Aripiprazole, a Novel Antipsychotic, Is a High-Affinity Partial Agonist at Human Dopamine D2 Receptors
Burris, Kevin D, Molski, Thaddeus F, Xu, Cen, Ryan, Elaine, Tottori, Katsura, Kikuchi, Tetsuro, Yocca, Frank D, Molinoff, Perry B
Published in The Journal of pharmacology and experimental therapeutics (01.07.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2002)
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The novel antipsychotic aripiprazole is a partial agonist at short and long isoforms of D2 receptors linked to the regulation of adenylyl cyclase activity and prolactin release
AIHARA, Koutoku, SHIMADA, Jun, MIWA, Takashi, TOTTORI, Katsura, BURRIS, Kevin D, YOCCA, Frank D, HORIE, Masato, KIKUCHI, Tetsuro
Published in Brain research (02.04.2004)
Published in Brain research (02.04.2004)
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Forebrain-selective AMPA-receptor antagonism guided by TARP γ-8 as an antiepileptic mechanism
Kato, Akihiko S, Burris, Kevin D, Gardinier, Kevin M, Gernert, Douglas L, Porter, Warren J, Reel, Jon, Ding, Chunjin, Tu, Yuan, Schober, Douglas A, Lee, Matthew R, Heinz, Beverly A, Fitch, Thomas E, Gleason, Scott D, Catlow, John T, Yu, Hong, Fitzjohn, Stephen M, Pasqui, Francesca, Wang, He, Qian, Yuewei, Sher, Emanuele, Zwart, Ruud, Wafford, Keith A, Rasmussen, Kurt, Ornstein, Paul L, Isaac, John T R, Nisenbaum, Eric S, Bredt, David S, Witkin, Jeffrey M
Published in Nature medicine (01.12.2016)
Published in Nature medicine (01.12.2016)
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Bias analyses of preclinical and clinical D2 dopamine ligands: studies with immediate and complex signaling pathways
Brust, Tarsis F, Hayes, Michael P, Roman, David L, Burris, Kevin D, Watts, Val J
Published in The Journal of pharmacology and experimental therapeutics (01.03.2015)
Published in The Journal of pharmacology and experimental therapeutics (01.03.2015)
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Discovery of the First α‑Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor Antagonist Dependent upon Transmembrane AMPA Receptor Regulatory Protein (TARP) γ‑8
Gardinier, Kevin M, Gernert, Douglas L, Porter, Warren J, Reel, Jon K, Ornstein, Paul L, Spinazze, Patrick, Stevens, F. Craig, Hahn, Patric, Hollinshead, Sean P, Mayhugh, Daniel, Schkeryantz, Jeff, Khilevich, Albert, De Frutos, Oscar, Gleason, Scott D, Kato, Akihiko S, Luffer-Atlas, Debra, Desai, Prashant V, Swanson, Steven, Burris, Kevin D, Ding, Chunjin, Heinz, Beverly A, Need, Anne B, Barth, Vanessa N, Stephenson, Gregory A, Diseroad, Benjamin A, Woods, Tim A, Yu, Hong, Bredt, David, Witkin, Jeffrey M
Published in Journal of medicinal chemistry (26.05.2016)
Published in Journal of medicinal chemistry (26.05.2016)
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Modulation of TARP γ8-Containing AMPA Receptors as a Novel Therapeutic Approach for Chronic Pain
Knopp, Kelly L, Simmons, Rosa Maria A, Guo, Wenhong, Adams, Benjamin L, Gardinier, Kevin M, Gernert, Douglas L, Ornstein, Paul L, Porter, Warren, Reel, Jon, Ding, Chunjin, Wang, He, Qian, Yuewei, Burris, Kevin D, Need, Anne, Barth, Vanessa, Swanson, Steven, Catlow, John, Witkin, Jeffrey M, Zwart, Ruud, Sher, Emanuele, Choong, Kar-Chan, Wall, Theron M, Schober, Douglas, Felder, Christian C, Kato, Akihiko S, Bredt, David S, Nisenbaum, Eric S
Published in The Journal of pharmacology and experimental therapeutics (01.06.2019)
Published in The Journal of pharmacology and experimental therapeutics (01.06.2019)
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Interaction of the novel antipsychotic aripiprazole with 5-HT1A and 5-HT2A receptors : functional receptor-binding and in vivo electrophysiological studies
STARK, Arlene D, JORDAN, Shaun, BURRIS, Kevin D, ALLERS, Kelly A, BERTEKAP, Robert L, CHEN, Ruoyan, MISTRY KANNAN, Tanaz, MOLSKI, Thaddeus F, YOCCA, Frank D, SHARP, Trevor, KIKUCHI, Tetsuro
Published in Psychopharmacologia (01.02.2007)
Published in Psychopharmacologia (01.02.2007)
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Modulation of TARP γ 8-Containing AMPA Receptors as a Novel Therapeutic Approach for Chronic Pain
Knopp, Kelly L, Simmons, Rosa Maria A, Guo, Wenhong, Adams, Benjamin L, Gardinier, Kevin M, Gernert, Douglas L, Ornstein, Paul L, Porter, Warren, Reel, Jon, Ding, Chunjin, Wang, He, Qian, Yuewei, Burris, Kevin D, Need, Anne, Barth, Vanessa, Swanson, Steven, Catlow, John, Witkin, Jeffrey M, Zwart, Ruud, Sher, Emanuele, Choong, Kar-Chan, Wall, Theron M, Schober, Douglas, Felder, Christian C, Kato, Akihiko S, Bredt, David S, Nisenbaum, Eric S
