Heterometallic Molecular Architectures Based on Fluorinated β-Diketone Ligands
Saloutin, Viktor I, Edilova, Yulia O, Kudyakova, Yulia S, Burgart, Yanina V, Bazhin, Denis N
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Published in Molecules (Basel, Switzerland) (15.11.2022)
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Conjugates of Tacrine and Salicylic Acid Derivatives as New Promising Multitarget Agents for Alzheimer's Disease
Makhaeva, Galina F, Kovaleva, Nadezhda V, Rudakova, Elena V, Boltneva, Natalia P, Grishchenko, Maria V, Lushchekina, Sofya V, Astakhova, Tatiana Y, Serebryakova, Olga G, Timokhina, Elena N, Zhilina, Ekaterina F, Shchegolkov, Evgeny V, Ulitko, Mariya V, Radchenko, Eugene V, Palyulin, Vladimir A, Burgart, Yanina V, Saloutin, Victor I, Bachurin, Sergey O, Richardson, Rudy J
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Published in International journal of molecular sciences (24.01.2023)
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Powerful Potential of Polyfluoroalkyl-Containing 4-Arylhydrazinylidenepyrazol-3-ones for Pharmaceuticals
Burgart, Yanina V, Elkina, Natalia A, Shchegolkov, Evgeny V, Krasnykh, Olga P, Makhaeva, Galina F, Triandafilova, Galina A, Solodnikov, Sergey Yu, Boltneva, Natalia P, Rudakova, Elena V, Kovaleva, Nadezhda V, Serebryakova, Olga G, Ulitko, Mariya V, Borisevich, Sophia S, Gerasimova, Natalia A, Evstigneeva, Natalia P, Kozlov, Sergey A, Korolkova, Yuliya V, Minin, Artem S, Belousova, Anna V, Mozhaitsev, Evgenii S, Klabukov, Artem M, Saloutin, Victor I
Published in Molecules (Basel, Switzerland) (21.12.2022)
Published in Molecules (Basel, Switzerland) (21.12.2022)
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Synthesis of Mono- and Polyazole Hybrids Based on Polyfluoroflavones
Panova, Mariya A, Shcherbakov, Konstantin V, Zhilina, Ekaterina F, Burgart, Yanina V, Saloutin, Victor I
Published in Molecules (Basel, Switzerland) (15.01.2023)
Published in Molecules (Basel, Switzerland) (15.01.2023)
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Multicomponent Domino Cyclization of Ethyl Trifluoropyruvate with Methyl Ketones and Amino Alcohols as A New Way to γ-Lactam Annulated Oxazacycles
Goryaeva, Marina V, Fefelova, Olesya A, Burgart, Yanina V, Ezhikova, Marina A, Kodess, Mikhail I, Slepukhin, Pavel A, Gaviko, Vasily S, Saloutin, Victor I
Published in Molecules (Basel, Switzerland) (20.02.2023)
Published in Molecules (Basel, Switzerland) (20.02.2023)
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Synthesis of 4-Aminopyrazol-5-ols as Edaravone Analogs and Their Antioxidant Activity
Burgart, Yanina V, Makhaeva, Galina F, Krasnykh, Olga P, Borisevich, Sophia S, Agafonova, Natalia A, Kovaleva, Nadezhda V, Boltneva, Natalia P, Rudakova, Elena V, Shchegolkov, Evgeny V, Triandafilova, Galina A, Gazizov, Denis A, Serebryakova, Olga G, Ulitko, Maria V, Khursan, Sergey L, Saloutin, Victor I, Richardson, Rudy J
Published in Molecules (Basel, Switzerland) (01.11.2022)
Published in Molecules (Basel, Switzerland) (01.11.2022)
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Cholinesterase and carboxylesterase inhibitors as pharmacological agents
Makhaeva, G. F., Rudakova, E. V., Kovaleva, N. V., Lushchekina, S. V., Boltneva, N. P., Proshin, A. N., Shchegolkov, E. V., Burgart, Ya. V., Saloutin, V. I.
