Turning Up the Heat on MYC: Progress in Small-Molecule Inhibitors
Truica, Mihai I, Burns, Michael C, Han, Huiying, Abdulkadir, Sarki A
Published in Cancer research (Chicago, Ill.) (15.01.2021)
Published in Cancer research (Chicago, Ill.) (15.01.2021)
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Journal Article
Approach for targeting Ras with small molecules that activate SOS-mediated nucleotide exchange
Burns, Michael C., Qi Sun, Daniels, R. Nathan, Camper, DeMarco, Kennedy, J. Phillip, Phan, Jason, Olejniczak, Edward T., Lee, Taekyu, Waterson, Alex G., Rossanese, Olivia W., Fesik, Stephen W.
Published in Proceedings of the National Academy of Sciences - PNAS (04.03.2014)
Published in Proceedings of the National Academy of Sciences - PNAS (04.03.2014)
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Journal Article
Discovery and Structure-Based Optimization of Benzimidazole-Derived Activators of SOS1-Mediated Nucleotide Exchange on RAS
Hodges, Timothy R, Abbott, Jason R, Little, Andrew J, Sarkar, Dhruba, Salovich, James M, Howes, Jennifer E, Akan, Denis T, Sai, Jiqing, Arnold, Allison L, Browning, Carrie, Burns, Michael C, Sobolik, Tammy, Sun, Qi, Beesetty, Yugandhar, Coker, Jesse A, Scharn, Dirk, Stadtmueller, Heinz, Rossanese, Olivia W, Phan, Jason, Waterson, Alex G, McConnell, Darryl B, Fesik, Stephen W
Published in Journal of medicinal chemistry (11.10.2018)
Published in Journal of medicinal chemistry (11.10.2018)
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Journal Article
Discovery of Small Molecules that Bind to K-Ras and Inhibit Sos-Mediated Activation
Sun, Qi, Burke, Jason P., Phan, Jason, Burns, Michael C., Olejniczak, Edward T., Waterson, Alex G., Lee, Taekyu, Rossanese, Olivia W., Fesik, Stephen W.
Published in Angewandte Chemie (International ed.) (18.06.2012)
Published in Angewandte Chemie (International ed.) (18.06.2012)
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Journal Article
High-throughput screening identifies small molecules that bind to the RAS:SOS:RAS complex and perturb RAS signaling
Burns, Michael C., Howes, Jennifer E., Sun, Qi, Little, Andrew J., Camper, DeMarco V., Abbott, Jason R., Phan, Jason, Lee, Taekyu, Waterson, Alex G., Rossanese, Olivia W., Fesik, Stephen W.
Published in Analytical biochemistry (01.05.2018)
Published in Analytical biochemistry (01.05.2018)
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Journal Article
Small Molecule-Mediated Activation of RAS Elicits Biphasic Modulation of Phospho-ERK Levels that Are Regulated through Negative Feedback on SOS1
Howes, Jennifer E, Akan, Denis T, Burns, Michael C, Rossanese, Olivia W, Waterson, Alex G, Fesik, Stephen W
Published in Molecular cancer therapeutics (01.05.2018)
Published in Molecular cancer therapeutics (01.05.2018)
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Journal Article
Epidemiology, mutational landscape and staging of hepatocellular carcinoma
Fenton, Sarah E, Burns, Michael C, Kalyan, Aparna
Published in Chinese Clinical Oncology (01.02.2021)
Published in Chinese Clinical Oncology (01.02.2021)
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Journal Article
Discovery of Aminopiperidine Indoles That Activate the Guanine Nucleotide Exchange Factor SOS1 and Modulate RAS Signaling
Abbott, Jason R, Hodges, Timothy R, Daniels, R. Nathan, Patel, Pratiq A, Kennedy, J. Phillip, Howes, Jennifer E, Akan, Denis T, Burns, Michael C, Sai, Jiqing, Sobolik, Tammy, Beesetty, Yugandhar, Lee, Taekyu, Rossanese, Olivia W, Phan, Jason, Waterson, Alex G, Fesik, Stephen W
Published in Journal of medicinal chemistry (26.07.2018)
Published in Journal of medicinal chemistry (26.07.2018)
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Journal Article
Early-onset metastatic and clinically advanced prostate cancer is a distinct clinical and molecular entity characterized by increased TMPRSS2-ERG fusions
Chalmers, Zachary R, Burns, Michael C, Ebot, Ericka M, Frampton, Garrett M, Ross, Jeffrey S, Hussain, Maha H A, Abdulkadir, Sarki A
Published in Prostate cancer and prostatic diseases (01.06.2021)
Published in Prostate cancer and prostatic diseases (01.06.2021)
