Design and Synthesis of Inhaled p38 Inhibitors for the Treatment of Chronic Obstructive Pulmonary Disease
Millan, David S, Bunnage, Mark E, Burrows, Jane L, Butcher, Kenneth J, Dodd, Peter G, Evans, Timothy J, Fairman, David A, Hughes, Samantha J, Kilty, Iain C, Lemaitre, Arnaud, Lewthwaite, Russell A, Mahnke, Axel, Mathias, John P, Philip, James, Smith, Robert T, Stefaniak, Mark H, Yeadon, Michael, Phillips, Christopher
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Published in Journal of medicinal chemistry (24.11.2011)
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Sustained delivery by leucine-modified chitosan spray-dried respirable powders
Learoyd, Tristan P., Burrows, Jane L., French, Eddie, Seville, Peter C.
Published in International journal of pharmaceutics (08.05.2009)
Published in International journal of pharmaceutics (08.05.2009)
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Inhalation by Design: Novel Ultra-Long-Acting beta(2)-Adrenoreceptor Agonists for Inhaled Once-Daily Treatment of Asthma and Chronic Obstructive Pulmonary Disease That Utilize a Sulfonamide Agonist Headgroup
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Published in Journal of medicinal chemistry (23.09.2010)
Published in Journal of medicinal chemistry (23.09.2010)
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Inhalation by Design: Novel Ultra-Long-Acting β2-Adrenoreceptor Agonists for Inhaled Once-Daily Treatment of Asthma and Chronic Obstructive Pulmonary Disease That Utilize a Sulfonamide Agonist Headgroup
Glossop, Paul A, Lane, Charlotte A. L, Price, David A, Bunnage, Mark E, Lewthwaite, Russell A, James, Kim, Brown, Alan D, Yeadon, Michael, Perros-Huguet, Christelle, Trevethick, Michael A, Clarke, Nicholas P, Webster, Robert, Jones, Rhys M, Burrows, Jane L, Feeder, Neil, Taylor, Stefan C. J, Spence, Fiona J
Published in Journal of medicinal chemistry (23.09.2010)
Published in Journal of medicinal chemistry (23.09.2010)
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Modified release of beclometasone dipropionate from chitosan-based spray-dried respirable powders
Learoyd, Tristan P., Burrows, Jane L., French, Eddie, Seville, Peter C.
Published in Powder technology (20.11.2008)
Published in Powder technology (20.11.2008)
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Molecular hybridization yields triazole bronchodilators for the treatment of COPD
Jones, Lyn H., Burrows, Jane, Feeder, Neil, Glossop, Paul, James, Kim, Jones, Rhys M., Kenyon, Amy S., Patel, Sheena, Roberts, Dannielle F., Selby, Matthew D., Strang, Ross S., Stuart, Emilio F., Trevethick, Michael A., Watson, Jessica, Wright, Karen N., Clarke, Nick
Published in Bioorganic & medicinal chemistry letters (15.11.2015)
Published in Bioorganic & medicinal chemistry letters (15.11.2015)
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Inhalation by Design: Novel Tertiary Amine Muscarinic M-3 Receptor Antagonists with Slow Off-Rate Binding Kinetics for Inhaled Once-Daily Treatment of Chronic Obstructive Pulmonary Disease
Glossop, Paul A., Watson, Christine A. L., Price, David A., Bunnage, Mark E., Middleton, Donald S., Wood, Anthony, James, Kim, Roberts, Dannielle, Strang, Ross S., Yeadon, Michael, Perros-Huguet, Christelle, Clarke, Nicholas P., Trevethick, Michael A., Machin, Ian, Stuart, Emilio F., Evans, Steven M., Harrison, Anthony C., Fairman, David A., Agoram, Balaji, Burrows, Jane L., Feeder, Neil, Fulton, Craig K., Dillon, Barry R., Entwistle, David A., Spence, Fiona J.
Published in Journal of medicinal chemistry (13.10.2011)
Published in Journal of medicinal chemistry (13.10.2011)
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Inhalation by design: Dual pharmacology β-2 agonists/M3 antagonists for the treatment of COPD
Jones, Lyn H., Baldock, Helen, Bunnage, Mark E., Burrows, Jane, Clarke, Nick, Coghlan, Michele, Entwistle, David, Fairman, David, Feeder, Neil, Fulton, Craig, Hilton, Laura, James, Kim, Jones, Rhys M., Kenyon, Amy S., Marshall, Stuart, Newman, Sandra D., Osborne, Rachel, Patel, Sheena, Selby, Matthew D., Stuart, Emilio F., Trevethick, Michael A., Wright, Karen N., Price, David A.
Published in Bioorganic & medicinal chemistry letters (01.05.2011)
Published in Bioorganic & medicinal chemistry letters (01.05.2011)
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Journal Article
Inhalation by Design: Novel Tertiary Amine Muscarinic M3 Receptor Antagonists with Slow Off-Rate Binding Kinetics for Inhaled Once-Daily Treatment of Chronic Obstructive Pulmonary Disease
Glossop, Paul A, Watson, Christine A. L, Price, David A, Bunnage, Mark E, Middleton, Donald S, Wood, Anthony, James, Kim, Roberts, Dannielle, Strang, Ross S, Yeadon, Michael, Perros-Huguet, Christelle, Clarke, Nicholas P, Trevethick, Michael A, Machin, Ian, Stuart, Emilio F, Evans, Steven M, Harrison, Anthony C, Fairman, David A, Agoram, Balaji, Burrows, Jane L, Feeder, Neil, Fulton, Craig K, Dillon, Barry R, Entwistle, David A, Spence, Fiona J
Published in Journal of medicinal chemistry (13.10.2011)
Published in Journal of medicinal chemistry (13.10.2011)
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Journal Article
Inhalation by Design: Novel Ultra-Long-Acting β 2 -Adrenoreceptor Agonists for Inhaled Once-Daily Treatment of Asthma and Chronic Obstructive Pulmonary Disease That Utilize a Sulfonamide Agonist Headgroup
Glossop, Paul A., Lane, Charlotte A. L., Price, David A., Bunnage, Mark E., Lewthwaite, Russell A., James, Kim, Brown, Alan D., Yeadon, Michael, Perros-Huguet, Christelle, Trevethick, Michael A., Clarke, Nicholas P., Webster, Robert, Jones, Rhys M., Burrows, Jane L., Feeder, Neil, Taylor, Stefan C. J., Spence, Fiona J.
Published in Journal of medicinal chemistry (23.09.2010)
Published in Journal of medicinal chemistry (23.09.2010)
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Optimized glucuronidation of dual pharmacology β-2 agonists/M3 antagonists for the treatment of COPD
Hilton, Laura, Osborne, Rachel, Kenyon, Amy S., Baldock, Helen, Bunnage, Mark E., Burrows, Jane, Clarke, Nick, Coghlan, Michele, Entwistle, David, Fairman, David, Feeder, Neil, James, Kim, Jones, Rhys M., Laouar, Nadia, Lunn, Graham, Marshall, Stuart, Newman, Sandra D., Patel, Sheena, Selby, Matthew D., Spence, Fiona, Stuart, Emilio F., Summerhill, Susan, Trevethick, Michael A., Wright, Karen N., Yeadon, Michael, Price, David A., Jones, Lyn H.
Published in MedChemComm (01.09.2011)
Published in MedChemComm (01.09.2011)
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