Salicylhydrazine-Containing Inhibitors of HIV-1 Integrase: Implication for a Selective Chelation in the Integrase Active Site
Neamati, Nouri, Hong, Huixiao, Owen, Joshua M, Sunder, Sanjay, Winslow, Heather E, Christensen, John L, Zhao, He, Burke, Terrence R, Milne, George W. A, Pommier, Yves
Published in Journal of medicinal chemistry (13.08.1998)
Published in Journal of medicinal chemistry (13.08.1998)
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Journal Article
Structure of the Catalytic Domain of Avian Sarcoma Virus Integrase with a Bound HIV-1 Integrase-Targeted Inhibitor
Lubkowski, Jacek, Yang, Fan, Alexandratos, Jerry, Wlodawer, Alexander, Zhao, He, Burke, Terrence R., Neamati, Nouri, Pommier, Yves, Merkel, George, Skalka, Anna Marie
Published in Proceedings of the National Academy of Sciences - PNAS (28.04.1998)
Published in Proceedings of the National Academy of Sciences - PNAS (28.04.1998)
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Peptide-based inhibitors of Plk1 polo-box domain containing mono-anionic phosphothreonine esters and their pivaloyloxymethyl prodrugs
Qian, Wen-Jian, Park, Jung-Eun, Lim, Dan, Park, Suk-Youl, Lee, Ki-Won, Yaffe, Michael B, Lee, Kyung S, Burke, Jr, Terrence R
Published in Chemistry & biology (24.10.2013)
Published in Chemistry & biology (24.10.2013)
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15-Deoxy-Δ12,14-prostaglandin j2 inhibits transcriptional activity of estrogen receptor-α via covalent modification of DNA-binding domain
KIM, Han-Jong, KIM, Joon-Young, ZHAOJING MENG, LI HUA WANG, FA LIU, CONRADS, Thomas P, BURKE, Terrence R, VEENSTRA, Timothy D, FARRAR, William L
Published in Cancer research (Chicago, Ill.) (15.03.2007)
Published in Cancer research (Chicago, Ill.) (15.03.2007)
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Examination of novel non-phosphorus-containing phosphotyrosyl mimetics against protein-tyrosine phosphatase-1B and demonstration of differential affinities toward Grb2 SH2 domains
Gao, Y, Wu, L, Luo, J H, Guo, R, Yang, D, Zhang, Z Y, Burke, Jr, T R
Published in Bioorganic & medicinal chemistry letters (01.05.2000)
Published in Bioorganic & medicinal chemistry letters (01.05.2000)
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Journal Article
Enantioselective synthesis of nonphosphorus-containing phosphotyrosyl mimetics and their use in the preparation of tyrosine phosphatase inhibitory peptides
Burke, Terrence R, Yao, Zhu-Jun, Zhao, He, Milne, George W.A, Wu, Li, Zhang, Zhong-Yin, Voigt, Johannes H
Published in Tetrahedron (20.08.1998)
Published in Tetrahedron (20.08.1998)
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Effect of DNA Modifications on DNA Processing by HIV-1 Integrase and Inhibitor Binding
Johnson, Allison A., Sayer, Jane M., Yagi, Haruhiko, Patil, Sachindra S., Debart, Françoise, Maier, Martin A., Corey, David R., Vasseur, Jean-Jacques, Burke, Terrence R., Marquez, Victor E., Jerina, Donald M., Pommier, Yves
Published in The Journal of biological chemistry (27.10.2006)
Published in The Journal of biological chemistry (27.10.2006)
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Phosphoryltyrosyl mimetics in the design of peptide-based signal transduction inhibitors
Burke Jr, Terrence R., Yao, Zhu-Jun, Liu, Ding-Guo, Voigt, Johannes, Gao, Yang
Published in Biopolymers (2001)
Published in Biopolymers (2001)
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Journal Article
4‘-O-[2-(2-Fluoromalonyl)]-l-tyrosine: A Phosphotyrosyl Mimic for the Preparation of Signal Transduction Inhibitory Peptides
Burke, Terrence R, Ye, Bin, Akamatsu, Miki, Ford, Harry, Yan, Xinjian, Kole, Hemanta K, Wolf, Gert, Shoelson, Steven E, Roller, Peter P
Published in Journal of medicinal chemistry (01.03.1996)
Published in Journal of medicinal chemistry (01.03.1996)
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Enantioselective Synthesis of N α-Fmoc Protected (2S,3R)-3-Phenylpipecolic Acid. A Constrained Phenylalanine Analogue Suitably Protected for Solid-Phase Peptide Synthesis
Liu, Ding-Guo, Gao, Yang, Wang, Xiangzhu, Kelley, James A, Burke, Terrence R
Published in Journal of organic chemistry (08.03.2002)
Published in Journal of organic chemistry (08.03.2002)
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Journal Article
Elucidation of New Binding Interactions with the Tumor Susceptibility Gene 101 (Tsg101) Protein Using Modified HIV-1 Gag-p6 Derived Peptide Ligands
Kim, Sung-Eun, Liu, Fa, Im, Young Jun, Stephen, Andrew G, Fivash, Matthew J, Waheed, Abdul A, Freed, Eric O, Fisher, Robert J, Hurley, James H, Burke, Jr, Terrence R
Published in ACS medicinal chemistry letters (12.05.2011)
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Published in ACS medicinal chemistry letters (12.05.2011)
Journal Article
A Phosphotyrosyl Mimetic Peptide Reverses Impairment of Insulin-Stimulated Translocation of GLUT4 Caused by Overexpression of PTP1B in Rat Adipose Cells
Chen, Hui, Cong, Li-Na, Li, Yunhua, Yao, Zhu-Jun, Wu, Li, Zhang, Zhong-Yin, Burke, Terrence R, Quon, Michael J
Published in Biochemistry (Easton) (05.01.1999)
Published in Biochemistry (Easton) (05.01.1999)
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Journal Article
Utilization of a Peptide Lead for the Discovery of a Novel PTP1B-Binding Motif
Gao, Yang, Voigt, Johannes, Zhao, He, Pais, Godwin C. G, Zhang, Xuechun, Wu, Li, Zhang, Zhong-Yin, Burke, Terrence R
Published in Journal of medicinal chemistry (30.08.2001)
Published in Journal of medicinal chemistry (30.08.2001)
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Journal Article
Inhibition of SH2 domain/phosphoprotein association by a nonhydrolyzable phosphonopeptide
Domchek, Susan M, Auger, Kurt R, Chatterjee, Swati, Burke, Terrence R, Shoelson, Steven E
Published in Biochemistry (Easton) (20.10.1992)
Published in Biochemistry (Easton) (20.10.1992)
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