Effects of channel modulators on cloned large-conductance calcium-activated potassium channels
V K Gribkoff, J T Lum-Ragan, C G Boissard, D J Post-Munson, N A Meanwell, J E Starrett, Jr, E S Kozlowski, J L Romine, J T Trojnacki, M C Mckay, J Zhong, S I Dworetzky
Published in Molecular pharmacology (01.07.1996)
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Published in Molecular pharmacology (01.07.1996)
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Targeting acute ischemic stroke with a calcium-sensitive opener of maxi-K potassium channels
Gribkoff, Valentin K, Starrett, John E, Dworetzky, Steven I, Hewawasam, Piyasena, Boissard, Christopher G, Cook, Deborah A, Frantz, Stephen W, Heman, Karen, Hibbard, Jeffrey R, Huston, Kevin, Johnson, Graham, Krishnan, Bala S, Kinney, Gene G, Lombardo, Lynn A, Meanwell, Nicholas A, Molinoff, Perry B, Myers, Robert A, Moon, Sandra L, Ortiz, Astrid, Pajor, Lorraine, Pieschl, Rick L, Post-Munson, Debra J, Signor, Laura J, Srinivas, Nugehally, Taber, Matthew T, Thalody, George, Trojnacki, Joanne T, Wiener, Harvey, Yeleswaram, Krishnaswamy, Yeola, Sarita W
Published in Nature medicine (01.04.2001)
Published in Nature medicine (01.04.2001)
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Age-dependence of effects of A1 adenosine receptor antagonism in rat hippocampal slices
Bauman, L A, Mahle, C D, Boissard, C G, Gribkoff, V K
Published in Journal of neurophysiology (01.08.1992)
Published in Journal of neurophysiology (01.08.1992)
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Journal Article
Formation of intermediate-conductance calcium-activated potassium channels by interaction of Slack and Slo subunits
Kaczmarek, Leonard K, Joiner, William J, Tang, Michael D, Wang, Lu-Yang, Dworetzky, Steven I, Boissard, Christopher G, Gan, Li, Gribkoff, Valentin K
Published in Nature neuroscience (01.10.1998)
Published in Nature neuroscience (01.10.1998)
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Suppressant effect of REM sleep deprivation on neophobia in normal rats and in rats with selective DSP-4 induced damage of locus coeruleus neurons
Mogilnicka, E., Boissard, C.G., Hunn, C., Delini-Stula, A.
Published in Pharmacology, biochemistry and behavior (01.07.1985)
Published in Pharmacology, biochemistry and behavior (01.07.1985)
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Synthesis and Structure−Activity Relationship of Acrylamides as KCNQ2 Potassium Channel Openers
Wu, Yong-Jin, He, Huan, Sun, Li-Qiang, L'Heureux, Alexandre, Chen, Jie, Dextraze, Pierre, Starrett, John E, Boissard, Christopher G, Gribkoff, Valentin K, Natale, Joanne, Dworetzky, Steven I
Published in Journal of medicinal chemistry (20.05.2004)
Published in Journal of medicinal chemistry (20.05.2004)
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The discovery of novel openers of Ca2+-dependent large-conductance potassium channels : Pharmacophore search and physiological evaluation of flavonoids
LI, Y, STARRETT, J. E, MEANWELL, N. A, JOHNSON, G, HARTE, W. E, DWORETZKY, S. I, BOISSARD, C. G, GRIBKOFF, V. K
Published in Bioorganic & medicinal chemistry letters (08.04.1997)
Published in Bioorganic & medicinal chemistry letters (08.04.1997)
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Synthesis and excitatory amino acid pharmacology of some novel quinoxalinediones
Epperson, James R., Hewawasam, Piyasena, Meanwell, Nicholas A., Boissard, Christopher G., Gribkoff, Valentin K., Post-Munson, Debra
Published in Bioorganic & medicinal chemistry letters (01.12.1993)
Published in Bioorganic & medicinal chemistry letters (01.12.1993)
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Journal Article
Synthesis and Structure−Activity Relationships of 3-Aryloxindoles: A New Class of Calcium-Dependent, Large Conductance Potassium (Maxi-K) Channel Openers with Neuroprotective Properties
Hewawasam, Piyasena, Erway, Matthew, Moon, Sandra L, Knipe, Jay, Weiner, Harvey, Boissard, Christopher G, Post-Munson, Debra J, Gao, Qi, Huang, Stella, Gribkoff, Valentin K, Meanwell, Nicholas A
Published in Journal of medicinal chemistry (28.03.2002)
Published in Journal of medicinal chemistry (28.03.2002)
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Synthesis and biological evaluation of an iodinated iberiotoxin analogue, [mono-iodo-Tyr5, Phe36]-iberiotoxin
Kozlowski, E S, Johnson, G, Dischino, D D, Dworetzky, S I, Boissard, C G, Gribkoff, V K
Published in International journal of peptide and protein research (01.08.1996)
Published in International journal of peptide and protein research (01.08.1996)
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Journal Article
Discovery of a novel class of BK channel openers : Enantiospecific synthesis and BK channel opening activity of 3-(5-chloro-2-hydroxyphenyl)-1,3-dihydro-3-hydroxy-6-(trifluoromethyl)-2H-indol-2-one
HEWAWASAM, P, MEANWELL, N. A, GRIBKOFF, V. K, DWORETZKY, S. I, BOISSARD, C. G
Published in Bioorganic & medicinal chemistry letters (20.05.1997)
Published in Bioorganic & medicinal chemistry letters (20.05.1997)
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Journal Article
The synthesis and characterization of BMS-204352 (MaxiPost) and related 3-fluorooxindoles as openers of maxi-K potassium channels
HEWAWASAM, Piyasena, GRIBKOFF, Valentin K, PAJOR, Lorraine M, KNIPE, Jay, QI GAO, PERRONE, Robert, STARRETT, John E, PENDRI, Yadagiri, DWORETZKY, Steven I, MEANWELL, Nicholas A, MARTINEZ, Eduardo, BOISSARD, Christopher G, POST-MUNSON, Debra J, TROJNACKI, Joanne T, YELESWARAM, Krishnaswamy
Published in Bioorganic & medicinal chemistry letters (08.04.2002)
Published in Bioorganic & medicinal chemistry letters (08.04.2002)
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Journal Article
4-Aryl-3-(hydroxyalkyl)quinolin-2-ones: Novel Maxi-K Channel Opening Relaxants of Corporal Smooth Muscle Targeted for Erectile Dysfunction
Hewawasam, Piyasena, Fan, Wenhong, Ding, Min, Flint, Kim, Cook, Deborah, Goggins, Gregory D, Myers, Robert A, Gribkoff, Valentin K, Boissard, Christopher G, Dworetzky, Steven I, Starrett, John E, Lodge, Nicholas J
Published in Journal of medicinal chemistry (03.07.2003)
Published in Journal of medicinal chemistry (03.07.2003)
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Journal Article
4,5-Diphenyltriazol-3-ones: Openers of Large-Conductance Ca super(2+)-Activated Potassium (Maxi-K) Channels
Romine, J L, Martin, S W, Gribkoff, V K, Boissard, C G, Dworetzky, SI, Natale, J, Li, Yi, Gao, Qi, Meanwell, NA, Starrett, JE Jr
Published in Journal of medicinal chemistry (04.07.2002)
Published in Journal of medicinal chemistry (04.07.2002)
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