Discovery of G Protein-Biased D2 Dopamine Receptor Partial Agonists
Chen, Xin, McCorvy, John D, Fischer, Matthew G, Butler, Kyle V, Shen, Yudao, Roth, Bryan L, Jin, Jian
Published in Journal of medicinal chemistry (08.12.2016)
Published in Journal of medicinal chemistry (08.12.2016)
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Journal Article
Development of a S-adenosylmethionine analog that intrudes the RNA-cap binding site of Zika methyltransferase
Jain, Rinku, Butler, Kyle V, Coloma, Javier, Jin, Jian, Aggarwal, Aneel K
Published in Scientific reports (09.05.2017)
Published in Scientific reports (09.05.2017)
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Journal Article
Discovery of a Selective, Substrate-Competitive Inhibitor of the Lysine Methyltransferase SETD8
Ma, Anqi, Yu, Wenyu, Li, Fengling, Bleich, Rachel M, Herold, J. Martin, Butler, Kyle V, Norris, Jacqueline L, Korboukh, Victoria, Tripathy, Ashutosh, Janzen, William P, Arrowsmith, Cheryl H, Frye, Stephen V, Vedadi, Masoud, Brown, Peter J, Jin, Jian
Published in Journal of medicinal chemistry (14.08.2014)
Published in Journal of medicinal chemistry (14.08.2014)
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Journal Article
Structure-Based Design of a Covalent Inhibitor of the SET Domain-Containing Protein 8 (SETD8) Lysine Methyltransferase
Butler, Kyle V, Ma, Anqi, Yu, Wenyu, Li, Fengling, Tempel, Wolfram, Babault, Nicolas, Pittella-Silva, Fabio, Shao, Jason, Wang, Junyi, Luo, Minkui, Vedadi, Masoud, Brown, Peter J, Arrowsmith, Cheryl H, Jin, Jian
Published in Journal of medicinal chemistry (10.11.2016)
Published in Journal of medicinal chemistry (10.11.2016)
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Journal Article
MS0621, a novel small-molecule modulator of Ewing sarcoma chromatin accessibility, interacts with an RNA-associated macromolecular complex and influences RNA splicing
Vital, Tamara, Wali, Aminah, Butler, Kyle V, Xiong, Yan, Foster, 2nd, Joseph P, Marcel, Shelsa S, McFadden, Andrew W, Nguyen, Valerie U, Bailey, Benton M, Lamb, Kelsey N, James, Lindsey I, Frye, Stephen V, Mosely, Amber L, Jin, Jian, Pattenden, Samantha G, Davis, Ian J
Published in Frontiers in oncology (30.01.2023)
Published in Frontiers in oncology (30.01.2023)
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Journal Article
Novel Inhibitors of Human Histone Deacetylase (HDAC) Identified by QSAR Modeling of Known Inhibitors, Virtual Screening, and Experimental Validation
Tang, Hao, Wang, Xiang S, Huang, Xi-Ping, Roth, Bryan L, Butler, Kyle V, Kozikowski, Alan P, Jung, Mira, Tropsha, Alexander
Published in Journal of Chemical Information and Modeling (23.02.2009)
Published in Journal of Chemical Information and Modeling (23.02.2009)
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Journal Article
Structure-inspired design of β-arrestin-biased ligands for aminergic GPCRs
McCorvy, John D, Butler, Kyle V, Kelly, Brendan, Rechsteiner, Katie, Karpiak, Joel, Betz, Robin M, Kormos, Bethany L, Shoichet, Brian K, Dror, Ron O, Jin, Jian, Roth, Bryan L
Published in Nature chemical biology (01.02.2018)
Published in Nature chemical biology (01.02.2018)
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Journal Article
A Potent, Selective, and Cell-Active Inhibitor of Human Type I Protein Arginine Methyltransferases
Eram, Mohammad S, Shen, Yudao, Szewczyk, Magdalena M, Wu, Hong, Senisterra, Guillermo, Li, Fengling, Butler, Kyle V, Kaniskan, H. Ümit, Speed, Brandon A, dela Seña, Carlo, Dong, Aiping, Zeng, Hong, Schapira, Matthieu, Brown, Peter J, Arrowsmith, Cheryl H, Barsyte-Lovejoy, Dalia, Liu, Jing, Vedadi, Masoud, Jin, Jian
Published in ACS chemical biology (18.03.2016)
Published in ACS chemical biology (18.03.2016)
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Journal Article
Dose-dependent activation of gene expression is achieved using CRISPR and small molecules that recruit endogenous chromatin machinery
Chiarella, Anna M, Butler, Kyle V, Gryder, Berkley E, Lu, Dongbo, Wang, Tiffany A, Yu, Xufen, Pomella, Silvia, Khan, Javed, Jin, Jian, Hathaway, Nathaniel A
Published in Nature biotechnology (01.01.2020)
Published in Nature biotechnology (01.01.2020)
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Journal Article
Report and Application of a Tool Compound Data Set
Butler, Kyle V, MacDonald, Ian A, Hathaway, Nathaniel A, Jin, Jian
Published in Journal of chemical information and modeling (27.11.2017)
Published in Journal of chemical information and modeling (27.11.2017)
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Journal Article
Stereoselective HDAC Inhibition from Cysteine-Derived Zinc-Binding Groups
Butler, Kyle V., He, Rong, McLaughlin, Kathryn, Vistoli, Giulio, Langley, Brett, Kozikowski, Alan P.
Published in ChemMedChem (03.08.2009)
Published in ChemMedChem (03.08.2009)
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Journal Article
Structure-activity relationship studies of SETD8 inhibitors
Ma, Anqi, Yu, Wenyu, Xiong, Yan, Butler, Kyle V, Brown, Peter J, Jin, Jian
Published in MedChemComm (01.12.2014)
Published in MedChemComm (01.12.2014)
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Journal Article
Non-substrate based, small molecule inhibitors of the human isoprenylcysteine carboxyl methyltransferase
Butler, Kyle V., Bohn, Kelsey, Hrycyna, Christine A., Jin, Jian
Published in MedChemComm (01.01.2016)
Published in MedChemComm (01.01.2016)
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Journal Article
Pathway-Based High-Throughput Chemical Screen Identifies Compounds That Decouple Heterochromatin Transformations
MacDonald, Ian A., Butler, Kyle V., Herring, Laura E., Clinkscales, Sarah E., Yelagandula, Ramesh, Stecher, Karin, Bell, Oliver, Graves, Lee M., Jin, Jian, Hathaway, Nathaniel A.
Published in SLAS discovery (01.09.2019)
Published in SLAS discovery (01.09.2019)
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