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Journal Article
Discovery of Quinazolines That Activate SOS1-Mediated Nucleotide Exchange on RAS
Abbott, Jason R, Patel, Pratiq A, Howes, Jennifer E, Akan, Denis T, Kennedy, J. Phillip, Burns, Michael C, Browning, Carrie F, Sun, Qi, Rossanese, Olivia W, Phan, Jason, Waterson, Alex G, Fesik, Stephen W
Published in ACS medicinal chemistry letters (13.09.2018)
Published in ACS medicinal chemistry letters (13.09.2018)
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Journal Article
Layered Heterometallic Iodoplumbate Containing a Novel Pb3Cu6I16 Net: Structure and Optical Properties
Burns, Michael C, Tershansy, Meredith A, Ellsworth, Joseph M, Khaliq, Zeeshan, Peterson, LeRoy, Smith, Mark D, zur Loye, Hans-Conrad
Published in Inorganic chemistry (25.12.2006)
Published in Inorganic chemistry (25.12.2006)
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Journal Article
Clinical utility of targeted next generation sequencing (NGS) to predict response to neoadjuvant therapy (NT) in rectal cancer (RC)
Carroll, Kristen, Burns, Michael C., Jones, Ryan, Kocherginsky, Masha, Burdett, Kirsten Bell, Yang, Guang-Yu, Benson, Al Bowen, Mahalingam, Devalingam
Published in Journal of clinical oncology (01.02.2020)
Published in Journal of clinical oncology (01.02.2020)
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Journal Article
Molecular profiling of early-stage colorectal cancer (CRC) using targeted next generation sequencing (NGS) to predict signatures of recurrence
Burns, Michael C., Carroll, Kristen, Jones, Ryan, Kocherginsky, Masha, Burdett, Kirsten Bell, Yang, Guang-Yu, Benson, Al Bowen, Mahalingam, Deva
Published in Journal of clinical oncology (01.02.2020)
Published in Journal of clinical oncology (01.02.2020)
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Journal Article
A phase II study of sEphB4-HSA in metastatic castration-resistant prostate cancer (mCRPC)
Burns, Michael C., Sagar, Vinay, Jovanovic, Borko, Morgans, Alicia K., VanderWeele, David James, Quinn, David I., Stadler, Walter Michael, Abdulkadir, Sarki, Hussain, Maha H. A.
Published in Journal of clinical oncology (20.02.2020)
Published in Journal of clinical oncology (20.02.2020)
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Journal Article
Abstract PS2-08: Identification of incidental putative germline variants in circulating tumor DNA
Davis, Andrew A, Burns, Michael C, Gerratana, Lorenzo, D'Amico, Paolo, Jacob, Saya, Shah, Ami, Katam, Neelima, Wehbe, Firas, Zhang, Qiang, Vagia, Elena, Flaum, Lisa, Siziopikou, Kalliopi P., Platanias, Leonidas C, Behdad, Amir, Gradishar, William J, Cristofanilli, Massimo
Published in Cancer research (Chicago, Ill.) (15.02.2021)
Published in Cancer research (Chicago, Ill.) (15.02.2021)
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Journal Article
Discovery of Small Molecules that Bind to K‐Ras and Inhibit Sos‐Mediated Activation
Sun, Qi, Burke, Jason P., Phan, Jason, Burns, Michael C., Olejniczak, Edward T., Waterson, Alex G., Lee, Taekyu, Rossanese, Olivia W., Fesik, Stephen W.
Published in Angewandte Chemie (18.06.2012)
Published in Angewandte Chemie (18.06.2012)
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Journal Article
Abstract 865: Small molecule-mediated modulation of Ras elicits inhibition of phospho ERK signaling through negative feedback on SOS1
Howes, Jennifer E., Akan, Denis T., Burns, Michael C., Sun, Qi, Little, Andrew J., Camper, DeMarco V., Abbott, Jason R., Phan, Jason, Lee, Taekyu, Rossanese, Olivia W., Waterson, Alex G., Fesik, Stephen W.
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
High-throughput screening identifies small molecules that bind to the RAS:SOS:RAS complex and perturb RAS signaling
Burns, Michael C., Howes, Jennifer E., Sun, Qi, Little, Andrew J., Camper, DeMarco V., Abbott, Jason R., Phan, Jason, Lee, Taekyu, Waterson, Alex G., Rossanese, Olivia W., Fesik, Stephen W.
Published in Analytical biochemistry (01.05.2018)
Published in Analytical biochemistry (01.05.2018)
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Journal Article