P.3.c.001 Pharmacological evaluation of new N-phenylpiperazine derivatives designed as homologues of the antipsychotic lead compound LASSBio-579
Noël, F, Pompeu, T.E.T, Alves, F.R.S, Figueiredo, C.D.M, Antonio, C.B, Herzfeldt, V, Rates, S.M.K, Barreiro, E.J, Fraga, C.A.M
Published in European neuropsychopharmacology (01.10.2013)
Published in European neuropsychopharmacology (01.10.2013)
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Impairment of locomotor activity induced by the novel N-acylhydrazone derivatives LASSBio-785 and LASSBio-786 in mice
Silva, G A P, Kummerle, A E, Antunes, F, Fraga, C A M, Barreiro, E J, Zapata-Sudo, G, Sudo, R T
Published in Brazilian journal of medical and biological research (01.03.2013)
Published in Brazilian journal of medical and biological research (01.03.2013)
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Dopaminergic profile of new heterocyclic N-phenylpiperazine derivatives
Neves, G, Fenner, R, Heckler, A P, Viana, A F, Tasso, L, Menegatti, R, Fraga, C A M, Barreiro, E J, Dalla-Costa, T, Rates, S M K
Published in Brazilian journal of medical and biological research (01.05.2003)
Published in Brazilian journal of medical and biological research (01.05.2003)
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Pulmonary hypertension: reduction of vascular and cardiac remodeling by a new inhibitor of p38-alpha MAPK
Silva, G.R.A, Beltrame, F, Alencar, A.K.N, Silva, M.M, Rocha, B, Da Silva, J.S, Montagnoli, T.L, Freitas, R.C, Fraga, C.A.M, Sudo, R.T, Zapata-Sudo, G
Published in European heart journal (01.11.2020)
Published in European heart journal (01.11.2020)
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Design, Synthesis, and Pharmacological Evaluation of N‑Acylhydrazones and Novel Conformationally Constrained Compounds as Selective and Potent Orally Active Phosphodiesterase‑4 Inhibitors
Kümmerle, Arthur E, Schmitt, Martine, Cardozo, Suzana V. S, Lugnier, Claire, Villa, Pascal, Lopes, Alexandra B, Romeiro, Nelilma C, Justiniano, Hélène, Martins, Marco A, Fraga, Carlos A. M, Bourguignon, Jean-Jacques, Barreiro, Eliezer J
Published in Journal of medicinal chemistry (13.09.2012)
Published in Journal of medicinal chemistry (13.09.2012)
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Journal Article
Impairment of locomotor activity induced by the novelN-acylhydrazone derivatives LASSBio-785 and LASSBio-786 in mice
Silva, G.A.P., Kummerle, A.E., Antunes, F., Fraga, C.A.M., Barreiro, E.J., Zapata-Sudo, G., Sudo, R.T.
Published in Brazilian journal of medical and biological research (01.03.2013)
Published in Brazilian journal of medical and biological research (01.03.2013)
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Journal Article
Impairment of locomotor activity induced by the novel N-acylhydrazone derivatives LASSBio-785 and LASSBio-786 in mice
G.A.P. Silva, A.E. Kummerle, F. Antunes, C.A.M. Fraga, E.J. Barreiro, G. Zapata-Sudo, R.T. Sudo
Published in Brazilian journal of medical and biological research (01.03.2013)
Published in Brazilian journal of medical and biological research (01.03.2013)
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Microbial reduction of alpha-substituted-alpha-acetyl-gamma-butyrolactones
Ribeiro, Joyce B., Sousa, L.M.A., Fraga, C.A.M., Leite, Selma G.F., Ramos, M.C.K.V., de Aquino Neto, F.R., Aguiar, L.C.S., de Souza, Rodrigo O.M.A., Antunes, O.A.C.
Published in Catalysis communications (20.04.2008)
Published in Catalysis communications (20.04.2008)
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Journal Article
Development and validation of a LC-MS/MS method with electrospray ionization for determination of LASSBio-579 in rat plasma
Conrado, D.J., Palma, E.C., Fraga, C.A.M., Barreiro, E.J., Rates, S.M.K., Dalla Costa, T.
Published in Journal of pharmaceutical and biomedical analysis (17.01.2007)
Published in Journal of pharmaceutical and biomedical analysis (17.01.2007)
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Journal Article
Validated HPLC method for determination of LASSBio-581, a new heterocyclic N-phenylpiperazine derivative, in rat plasma
Tasso, L., Neves, G., Menegatti, R., Fraga, C.A.M., Barreiro, E.J., Eifler-Lima, V.L., Rates, S.M.K., Dalla Costa, Teresa
Published in Journal of pharmaceutical and biomedical analysis (04.12.2003)
Published in Journal of pharmaceutical and biomedical analysis (04.12.2003)
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Journal Article
Selective PGHS-2 Inhibitors: A Rational Approach for Treatment of theInflammation
Rodrigues, C., Veloso, M., Verli, H., Fraga, C., Miranda, A., Barreiro, E.
Published in Current medicinal chemistry (01.04.2002)
Published in Current medicinal chemistry (01.04.2002)
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A possible molecular mechanism for the inhibition of cysteine proteases by salicylaldehyde N-acylhydrazones and related compounds
Ifa, D.R, Rodrigues, C.R, de Alencastro, R.B, Fraga, C.A.M, Barreiro, E.J
Published in Journal of molecular structure. Theochem (26.06.2000)
Published in Journal of molecular structure. Theochem (26.06.2000)
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