Published in The Journal of pharmacology and experimental therapeutics (01.06.2019)
Published in The Journal of pharmacology and experimental therapeutics (01.06.2019)
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An Integrated Approach for Screening and Identification of Positive Allosteric Modulators of N-Methyl-D-Aspartate Receptors
Jambrina, Enrique, Cerne, Rok, Smith, Emery, Scampavia, Louis, Cuadrado, Maria, Findlay, Jeremy, Krambis, Michael J, Wakulchik, Mark, Chase, Peter, Brunavs, Michael, Burris, Kevin D, Gallagher, Peter, Spicer, Timothy P, Ursu, Daniel
Published in Journal of biomolecular screening (01.06.2016)
Published in Journal of biomolecular screening (01.06.2016)
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Aripiprazole's low intrinsic activities at human dopamine D2L and D2S receptors render it a unique antipsychotic
Tadori, Yoshihiro, Miwa, Takashi, Tottori, Katsura, Burris, Kevin D., Stark, Arlene, Mori, Toyoki, Kikuchi, Tetsuro
Published in European journal of pharmacology (16.05.2005)
Published in European journal of pharmacology (16.05.2005)
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Mechanism of action of aripiprazole predicts clinical efficacy and a favourable side-effect profile
Hirose, Tsuyoshi, Uwahodo, Yasufumi, Yamada, Sakiko, Miwa, Takashi, Kikuchi, Tetsuro, Kitagawa, Hisashi, Burris, Kevin D, Altar, C Anthony, Nabeshima, Toshitaka
Published in Journal of psychopharmacology (Oxford) (01.09.2004)
Published in Journal of psychopharmacology (Oxford) (01.09.2004)
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Drug-induced sensitization of adenylyl cyclase: assay streamlining and miniaturization for small molecule and siRNA screening applications
Conley, Jason M, Brust, Tarsis F, Xu, Ruqiang, Burris, Kevin D, Watts, Val J
Published in Journal of visualized experiments (27.01.2014)
Published in Journal of visualized experiments (27.01.2014)
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Oxime Carbamate—Discovery of a series of novel FAAH inhibitors
Sit, S.Y., Conway, Charles M., Xie, Kai, Bertekap, Robert, Bourin, Clotilde, Burris, Kevin D.
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Design, synthesis and evaluation of constrained tetrahydroimidazopyrimidine derivatives as antagonists of corticotropin-releasing factor type 1 receptor (CRF 1R)
Vrudhula, Vivekananda M., Dasgupta, Bireshwar, Pin, Sokhom S., Burris, Kevin D., Balanda, Lynn A., Fung, Lawrence K., Fiedler, Tracey, Browman, Kaitlin E., Taber, Matthew T., Zhang, Jie, Macor, John E., Dubowchik, Gene M.
Published in Bioorganic & medicinal chemistry letters (15.03.2010)
Published in Bioorganic & medicinal chemistry letters (15.03.2010)
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Diminished catalepsy and dopamine metabolism distinguish aripiprazole from haloperidol or risperidone
Nakai, Satoru, Hirose, Tsuyoshi, Uwahodo, Yasufumi, Imaoka, Takeshi, Okazaki, Hiroshi, Miwa, Takashi, Nakai, Masami, Yamada, Sakiko, Dunn, Bob, Burris, Kevin D, Molinoff, Perry B, Tottori, Katsura, Altar, C.Anthony, Kikuchi, Tetsuro
Published in European journal of pharmacology (04.07.2003)
Published in European journal of pharmacology (04.07.2003)
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Synthesis, structure–activity relationships, and anxiolytic activity of 7-aryl-6,7-dihydroimidazoimidazole corticotropin-releasing factor 1 receptor antagonists
Han, Xiaojun, Michne, Jodi A., Pin, Sokhom S., Burris, Kevin D., Balanda, Lynn A., Fung, Lawrence K., Fiedler, Tracey, Browman, Kaitlin E., Taber, Matthew T., Zhang, Jie, Dubowchik, Gene M.
Published in Bioorganic & medicinal chemistry letters (01.09.2005)
Published in Bioorganic & medicinal chemistry letters (01.09.2005)
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Synthesis and SAR exploration of dinapsoline analogues
Sit, Sing-Yuen, Xie, Kai, Jacutin-Porte, Swanee, Boy, Kenneth M, Seanz, James, Taber, Matthew T, Gulwadi, Amit G, Korpinen, Carolyn D, Burris, Kevin D, Molski, Thaddeus F, Ryan, Elaine, Xu, Cen, Verdoorn, Todd, Johnson, Graham, Nichols, David E, Mailman, Richard B
Published in Bioorganic & medicinal chemistry (15.02.2004)
Published in Bioorganic & medicinal chemistry (15.02.2004)
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