-oxazole-4-carboxamide derivatives as potent apoptosis inducers
Tai, Vincent W.-F., Sperandio, David, Shelton, Emma J., Litvak, Joane, Pararajasingham, Keith, Cebon, Ben, Lohman, Julia, Eksterowicz, John, Kantak, Seema, Sabbatini, Peter, Brown, Cindy, Zeitz, Jennifer, Reed, Chris, Maske, Bill, Graupe, Doris, Estevez, Alberto, Oeh, Jason, Wong, Darren, Ni, Yong, Sprengeler, Paul, Yee, Robert, Magill, Catherine, Neri, Anthony, Cai, Sui Xiong, Drewe, John, Qiu, Ling, Herich, John, Tseng, Ben, Kasibhatla, Shailaja, Spencer, Jeffrey R.
Published in Bioorganic & medicinal chemistry letters (01.09.2006)
Published in Bioorganic & medicinal chemistry letters (01.09.2006)
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The discovery of a potent PARP1 inhibitor Senaparib
Cai, Sui Xiong, Ma, Ning, Wang, Xiaozhu, Guo, Mingchuan, Jiang, Yangzhen, Tian, Ye E
Published in Molecular cancer therapeutics (26.06.2024)
Published in Molecular cancer therapeutics (26.06.2024)
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Synthesis and SAR of novel di- and trisubstituted 1,4-dihydroquinoxaline-2,3-diones related to licostinel (Acea 1021) as NMDA/glycine site antagonists
Zhou, Zhang-Lin, Kher, Sunil M, Cai, Sui Xiong, Whittemore, Edward R, Espitia, Stephen A, Hawkinson, Jon E, Tran, Minhtam, Woodward, Richard M, Weber, Eckard, Keana, John F.W
Published in Bioorganic & medicinal chemistry (17.04.2003)
Published in Bioorganic & medicinal chemistry (17.04.2003)
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