Cell panel profiling of pre-clinical and clinical anti-cancer agents reveals conserved therapeutic clusters and differentiates the mechanism of action of different PI3K/mTOR, Aurora kinase and EZH2 inhibitors
Uitdehaag, J.C.M, De Roos, J.A.D.M, Prinsen, M.B.W, Willemsen-Seegers, N, De Vetter, J.R.F, Dylus, J, Van Doornmalen, A.M, Kooijman, J, Sawa, M, Van Gerwen, S.J.C, De Man, J, Buijsman, R.C, Zaman, G.J.R
Published in European journal of cancer (1990) (01.12.2016)
Published in European journal of cancer (1990) (01.12.2016)
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Journal Article
Ruthenium-Catalyzed Olefin Metathesis in Ionic Liquids
Buijsman, Rogier C, van Vuuren, Elizabeth, Sterrenburg, Jan Gerard
Published in Organic letters (15.11.2001)
Published in Organic letters (15.11.2001)
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Journal Article
Synthetic heparin derivatives as new anticoagulant drugs
de Kort, Martin, Buijsman, Rogier C., van Boeckel, Constant A.A.
Published in Drug discovery today (01.06.2005)
Published in Drug discovery today (01.06.2005)
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Journal Article
PO-495 Prediction of chemotherapy sensitivity on ascites of ovarian cancer patients
Ouden, JE Den, Zaman, GJR, Dylus, J, Buijsman, RC, Massuger, LFAG, Altena, AM Van
Published in ESMO open (01.07.2018)
Published in ESMO open (01.07.2018)
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Journal Article
PO-484 Development of a two-step screening-and-confirmation approach to efficiently identify synergistic drug combinations with the PARP inhibitor niraparib
Prinsen, MBW, Vetter, JRF De, Dylus, J, Roos, JADMDe, Gerwen, SJC Van, Buijsman, RC, UItdehaag, JCM
Published in ESMO open (01.07.2018)
Published in ESMO open (01.07.2018)
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Journal Article
PO-456 Cell line panel profiling of all clinically approved kinase inhibitors for cancer treatment
Kooijman, JJ, Uitdehaag, JCM, Roos, JADMDe, Vetter, JRF De, Prinsen, MBW, Dylus, J, Man, J De, Gerwen, SJC Van, Buijsman, RC, Zaman, GJR
Published in ESMO open (01.07.2018)
Published in ESMO open (01.07.2018)
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Journal Article
Development of a novel ionic support and its application in the ionic liquid phase assisted synthesis of a potent antithrombotic
de Kort, Martin, Tuin, Adriaan W., Kuiper, Suzanne, Overkleeft, Hermen S., van der Marel, Gijs A., Buijsman, Rogier C.
Published in Tetrahedron letters (01.03.2004)
Published in Tetrahedron letters (01.03.2004)
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Journal Article
Non-Steroidal Steroid Receptor Modulators
Buijsman, Rogier C, Hermkens, Pedro H H, van Rijn, Rachel D, Stock, H Thijs, Teerhuis, N Miranda
Published in Current medicinal chemistry (01.01.2005)
Published in Current medicinal chemistry (01.01.2005)
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Journal Article
Synthesis and inhibitory effect of a trisubstrate transition state analogue for UDP glucuronosyltransferases
Timmers, C.M., Dekker, M., Buijsman, R.C., van der Marel, G.A., Ethell, B., Anderson, G., Burchell, B., Mulder, G.J., van Boom, J.H.
Published in Bioorganic & medicinal chemistry letters (17.06.1997)
Published in Bioorganic & medicinal chemistry letters (17.06.1997)
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Journal Article
Design and synthesis of a possible mimic of a thrombin-binding DNA aptamer
Buijsman, Rogier C., Schipperijn, Jeroen W.J., Kuyl-Yeheskiely, Esther, van der Marel, Gijs A., van Boeckel, Constant A.A., van Boom, Jacques H.
Published in Bioorganic & medicinal chemistry letters (05.08.1997)
Published in Bioorganic & medicinal chemistry letters (05.08.1997)
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