Published in Russian chemical bulletin (01.05.2019)
Published in Russian chemical bulletin (01.05.2019)
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Journal Article
Conjugates of tacrine with aminomethylidene derivatives of ethyl acetoacetate as promising agents for the treatment of Alzheimer’s disease
Grishchenko, M. V., Makhaeva, G. F., Burgart, Ya. V., Boltneva, N. P., Rudakova, E. V., Zhilina, E. F., Shchegolkov, E. V., Kovaleva, N. V., Serebryakova, O. G., Saloutin, V. I., Charushin, V. N.
Published in Russian chemical bulletin (01.12.2023)
Published in Russian chemical bulletin (01.12.2023)
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Synthesis and biological activity of 2-sulfonarylhydrazinylidene 1,3-diketones and their pyrazole derivatives
Khudina, O. G., Elkina, N. A., Burgart, Ya. V., Ezhikova, M. A., Kodess, M. I., Esaulkova, Ya. L., Zarubaev, V. V., Shtro, A. A., Triandafilova, G. A., Krasnykh, O. P., Malysheva, K. O., Gerasimova, N. A., Evstigneeva, N. P., Saloutin, V. I.
Published in Russian chemical bulletin (01.12.2022)
Published in Russian chemical bulletin (01.12.2022)
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Journal Article
Conjugates of Tacrine with Aminomethylidene-Substituted Malonates: Synthesis and Biological Evaluation
Grishchenko, M. V., Elkina, N. A., Makhaeva, G. F., Burgart, Ya. V., Boltneva, N. P., Rudakova, E. V., Shchegolkov, E. V., Kovaleva, N. V., Serebryakova, O. G., Saloutin, V. I.
Published in Russian journal of general chemistry (01.11.2022)
Published in Russian journal of general chemistry (01.11.2022)
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Journal Article
Synthesis of new efficient and selective carboxylesterase inhibitors based on adamantyl and citronellyl 4,4,4-trifluoro-2-arylhydrazonylidene-3-oxobutanoates
Elkina, N. A., Shchegolkov, E. V., Burgart, Ya. V., Saloutin, V. I., Boltneva, N. P., Serebryakova, O. G., Lushchekina, S. V., Makhaeva, G. F.
Published in Russian chemical bulletin (01.03.2021)
Published in Russian chemical bulletin (01.03.2021)
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Journal Article
Polyfluorinated salicylic acid derivatives as analogs of known drugs: Synthesis, molecular docking and biological evaluation
Shchegol'kov, E.V., Shchur, I.V., Burgart, Ya.V., Saloutin, V.I., Trefilova, A.N., Ljushina, G.A., Solodnikov, S.Yu, Markova, L.N., Maslova, V.V., Krasnykh, O.P., Borisevich, S.S., Khursan, S.L.
Published in Bioorganic & medicinal chemistry (01.01.2017)
Published in Bioorganic & medicinal chemistry (01.01.2017)
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Journal Article
3-(2-Arylhydrazono)-1,1,1-trifluro-3-(phenylsulfonyl)propan-2-ones as selective carboxylesterase inhibitors
Shchegolkov, E. V., Boltneva, N. P., Burgart, Ya. V., Lushchekina, S. V., Serebryakova, O. G., Elkina, N. A., Rudakova, E. V., Perminova, A. N., Makhaeva, G. F., Saloutin, V. I.
Published in Russian chemical bulletin (2022)
Published in Russian chemical bulletin (2022)
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Journal Article
New Multifunctional Agents for Potential Alzheimer's Disease Treatment Based on Tacrine Conjugates with 2-Arylhydrazinylidene-1,3-Diketones
Elkina, Natalia A, Grishchenko, Maria V, Shchegolkov, Evgeny V, Makhaeva, Galina F, Kovaleva, Nadezhda V, Rudakova, Elena V, Boltneva, Natalia P, Lushchekina, Sofya V, Astakhova, Tatiana Y, Radchenko, Eugene V, Palyulin, Vladimir A, Zhilina, Ekaterina F, Perminova, Anastasiya N, Lapshin, Luka S, Burgart, Yanina V, Saloutin, Victor I, Richardson, Rudy J
Published in Biomolecules (Basel, Switzerland) (24.10.2022)
Published in Biomolecules (Basel, Switzerland) (24.10.2022)
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